{"id":5183,"date":"2024-08-04T17:42:52","date_gmt":"2024-08-04T17:42:52","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=5183"},"modified":"2024-08-04T17:42:52","modified_gmt":"2024-08-04T17:42:52","slug":"huperzine","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/tr\/huperzin\/","title":{"rendered":"Simbiyotik yeti\u015ftirme y\u00f6ntemi ile huperzin A'n\u0131n artan zenginle\u015ftirilmesinin te\u015fvik edilmesi \u00fczerine \u00e7al\u0131\u015fma"},"content":{"rendered":"<p>Simbiyotik yeti\u015ftirme y\u00f6ntemi ile huperzin A'n\u0131n artan zenginle\u015ftirilmesinin te\u015fvik edilmesi \u00fczerine \u00e7al\u0131\u015fma<br \/>\nHuperzia serrata (Thunb. ex Murray), Taxaceae familyas\u0131ndan Taxodium cinsine ait bir e\u011frelti otu bitkisidir. Travmatik yaralanmalar\u0131n tedavisi, detoksifikasyon, a\u011fr\u0131 kesici ve \u015fizofreni tedavisinde kullan\u0131lan nadir bir \u00c7in bitkisel ilac\u0131d\u0131r. Y\u0131lan aya\u011f\u0131 k\u00f6knar\u0131 \u015fu anda Alzheimer hastal\u0131\u011f\u0131n\u0131n tedavisi i\u00e7in en iyi ara\u015ft\u0131r\u0131lan ila\u00e7lardan biridir. Aktif bile\u015feni olan huperzin A, myastenia gravis ve Alzheimer hastal\u0131\u011f\u0131n\u0131n tedavisi i\u00e7in etkili, d\u00fc\u015f\u00fck toksisiteli, geri d\u00f6n\u00fc\u015f\u00fcml\u00fc ve olduk\u00e7a se\u00e7ici bir asetilkolinesteraz (AChE) inhibit\u00f6r\u00fcd\u00fcr. Dikkat, uyan\u0131kl\u0131k, konsantrasyon ve haf\u0131za ile ilgili bir merkezi sinir n\u00f6rotransmitteri olan asetilkolinin etkisini art\u0131rabilir. 1982 y\u0131l\u0131nda huperzin A, y\u0131lan ayakl\u0131 k\u00f6knardan ba\u015far\u0131yla izole edilmi\u015f ve \"Umut Y\u0131ld\u0131z\u0131\" olarak kabul edilmi\u015ftir. Bir ara\u015ft\u0131rmaya g\u00f6re, 2025 y\u0131l\u0131na kadar geli\u015fmi\u015f \u00fclkelerde 65 ya\u015f ve \u00fczeri Alzheimer hastalar\u0131n\u0131n say\u0131s\u0131 2018'deki 5,5 milyondan yakla\u015f\u0131k 29%'lik bir art\u0131\u015fla 7,1 milyona ula\u015facak. T\u0131bbi bir at\u0131l\u0131m olmad\u0131\u011f\u0131 takdirde, hastal\u0131\u011fa yakalananlar\u0131n say\u0131s\u0131 2050 y\u0131l\u0131na kadar 5,5 milyondan 13,8 milyona \u00e7\u0131kabilir. Sadece Amerika Birle\u015fik Devletleri'nde, her 100000 ki\u015fiden yakla\u015f\u0131k 14-20'si myastenia gravis hastas\u0131d\u0131r ve toplamda yakla\u015f\u0131k 36000-60000 hasta vard\u0131r ki bu da olduk\u00e7a endi\u015fe verici bir say\u0131d\u0131r. Alzheimer hastal\u0131\u011f\u0131 ve myastenia gravis i\u00e7in \u015fu anda piyasada bulunan ila\u00e7larla ilgili en b\u00fcy\u00fck sorun ila\u00e7 toksisitesi ve direncidir. Mevcut ila\u00e7larla kar\u015f\u0131la\u015ft\u0131r\u0131ld\u0131\u011f\u0131nda, huperzin A iyi g\u00fcvenlikli, daha az yan etkiye sahip ve insan v\u00fccudu taraf\u0131ndan h\u0131zla emilebilen do\u011fal bir bitki \u00f6z\u00fcd\u00fcr. \u0130nhibisyon y\u00f6ntemi, kar\u0131\u015f\u0131k bir rekabet\u00e7i ve rekabet\u00e7i olmayan inhibisyon t\u00fcr\u00fcd\u00fcr ve terap\u00f6tik etki, uzun bir etkili s\u00fcre ile \u00f6nemlidir.