{"id":7458,"date":"2024-08-06T19:58:27","date_gmt":"2024-08-06T19:58:27","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=7458"},"modified":"2024-08-06T19:58:27","modified_gmt":"2024-08-06T19:58:27","slug":"jinlu","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/tr\/jinlu\/","title":{"rendered":"Jinlu Eri\u011finden Bir Alfa Glukozidaz \u0130nhibit\u00f6r\u00fcn\u00fcn Ekstraksiyonu, Zenginle\u015ftirilmesi ve Aktivite \u00c7al\u0131\u015fmas\u0131"},"content":{"rendered":"<p>Jinlu Eri\u011finden Bir Alfa Glukozidaz \u0130nhibit\u00f6r\u00fcn\u00fcn Ekstraksiyonu, Zenginle\u015ftirilmesi ve Aktivite \u00c7al\u0131\u015fmas\u0131<br \/>\n\u03b1 - glukozidaz (AG) diyabetle yak\u0131ndan ili\u015fkili bir enzimdir. Karbonhidratlar\u0131 v\u00fccutta insan v\u00fccudu taraf\u0131ndan emilebilen ve kullan\u0131labilen glikoz, fruktoz ve galaktoza metabolize edebilir. \u03b1 - glukozidaz inhibit\u00f6r\u00fc (AGI), AG ve \u015feker kombinasyonunu bloke edebilir ve AG'nin aktivitesini rekabet\u00e7i bir \u015fekilde inhibe ederek a\u00e7l\u0131k kan \u015fekerini d\u00fc\u015f\u00fcrebilir. Son y\u0131llarda, diyabetli hastalar\u0131n artmas\u0131yla birlikte, \u00c7in ve Tibet ila\u00e7lar\u0131n\u0131n etkili bile\u015fenleri diyabet tedavisinin klinik uygulamas\u0131nda giderek artm\u0131\u015ft\u0131r. Do\u011fal \u03b1 - glukozidaz inhibit\u00f6rleri, istikrarl\u0131 etkinlik, g\u00fcvenlik, k\u00fc\u00e7\u00fck yan etkiler vb. avantajlara sahiptir ve t\u0131p ara\u015ft\u0131rma alan\u0131nda s\u0131cak bir nokta haline gelmektedir.<br \/>\nPotentilla fruticosa L., Rosaceae familyas\u0131na ve Potentilla cinsine ait, \u00e7o\u011funlukla Qinghai Tibet Platosu'nun y\u00fcksek rak\u0131ml\u0131 b\u00f6lgelerinde da\u011f\u0131lm\u0131\u015f, yaprak d\u00f6ken bir \u00e7al\u0131 bitkisidir. Jin Lu Mei'nin k\u00f6kleri, g\u00f6vdeleri, yapraklar\u0131, \u00e7i\u00e7ekleri ve dallar\u0131 g\u00fc\u00e7l\u00fc farmakolojik aktiviteye sahiptir. Yapraklar yayg\u0131n olarak g\u0131da ve kozmetikte katk\u0131 maddesi olarak kullan\u0131l\u0131r ve k\u00f6k ve g\u00f6vde \u00f6zleri, Ci Wu Jia'dan daha g\u00fc\u00e7l\u00fc bir etkiye sahip g\u00fc\u00e7l\u00fc ba\u011f\u0131\u015f\u0131kl\u0131k d\u00fczenleyici \u00f6zelliklere sahiptir; Dal\u0131n \u00f6z\u00fc yenilebilir ve in vitro deneyler, kandaki kolesterol ve kan \u015fekeri seviyelerini d\u00fc\u015f\u00fcrmede iyi bir aktiviteye sahip oldu\u011funu g\u00f6stermi\u015ftir. Ara\u015ft\u0131rma grubumuz taraf\u0131ndan Primulaceae'nin kimyasal bile\u015fimi \u00fczerine yap\u0131lan \u00f6nceki \u00e7al\u0131\u015fmalar, flavonoid bile\u015fik kuersetin-7-O - \u03b2 - D-glukuronidin Primulaceae'de ilk kez izole edildi\u011fini ve alfa glukozidaz inhibit\u00f6r aktivitesine sahip oldu\u011funu g\u00f6stermi\u015ftir.