{"id":7370,"date":"2024-08-06T19:36:02","date_gmt":"2024-08-06T19:36:02","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=7370"},"modified":"2024-08-06T19:36:02","modified_gmt":"2024-08-06T19:36:02","slug":"proliferation-migration","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/tr\/cogalma-goc\/","title":{"rendered":"Resveratrol\u00fcn endometriyal kanser HEC-1A h\u00fccrelerinin proliferasyonu, migrasyonu ve invazyonu \u00fczerindeki etkisi"},"content":{"rendered":"<p>Resveratrol\u00fcn endometriyal kanser HEC-1A h\u00fccrelerinin proliferasyonu, migrasyonu ve invazyonu \u00fczerindeki etkisi<br \/>\nEndometrial karsinom (EC), kad\u0131n \u00fcreme sisteminde meme kanseri, akci\u011fer kanseri ve kolorektal kanserden sonra en s\u0131k g\u00f6r\u00fclen t\u00fcm\u00f6rd\u00fcr. D\u00fcnyada her y\u0131l yakla\u015f\u0131k 380000 yeni endometriyal kanser vakas\u0131 g\u00f6r\u00fclmekte ve her y\u0131l yakla\u015f\u0131k 89000 ki\u015fi endometriyal kanser nedeniyle hayat\u0131n\u0131 kaybetmekte olup, g\u00f6r\u00fclme oran\u0131 y\u0131ldan y\u0131la artmaktad\u0131r. \u015eu anda, endometriyal kanserin spesifik patogenezi hala belirsizdir ve risk fakt\u00f6rleri obezite, metabolik sendrom, hiperlipidemi, diyabet, polikistik over sendromu ve y\u00fcksek \u00f6strojen durumunun neden oldu\u011fu endometriyal hiperplaziye yol a\u00e7an di\u011fer hastal\u0131klarla ili\u015fkilidir. Erken endometriyal kanser tek ba\u015f\u0131na cerrahi veya adjuvan kemoradyoterapi ile kombine cerrahi ile tedavi edilebilir ve 5 y\u0131ll\u0131k genel sa\u011fkal\u0131m oran\u0131 74% ila 91% aras\u0131ndad\u0131r. \u0130lerlemi\u015f veya tekrarlayan endometriyal kanser tan\u0131s\u0131 konan hastalar\u0131n prognozu k\u00f6t\u00fcd\u00fcr ve sa\u011fkal\u0131m oran\u0131 d\u00fc\u015f\u00fckt\u00fcr; be\u015f y\u0131ll\u0131k genel sa\u011fkal\u0131m oran\u0131 yakla\u015f\u0131k 15%'dir. Cerrahi, radyoterapi, kemoterapi ve hedefe y\u00f6nelik tedavi gibi geleneksel tedaviler pahal\u0131d\u0131r ve ciddi yan etkilere e\u011filimlidir. T\u00fcm\u00f6r n\u00fcks\u00fc ve metastaz\u0131n\u0131n yan\u0131 s\u0131ra kemoterapi direnci gibi sorunlar\u0131n ortaya \u00e7\u0131kmas\u0131yla birlikte, EC'yi tedavi etmek i\u00e7in kolay eri\u015filebilir, d\u00fc\u015f\u00fck yan etkili ve d\u00fc\u015f\u00fck maliyetli alternatif ila\u00e7lar\u0131n bulunmas\u0131na acil ihtiya\u00e7 duyulmaktad\u0131r. Bu nedenle, t\u00fcm\u00f6r h\u00fccresi proliferasyonu, migrasyonu ve invazyonunun i\u00e7sel mekanizmalar\u0131n\u0131n anla\u015f\u0131lmas\u0131, AK hastalar\u0131n\u0131n tedavisinde yeni y\u00f6ntemlerin ke\u015ffedilmesi i\u00e7in b\u00fcy\u00fck de\u011fer ta\u015f\u0131maktad\u0131r.<\/p>\n<p>Kimyasal form\u00fcl\u00fc C14H12O4 olan Piceatannol (PIC), \u00e7ark\u0131felek meyvesi, \u00e7ark\u0131felek \u00e7i\u00e7e\u011fi, beyaz \u00e7ay ve Japon kaplan \u00e7i\u00e7e\u011fi gibi bitkilerde yayg\u0131n olarak bulunan do\u011fal bir polifenolik bile\u015fiktir. Ara\u015ft\u0131rmalar PIC'in resveratrol benzeri anti-t\u00fcm\u00f6r, anti-inflamatuar, antioksidan ve ba\u011f\u0131\u015f\u0131kl\u0131k d\u00fczenleyici etkilere sahip oldu\u011funu ve \u00e7ok hedefli do\u011fas\u0131 nedeniyle kanser \u00f6nleme ve tedavisinde \u00f6nemli bir rol oynad\u0131\u011f\u0131n\u0131 g\u00f6stermi\u015ftir. Baz\u0131 \u00e7al\u0131\u015fmalar PIC'in kemopreventif