<br \/>\nY\u0131lan ayakl\u0131 Cryptomeria t\u00fcm d\u00fcnyaya yay\u0131lm\u0131\u015ft\u0131r, ancak kaynaklar\u0131 \u00e7ok s\u0131n\u0131rl\u0131d\u0131r. S\u0131n\u0131rlay\u0131c\u0131 fakt\u00f6rlerden biri, sporlardan olgunlu\u011fa kadar en az 15 y\u0131l s\u00fcren y\u0131lan ayakl\u0131 Cryptomeria'n\u0131n yava\u015f b\u00fcy\u00fcmesidir. Ve olgunluk a\u015famas\u0131nda, y\u0131lan ayakl\u0131 k\u00f6knar\u0131n boyu sadece 10-30 cm'dir. Ayn\u0131 zamanda, b\u00fcy\u00fcme ortam\u0131n\u0131n \u00e7o\u011falt\u0131lmas\u0131 ve ger\u00e7ek yeti\u015ftirme s\u00fcre\u00e7lerinde te\u015fvik edilmesi zordur. Bu nedenle, yak\u0131n gelecekte y\u0131lan ayakl\u0131 k\u00f6knar yok olma tehdidiyle kar\u015f\u0131 kar\u015f\u0131ya kalacakt\u0131r. Son y\u0131llarda, bu nadir bitki \u00fczerinde, eksplant ve kallus dokular\u0131n\u0131n in vitro yeti\u015ftirilmesi gibi \u00e7ok say\u0131da \u00e7al\u0131\u015fma yap\u0131lm\u0131\u015ft\u0131r. Kan'ichiro Ishiuchi'nin ekibi, H Pinifolia'n\u0131n k\u00f6k ucundan eksplantlar elde etmi\u015f ve steril ortamda 2 d\u00f6ng\u00fc boyunca (her d\u00f6ng\u00fc 7 g\u00fcn) k\u00fclt\u00fcrlenmi\u015ftir. Son olarak, eksplantlar ba\u015far\u0131l\u0131 bir \u015fekilde kallus b\u00fcy\u00fcme ortam\u0131na aktar\u0131ld\u0131. Buna ek olarak, ara\u015ft\u0131rmac\u0131lar Huperzia serrata'n\u0131n k\u00fclt\u00fcr y\u00f6nteminde ortam bile\u015fenlerinin taranmas\u0131 ve k\u00f6k ucu k\u00fclt\u00fcr teknolojisinin ara\u015ft\u0131r\u0131lmas\u0131 gibi \u00e7e\u015fitli iyile\u015ftirmeler yapm\u0131\u015flard\u0131r. Bununla birlikte, doku k\u00fclt\u00fcr\u00fc s\u00fcrecinde eksplantlar\u0131n dezenfeksiyonu ve sterilizasyonu sorunu etkili bir \u015fekilde \u00e7\u00f6z\u00fclememi\u015ftir ve bu da huperzin A'n\u0131n b\u00fcy\u00fck \u00f6l\u00e7ekli \u00fcretimini s\u0131n\u0131rlamaktad\u0131r. Do\u011fal kaynaklar\u0131n k\u0131tl\u0131\u011f\u0131 ve yukar\u0131da belirtilen nedenlerden dolay\u0131, huperzin A i\u00e7eri\u011fini daha d\u00fc\u015f\u00fck bir maliyetle art\u0131rabilecek yeni bir y\u00f6ntem bulmaya acil ihtiya\u00e7 vard\u0131r.<br \/>\nEndofitik mantarlar, bitki k\u00f6k ve yaprak dokular\u0131nda ya\u015fayan bir mantar t\u00fcr\u00fcd\u00fcr. Ara\u015ft\u0131rmalar, endofitik mantarlar\u0131n bitkilerle uzun s\u00fcre simbiyoz halinde geli\u015fmeleri halinde, genetik rekombinasyon yoluyla konuk\u00e7u bitkinin baz\u0131 genlerini elde edebildiklerini ve konuk\u00e7u bitkininkilerle ayn\u0131 olan ikincil metabolitler \u00fcretebildiklerini ortaya koymu\u015ftur. Bu arada endofitik mantarlar, konuk\u00e7u bitkilerin b\u00fcy\u00fcme ve geli\u015fimini