<br \/>\nBitki flavonoidlerinin ay\u0131rma ve safla\u015ft\u0131rma y\u00f6ntemleri temel olarak re\u00e7ine adsorpsiyonu, y\u00fcksek performansl\u0131 s\u0131v\u0131 kromatografisi vb. i\u00e7erir. Re\u00e7ine adsorpsiyon y\u00f6ntemi, geni\u015f y\u00fczey alan\u0131, b\u00fcy\u00fck adsorpsiyon kapasitesi, iyi se\u00e7icilik, uzun re\u00e7ine hizmet \u00f6mr\u00fc ve d\u00fc\u015f\u00fck i\u015fletme maliyeti avantajlar\u0131 nedeniyle flavonoidlerin zenginle\u015ftirilmesi i\u00e7in yayg\u0131n olarak kullan\u0131lmaktad\u0131r. Bu \u00e7al\u0131\u015fmada, Prunus mume'da quercetin-7-O - \u03b2 - D-glukuronid bile\u015fi\u011finin AG aktivitesini zenginle\u015ftirmek ve inhibe etmek i\u00e7in makro g\u00f6zenekli adsorpsiyon re\u00e7inesi (AB-8) y\u00f6ntemi kullan\u0131lm\u0131\u015f ve Prunus mume'da do\u011fal \u03b1 - glukozidaz inhibit\u00f6rlerinin kapsaml\u0131 geli\u015fimi ve kullan\u0131m\u0131 i\u00e7in teorik bir temel sa\u011flanm\u0131\u015ft\u0131r.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7459\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-36.jpg\" alt=\"\" width=\"402\" height=\"132\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7460\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-32.jpg\" alt=\"\" width=\"408\" height=\"174\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7461\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-243.png\" alt=\"\" width=\"690\" height=\"677\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7462\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-223.png\" alt=\"\" width=\"690\" height=\"271\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7463\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-17.jpg\" alt=\"\" width=\"1182\" height=\"505\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-17.jpg 1182w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-17-768x328.jpg 768w\" sizes=\"(max-width: 1182px) 100vw, 1182px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7464\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-17.jpg\" alt=\"\" width=\"688\" height=\"498\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7465\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-168.png\" alt=\"\" width=\"690\" height=\"267\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7466\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-151.png\" alt=\"\" width=\"690\" height=\"305\" \/><br \/>\nBu makale Tibet ilac\u0131 Jin Lu Mei'yi ara\u015ft\u0131rma nesnesi olarak ele almakta ve hedef hipoglisemik bile\u015fi\u011fi Jin Lu Mei'den ilk kez y\u00fcksek safl\u0131kta izole etmek i\u00e7in DAC-50 yar\u0131 preparatif y\u00fcksek performansl\u0131 s\u0131v\u0131 kromatografisi ve y\u00fcksek performansl\u0131 s\u0131v\u0131 kromatografisi kullanmaktad\u0131r. Jin Lu Mei'den Quercetin-7-O - \u03b2 - D-glukuronid monomer bile\u015fiklerini ay\u0131rmak i\u00e7in bir y\u00f6ntem olu\u015fturulmu\u015ftur. Jinlu Mei'de bulunan kimyasal bile\u015fenler 75% etanol kullan\u0131larak ekstrakte edilmi\u015ftir. Ekstraksiyon \u00e7\u00f6zeltisi AB-8 kolon kromatografisi kullan\u0131larak 0, 10%, 20%, 30%, 40% ve 50% su etanol \u00e7\u00f6zeltileri ile ayr\u0131lm\u0131\u015f ve b\u00f6l\u00fcmlere ayr\u0131lm\u0131\u015ft\u0131r. Bile\u015fikler polaritelerine g\u00f6re \u00f6n s\u0131n\u0131fland\u0131rmaya tabi tutuldu ve Jinlumei'nin 20% AB-8 eluentindeki monomer bile\u015fikleri esas olarak izole edildi ve haz\u0131rland\u0131.