aktiviteye sahip oldu\u011funu ve prostat kanseri, kolorektal kanser, meme kanseri, akci\u011fer kanseri, melanom, lenfoma vb. migrasyon ve invazyonunu engelleyebildi\u011fini g\u00f6stermi\u015ftir. Wnt\/\u03b2 - catenin sinyal yolunun anormal aktivasyonu, \u00e7e\u015fitli k\u00f6t\u00fc huylu t\u00fcm\u00f6rlerin olu\u015fumunu ve geli\u015fimini te\u015fvik edebilir ve h\u00fccre \u00e7o\u011falmas\u0131n\u0131 ve farkl\u0131la\u015fmas\u0131n\u0131 d\u00fczenleyebilir. Ara\u015ft\u0131rmalar, PIC'in Wnt\/\u03b2 - catenin yolunun bir inhibit\u00f6r\u00fc ve miyelom h\u00fccrelerinde apoptozun bir ind\u00fckleyicisi olarak da hareket edebilece\u011fini bulmu\u015ftur. \u015eu anda, PIC'in endometriyal kanser \u00fczerindeki anti-t\u00fcm\u00f6r etkisi hakk\u0131nda hi\u00e7bir ara\u015ft\u0131rma raporu bulunmamaktad\u0131r ve endometriyal kanser h\u00fccrelerinin etkisine arac\u0131l\u0131k etme mekanizmas\u0131 hala belirsizdir. Bu deney, endometriyal kanser h\u00fccrelerinin proliferasyonu, migrasyonu ve invazyonu \u00fczerindeki etkilerini g\u00f6zlemleyerek PIC'in \u00f6n anti-t\u00fcm\u00f6r mekanizmas\u0131n\u0131 ke\u015ffetmeyi ve endometriyal kanser tedavisinde yeni stratejilerin ara\u015ft\u0131r\u0131lmas\u0131 i\u00e7in teorik ve deneysel temel sa\u011flamay\u0131 ama\u00e7lamaktad\u0131r.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7371\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-298.png\" alt=\"\" width=\"365\" height=\"240\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7372\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-250.png\" alt=\"\" width=\"784\" height=\"341\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-250.png 784w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-250-768x334.png 768w\" sizes=\"(max-width: 784px) 100vw, 784px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7373\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-235.png\" alt=\"\" width=\"784\" height=\"313\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-235.png 784w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-235-768x307.png 768w\" sizes=\"(max-width: 784px) 100vw, 784px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7374\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-215.png\" alt=\"\" width=\"783\" height=\"382\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-215.png 783w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-215-768x375.png 768w\" sizes=\"(max-width: 783px) 100vw, 783px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7375\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-194.png\" alt=\"\" width=\"786\" height=\"269\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-194.png 786w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-194-768x263.png 768w\" sizes=\"(max-width: 786px) 100vw, 786px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7376\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-177.png\" alt=\"\" width=\"780\" height=\"354\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-177.png 780w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-177-768x349.png 768w\" sizes=\"(max-width: 780px) 100vw, 780px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7377\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-162.png\" alt=\"\" width=\"784\" height=\"186\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-162.png 