desteklemek i\u00e7in hormon da \u00fcretebilir. Bu nedenle, birlikte k\u00fclt\u00fcr sisteminde, endofitik mantarlar elisit\u00f6r olarak kabul edilir, bu da bitki h\u00fccrelerinin belirli bir konsantrasyon aral\u0131\u011f\u0131nda endofitik mantarlarla birlikte k\u00fclt\u00fcrlenebilece\u011fi anlam\u0131na gelir. Birlikte k\u00fclt\u00fcr sisteminde, endofitik mantarlar ve bitki h\u00fccreleri birbirleriyle etkile\u015fime girerek bitkisel \u00fcr\u00fcnlerin birikimini te\u015fvik eder. Ergosterol, mantar h\u00fccre zar\u0131n\u0131n \u00f6nemli bir bile\u015feni ve mantarlar\u0131n karakteristik bir sterol\u00fcd\u00fcr. Mantar biyok\u00fctlesini \u00f6l\u00e7mek i\u00e7in temsili bir g\u00f6sterge olarak kullan\u0131labilir.<br \/>\nBu \u00e7al\u0131\u015fma, \u00c7in g\u00f6knar\u0131n\u0131n kaynak k\u0131tl\u0131\u011f\u0131 nedeniyle yayg\u0131n olarak kullan\u0131lamad\u0131\u011f\u0131 mevcut durumu iyile\u015ftirmek amac\u0131yla \u00c7in g\u00f6knar\u0131nda huperzin A i\u00e7eri\u011fini ekonomik ve uygun bir \u015fekilde art\u0131rmak i\u00e7in yeni bir ortak k\u00fclt\u00fcr sistemi (CCS) sunmaktad\u0131r. <img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5184\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-124.png\" alt=\"\" width=\"754\" height=\"191\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5185\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-110.png\" alt=\"\" width=\"736\" height=\"407\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5186\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-104.png\" alt=\"\" width=\"780\" height=\"221\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-104.png 780w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-104-768x218.png 768w\" sizes=\"(max-width: 780px) 100vw, 780px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5187\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-93.png\" alt=\"\" width=\"744\" height=\"401\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5188\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-85.png\" alt=\"\" width=\"749\" height=\"579\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5189\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-78.png\" alt=\"\" width=\"774\" height=\"142\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-78.png 774w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-78-768x141.png 768w\" sizes=\"(max-width: 774px) 100vw, 774px\" \/><\/p>\n<p>Huperzine A, Alzheimer hastal\u0131\u011f\u0131 ve myastenia gravis tedavisinde kullan\u0131lan bir AChE inhibit\u00f6r\u00fcd\u00fcr. Ana kayna\u011f\u0131 Cryptomeria lanceolata'd\u0131r, ancak Cryptomeria lanceolata'daki Huperzine A i\u00e7eri\u011fi d\u00fc\u015f\u00fckt\u00fcr ve Cryptomeria lanceolata'n\u0131n s\u0131n\u0131rl\u0131 kaynaklar\u0131 farmas\u00f6tik alanda daha fazla geli\u015fmesini