<br \/>\nBile\u015fi\u011fin yap\u0131sal analizi ile flavonoid bir bile\u015fik oldu\u011fu bulunmu\u015ftur. Bu bile\u015fi\u011fin aktivite tespiti ve inhibit\u00f6r tipi tan\u0131mlama sonu\u00e7lar\u0131, quercetin-7-O - \u03b2 - D-glukuronidin 94.67%'lik en y\u00fcksek inhibisyon oran\u0131 ile rekabet\u00e7i bir inhibit\u00f6r oldu\u011funu g\u00f6stermi\u015ftir. Bu, bile\u015fi\u011fin AG'ye ba\u011flanmada g\u00fc\u00e7l\u00fc bir rekabet g\u00fcc\u00fcne sahip oldu\u011funu ve AG'nin \u015fekerlere ba\u011flanmas\u0131n\u0131 b\u00fcy\u00fck \u00f6l\u00e7\u00fcde azaltt\u0131\u011f\u0131n\u0131 g\u00f6sterir ki bu da \u00f6nceki ara\u015ft\u0131rma sonu\u00e7lar\u0131yla tutarl\u0131d\u0131r. Bile\u015fik ve AG aras\u0131ndaki olas\u0131 ba\u011flanma modeli bilgisayar destekli molek\u00fcler yerle\u015ftirme y\u00f6ntemi kullan\u0131larak incelenmi\u015f ve olas\u0131 etki mekanizmas\u0131 ara\u015ft\u0131r\u0131lm\u0131\u015ft\u0131r. Bile\u015fi\u011fin flavonoid ana \u00e7ekirde\u011finin \u00fc\u00e7 benzen halkas\u0131, AG protein kal\u0131nt\u0131lar\u0131 ile \u03c0 - \u03c0 konjuge ba\u011flar\u0131, \u03c0 - alkil ba\u011flar\u0131, \u03c0 - \u03c3 konjuge ba\u011flar\u0131, hidrojen ba\u011flar\u0131 vb. yoluyla kararl\u0131 bir ba\u011flanma durumu olu\u015fturmu\u015f ve b\u00f6ylece a\u00e7l\u0131k kan glikozunu azaltm\u0131\u015ft\u0131r. Bu bile\u015fik, Jinlumei'nin diyabet tedavisi i\u00e7in ila\u00e7 geli\u015ftirme potansiyeline sahip oldu\u011funu g\u00f6steren ve Jinlumei'nin hipoglisemik farmas\u00f6tik bile\u015fenlerinin ara\u015ft\u0131r\u0131lmas\u0131 ve geli\u015ftirilmesi i\u00e7in bilimsel teorik temel sa\u011flayan iyi bir \u03b1 - glukozidaz inhibit\u00f6r aktivitesine sahiptir.<\/p>","protected":false},"excerpt":{"rendered":"<p>Extraction, Enrichment, and Activity Study of an Alpha Glucosidase Inhibitor from Jinlu Plum \u03b1 &#8211; glucosidase (AG) is an enzyme closely related to diabetes. It can metabolize carbohydrates into glucose, fructose and galactose that can be absorbed and utilized by the human body in the body. \u03b1 &#8211; glucosidase inhibitor (AGI) can block the combination [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Extraction, Enrichment, and Activity Study of an Alpha Glucosidase Inhibitor from Jinlu Plum - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/tr\/jinlu\/\" \/>\n<meta property=\"og:locale\" content=\"tr_TR\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Extraction, Enrichment, and Activity Study of an Alpha Glucosidase Inhibitor from Jinlu Plum - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Extraction, Enrichment, and Activity Study of an Alpha Glucosidase Inhibitor from Jinlu Plum \u03b1 &#8211; glucosidase (AG) is an enzyme closely related to diabetes. 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