784w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-162-768x182.png 768w\" sizes=\"(max-width: 784px) 100vw, 784px\" \/><br \/>\nEpitelyal mezenkimal ge\u00e7i\u015f (EMT), t\u00fcm\u00f6r metastaz\u0131nda \u00e7ok \u00f6nemli bir s\u00fcre\u00e7tir ve h\u00fccrelere g\u00fc\u00e7l\u00fc g\u00f6\u00e7 ve invaziv embriyonik programlar kazand\u0131r\u0131r. Normal ko\u015fullar alt\u0131nda EMT yara iyile\u015fmesinde \u00f6nemli bir rol oynarken, anormal durumlarda t\u00fcm\u00f6r metastaz\u0131n\u0131 te\u015fvik eder. Ara\u015ft\u0131rmalar EMT'nin endometriyal kanser t\u00fcm\u00f6r h\u00fccrelerinin olu\u015fumu, metastaz\u0131, anti apoptoz ve invazyon s\u00fcre\u00e7lerinde rol oynad\u0131\u011f\u0131n\u0131 do\u011frulam\u0131\u015ft\u0131r. Ara\u015ft\u0131rmalar, ERK\/MAPK sinyal yolunun ve PI3K\/AKT\/mTOR sinyal yolunun EC'de anormal \u015fekilde aktive oldu\u011funu g\u00f6stermi\u015ftir. Normalden maligne h\u00fccre d\u00f6n\u00fc\u015f\u00fcm\u00fc s\u00fcrecinde, EMT PI3K\/AKT\/mTOR sinyal yola\u011f\u0131 taraf\u0131ndan d\u00fczenlenirken, Wnt sinyal yola\u011f\u0131 t\u00fcm\u00f6r h\u00fccrelerinde EMT'yi ind\u00fckler ve b\u00f6ylece t\u00fcm\u00f6r invazyonu ve metastaz\u0131n\u0131 etkiler. Bu \u00e7al\u0131\u015fmada, PIC'in endometriyal kanser HEC-1A h\u00fccrelerinde epitel benzeri belirte\u00e7 E-cdaherin'in ekspresyon seviyesini y\u00fckseltebildi\u011fini ve Wnt sinyal yola\u011f\u0131ndaki transkripsiyon inhibit\u00f6r fakt\u00f6r Slug ve anahtar efekt\u00f6r molek\u00fcller \u03b2 - catenin ve CD44 proteinlerinin ekspresyon seviyelerini d\u00fc\u015f\u00fcrebildi\u011fini bulduk. Sonu\u00e7lar, PIC'in endometriyal kanser h\u00fccrelerinde EMT d\u00f6n\u00fc\u015f\u00fcm\u00fcn\u00fc ind\u00fcklemek i\u00e7in Wnt sinyal yolunu inhibe edebilece\u011fini ve b\u00f6ylece HEC-1A h\u00fccrelerinin g\u00f6\u00e7\u00fcn\u00fc ve istilas\u0131n\u0131 bask\u0131layabilece\u011fini g\u00f6stermektedir.<br \/>\nAra\u015ft\u0131rma raporlar\u0131, PIC'in t\u00fcm\u00f6rleri geriletme, apoptozu ind\u00fckleme ve anjiyogenez, invazyon, migrasyon ve metastaz\u0131 inhibe etme potansiyeline sahip oldu\u011funu g\u00f6stermektedir. \u00d6nceki ara\u015ft\u0131rmam\u0131z, PIC'in Wnt\/\u03b2 - catenin sinyal yolunu inhibe ederek \u00fc\u00e7l\u00fc negatif meme kanseri h\u00fccre hatt\u0131 MDA-MB-468'in proliferasyonunu inhibe edebildi\u011fini, h\u00fccre d\u00f6ng\u00fcs\u00fcn\u00fc bloke edebildi\u011fini ve apoptozu ind\u00fckleyebildi\u011fini ve iyi bir anti \u00fc\u00e7l\u00fc negatif meme kanseri etkisine sahip oldu\u011funu buldu. Ba\u015fka bir \u00e7al\u0131\u015fma, PIC'in Hras kaynakl\u0131 AKR fosforilasyonunu, MMP-2 ve fosfatidilinositol 3-kinaz (PI3K) aktivitelerini inhibe ederek ve fosfatidilinositol (3,4,5) - trifosfat (PI3K) ekspresyonunu a\u015fa\u011f\u0131 d\u00fczenleyerek meme kanseri MCF-10A h\u00fccrelerinin metastaz\u0131n\u0131 ve invazyonunu inhibe etti\u011fini ve anti meme kanseri rol\u00fcn\u00fc oynad\u0131\u011f\u0131n\u0131 g\u00f6stermi\u015ftir. Bu \u00e7al\u0131\u015fman\u0131n in vitro sonu\u00e7lar\u0131, PIC'in endometriyal kanser h\u00fccreleri HEC-1A'n\u0131n proliferasyonu, migrasyonu ve invazyonu \u00fczerinde \u00f6nemli bir ila\u00e7 konsantrasyonuna ba\u011fl\u0131 inhibit\u00f6r etkiye sahip oldu\u011funu bulmu\u015ftur. MAPK sinyal yolunun aktivasyonu, t\u00fcm\u00f6rlerin olu\u015fumu