s\u0131n\u0131rlamaktad\u0131r. Bitkilerde \u00e7e\u015fitli endofitik mantarlar\u0131n bulundu\u011funu ve bunlar\u0131n uzun s\u00fcreli evrim s\u0131ras\u0131nda konak\u00e7\u0131 bitkilerle karma\u015f\u0131k bir mutualistik ili\u015fki kurdu\u011funu g\u00f6steren \u00e7al\u0131\u015fmalar vard\u0131r. Bir yandan, endofitik mantarlar\u0131n kendi hayatta kalma ihtiya\u00e7lar\u0131n\u0131 kar\u015f\u0131lamak i\u00e7in bitkilerden besin almalar\u0131 gerekir. Di\u011fer yandan endofitik mantarlar, konuk\u00e7u bitkinin savunma sistemine kar\u015f\u0131 koymak i\u00e7in konuk\u00e7u bitkilerle \u00f6zel biyokimyasal ileti\u015fim kurarlar. Konuk\u00e7unun kimyasal sinyallerini tan\u0131yarak veya konuk\u00e7u enzim sistemlerini kullanarak konuk\u00e7uya benzer ikincil metabolitler sentezleyebilirler. Jiang ve arkada\u015flar\u0131, yar\u0131 k\u0131rm\u0131z\u0131 mangrov bitkisi Hibiscus'tan endofitik mantarlar\u0131 izole edip safla\u015ft\u0131rm\u0131\u015f ve kat\u0131 hal fermantasyonu yoluyla konuk\u00e7uyla ayn\u0131 ikincil metabolitleri elde etmi\u015ftir. Tong ve arkada\u015flar\u0131, Cryptomeria serrata'daki endofitik mantar FS4'\u00fcn ikincil metabolitlerini izole edip incelemi\u015f ve be\u015f metabolitinin huperzin A'ya benzer g\u00fc\u00e7l\u00fc inhibit\u00f6r asetilkolinesteraz biyolojik aktivitesi sergiledi\u011fini bulmu\u015ftur.<br \/>\nBu \u00e7al\u0131\u015fmada, yabani y\u0131lanaya\u011f\u0131 bald\u0131ran\u0131n\u0131n evcille\u015ftirme ko\u015fullar\u0131 ve doku k\u00fclt\u00fcr\u00fc ortam\u0131 ko\u015fullar\u0131 \u00fczerinde deneyler yap\u0131lm\u0131\u015ft\u0131r. En uygun k\u00fclt\u00fcr ko\u015fullar\u0131 100 Lux \u0131\u015f\u0131k yo\u011funlu\u011fu, 95% nem, MS s\u0131v\u0131 ortam\u0131, 20.0g\/L s\u00fckroz, 2,4-D5.0mg\/L ve KT1.0mg\/L olarak belirlenmi\u015ftir. CCS'nin dinamik b\u00fcy\u00fcme s\u00fcrecini yans\u0131tmak i\u00e7in huperzine A ve ergosterol olmak \u00fczere iki bile\u015fi\u011fin g\u00f6receli de\u011fi\u015fimleri kullan\u0131lm\u0131\u015ft\u0131r. D\u00f6rd\u00fcnc\u00fc g\u00fcn, d\u00f6n\u00fcm noktas\u0131na dayal\u0131 olarak hasat ve alt k\u00fclt\u00fcr i\u00e7in en uygun zaman olarak belirlenmi\u015ftir. CCS ile 4 g\u00fcnl\u00fck ekimden sonra, huperzin A i\u00e7eri\u011fi 49.34% artarak maksimum de\u011ferine ula\u015fm\u0131\u015ft\u0131r. K\u00fclt\u00fcr sistemindeki genel huperzin A i\u00e7eri\u011fi \u00f6nce artan sonra azalan bir e\u011filim g\u00f6stermi\u015ftir. Bunun nedeni, b\u00fcy\u00fcmenin sonraki a\u015famas\u0131nda, endofitik mantarlar\u0131n bitki h\u00fccresi farkl\u0131la\u015fma yetene\u011finden daha g\u00fc\u00e7l\u00fc \u00fcreme yetene\u011fine sahip olmas\u0131, k\u00fclt\u00fcr ortam\u0131ndaki besinler ve b\u00fcy\u00fcme alan\u0131 i\u00e7in rekabet etmesi ve h\u00fccre say\u0131s\u0131nda azalmaya neden olmas\u0131d\u0131r. Bu nedenle, hasat ve alt k\u00fclt\u00fcr zaman\u0131n\u0131n se\u00e7imi, ortak k\u00fclt\u00fcr sisteminde huperzin A'n\u0131n giderek zenginle\u015fmesini sa\u011flaman\u0131n anahtar\u0131d\u0131r. Ayn\u0131 zamanda, bitki hormonu 2,4-D konsantrasyonunun sistem \u00fczerinde \u00f6nemli bir etkisi vard\u0131r. 2,4-D, bitki organlar\u0131n\u0131n farkl\u0131la\u015fmas\u0131n\u0131 ve kallus dokusunun ind\u00fcklenmesini te\u015fvik eder, ancak konsantrasyon \u00e7ok y\u00fcksek oldu\u011funda h\u00fccre farkl\u0131la\u015fmas\u0131 \u00fczerinde inhibe edici bir etkiye sahiptir. Bu nedenle, k\u00fclt\u00fcr sisteminde optimum konsantrasyon olarak 5mg\/L kullan\u0131lm\u0131\u015ft\u0131r. Bu deney, huperzin A'n\u0131n biyosentezini sa\u011flamak i\u00e7in bir ortak k\u00fclt\u00fcr sistemini ba\u015far\u0131yla kullanm\u0131\u015ft\u0131r. Bu y\u00f6ntem, geleneksel sabit kavramlar\u0131n \u00fcstesinden gelir \u00e7\u00fcnk\u00fc bitki somatik h\u00fccre k\u00fclt\u00fcr\u00fc \u00f6nceden kapsaml\u0131 bir sterilizasyon gerektirmez. Bitki somatik h\u00fccreleri ve endofitik mantarlar birlikte k\u00fclt\u00fcre al\u0131nabilir ve huperzin A \u00fcretimi belirli oranlarda te\u015fvik edilebilir. Yeti\u015ftirme d\u00f6ng\u00fcs\u00fc do\u011fru bir \u015fekilde kavrand\u0131\u011f\u0131 s\u00fcrece, bu kullan\u0131\u015fl\u0131 ve h\u0131zl\u0131 y\u00f6ntem, bitki kaynaklar\u0131n\u0131n korunmas\u0131 ve huperzin A'n\u0131n \u00f6nemli biyoaktif maddelerinin zenginle\u015ftirilmesi i\u00e7in b\u00fcy\u00fck \u00f6nem ta\u015f\u0131yan huperzin A'y\u0131 biriktirmek i\u00e7in kullan\u0131labilir.<\/p>","protected":false},"excerpt":{"rendered":"<p>Study on the promotion of incremental enrichment of huperzine A by symbiotic cultivation method Huperzia serrata (Thunb. ex Murray) is a fern plant in the family Taxaceae, belonging to the genus Taxodium. It is a rare Chinese herbal medicine used for treating traumatic injuries, detoxification, pain relief, and treating schizophrenia. Snake foot fir is currently [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Study on the promotion of incremental enrichment of huperzine A by symbiotic cultivation method - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/tr\/huperzin\/\" \/>\n<meta property=\"og:locale\" content=\"tr_TR\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Study on the promotion of incremental enrichment of huperzine A by symbiotic cultivation method - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Study on the promotion of incremental enrichment of huperzine A by symbiotic cultivation method Huperzia serrata (Thunb. ex Murray) is a fern plant in the family Taxaceae, belonging to the genus Taxodium. It is a rare Chinese herbal medicine used for treating traumatic injuries, detoxification, pain relief, and treating schizophrenia. 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