ve geli\u015fimi ile ilgilidir ve h\u00fccre b\u00fcy\u00fcmesi, farkl\u0131la\u015fmas\u0131, hayatta kalmas\u0131 ve \u00f6l\u00fcm\u00fcn\u00fcn d\u00fczenlenmesinde rol oynar. Erk ve p38MAPK proteinleri, MAPK sinyal yolunun anahtar efekt\u00f6r molek\u00fclleridir. Yan ve arkada\u015flar\u0131, PIC'in MAPK ve AKT sinyal yollar\u0131n\u0131 etkileyerek Erk1\/2 ve Akt proteinlerinin fosforilasyonunu inhibe etti\u011fini ve b\u00f6ylece RANKL kaynakl\u0131 osteoklast olu\u015fumunu ve kemik rezorpsiyonunu bask\u0131lad\u0131\u011f\u0131n\u0131 bulmu\u015flard\u0131r. Molek\u00fcler d\u00fczeyde, bu \u00e7al\u0131\u015fma ayr\u0131ca PIC'in HEC-1A h\u00fccrelerinde proliferasyonla ilgili proteinler Akt, Erk1\/2 ve p38MAPK'nin fosforilasyonunu inhibe ederek endometriyal kanser h\u00fccrelerinin proliferasyonunu, migrasyonunu ve invazyonunu etkili bir \u015fekilde bask\u0131layabildi\u011fini g\u00f6stermi\u015ftir.<br \/>\n\u00d6zetle, bu \u00e7al\u0131\u015fman\u0131n sonu\u00e7lar\u0131 PIC'in HEC-1A endometriyal kanser h\u00fccrelerinin proliferasyonunu etkili bir \u015fekilde inhibe edebilece\u011fini, h\u00fccre apoptozunu ind\u00fckleyebilece\u011fini ve HEC-1A h\u00fccrelerinin g\u00f6\u00e7 ve invazyon yetene\u011fini \u00f6nemli \u00f6l\u00e7\u00fcde azaltabilece\u011fini g\u00f6stermektedir. Mekanizmas\u0131, Akt\/ERK\/MAPK sinyal yola\u011f\u0131nda Akt, Erk1\/2 ve p38MAPK fosforilasyonunun inhibisyonu, invazyon ve migrasyon proteinleri \u03b2 - catenin, CD44 ve Slug ekspresyon seviyelerinin a\u015fa\u011f\u0131 reg\u00fclasyonu ve E-cdaherin protein ekspresyon seviyelerinin yukar\u0131 reg\u00fclasyonu ile ili\u015fkili olabilir. PIC'in endometriyal kanser h\u00fccrelerinin proliferasyonu, migrasyonu ve invazyonu \u00fczerinde inhibe edici etkileri oldu\u011fu \u00f6nceden do\u011frulanm\u0131\u015ft\u0131r. Bununla birlikte, bu deney sadece h\u00fccresel d\u00fczeyde \u00f6n in vitro \u00e7al\u0131\u015fmalar y\u00fcr\u00fctm\u00fc\u015ft\u00fcr ve anti endometriyal kanser etkisinin spesifik molek\u00fcler mekanizmas\u0131n\u0131n in vivo \u00e7al\u0131\u015fmalarla daha fazla a\u00e7\u0131kl\u0131\u011fa kavu\u015fturulmas\u0131 gerekmektedir.<\/p>","protected":false},"excerpt":{"rendered":"<p>The effect of resveratrol on proliferation, migration, and invasion of endometrial cancer HEC-1A cells Endometrial carcinoma (EC) is the most common tumor in the female reproductive tract, second only to breast cancer, lung cancer and colorectal cancer. In the world, there are about 380000 new cases of endometrial cancer every year, and about 89000 people [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>The effect of resveratrol on proliferation, migration, and invasion of endometrial cancer HEC-1A cells - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/tr\/cogalma-goc\/\" \/>\n<meta property=\"og:locale\" content=\"tr_TR\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"The effect of resveratrol on proliferation, migration, and invasion of endometrial cancer HEC-1A cells - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"The effect of resveratrol on proliferation, migration, and invasion of endometrial cancer HEC-1A cells Endometrial carcinoma (EC) is the most common tumor in the female reproductive tract, second only to breast cancer, lung cancer and colorectal cancer. 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