{"id":4566,"date":"2024-08-04T14:53:22","date_gmt":"2024-08-04T14:53:22","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=4566"},"modified":"2024-08-04T14:53:22","modified_gmt":"2024-08-04T14:53:22","slug":"callicarpa-nudiflora","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/tr\/callicarpa-nudiflora\/","title":{"rendered":"\u00c7\u0131plak Mor Boncuklar\u0131n Anti H1N1 Aktif Bile\u015fenlerinin ve Mekanizmalar\u0131n\u0131n UPLC-Q-Exactive-Orbitrap-MS, A\u011f Farmakolojisi ve Deneysel Do\u011frulamaya Dayal\u0131 Olarak Ara\u015ft\u0131r\u0131lmas\u0131"},"content":{"rendered":"<p>\u00c7\u0131plak Mor Boncuklar\u0131n Anti H1N1 Aktif Bile\u015fenlerinin ve Mekanizmalar\u0131n\u0131n UPLC-Q-Exactive-Orbitrap-MS, A\u011f Farmakolojisi ve Deneysel Do\u011frulamaya Dayal\u0131 Olarak Ara\u015ft\u0131r\u0131lmas\u0131<br \/>\nGeleneksel \u00c7in ilac\u0131 olan Callicarpa nudiflora Hook.&amp;Arn., Verbenaceae familyas\u0131ndan Callicarpa nudiflora Hook.&amp;Arn. bitkisinin kurutulmu\u015f bir yapra\u011f\u0131d\u0131r. \u00c7\u0131plak Mor Boncuklar \u00e7o\u011funlukla Hainan, Guangxi, Guangdong ve di\u011fer b\u00f6lgelerde da\u011f\u0131t\u0131lmaktad\u0131r ve otantik \u00fcretim alan\u0131 Hainan Eyaletindeki Wuzhishan B\u00f6lgesidir. \u00c7\u0131plak \u00c7i\u00e7ek Mor \u0130nci, \u00c7in Halk Cumhuriyeti Farmakopesi'nin 2020 bask\u0131s\u0131na yeni eklenen tek geleneksel \u00c7in ilac\u0131d\u0131r. Tek tarafl\u0131 preparatlar\u0131 olan \u00c7\u0131plak \u00c7i\u00e7ek Mor \u0130nci Tabletleri ve \u00c7\u0131plak \u00c7i\u00e7ek Mor \u0130nci Kaps\u00fclleri, a\u015f\u0131r\u0131 kan \u0131s\u0131s\u0131 ve toksisitenin neden oldu\u011fu solunum ve sindirim kanamalar\u0131n\u0131 ve bakteriyel enfeksiy\u00f6z iltihaplar\u0131 tedavi etmek i\u00e7in yayg\u0131n olarak kullan\u0131lmaktad\u0131r. Fitokimyac\u0131lar, fenilpropanoidler, flavonoidler, triterpenoidler, diterpenler, iridoidler, u\u00e7ucu ya\u011flar ve daha fazlas\u0131 dahil olmak \u00fczere \u00e7\u0131plak mor incilerden 300'den fazla bile\u015fik tan\u0131mlam\u0131\u015ft\u0131r. Modern farmakolojik ara\u015ft\u0131rmalar, \u00e7\u0131plak \u00e7i\u00e7ek mor incisinin anti-enflamatuar, antitrombotik, anti-t\u00fcm\u00f6r, antibakteriyel ve hepatoprotektif aktivitelere sahip oldu\u011funu do\u011frulam\u0131\u015ft\u0131r. Antiviral aktiviteye sahip geleneksel \u00c7in t\u0131bb\u0131n\u0131n taranmas\u0131 s\u00fcrecinde, \u00e7\u0131plak \u00e7i\u00e7ek mor incisinin ekstrakt\u0131n\u0131n iyi bir antiviral aktiviteye sahip oldu\u011fu bulunmu\u015ftur (H1N1 influenza vir\u00fcs\u00fc, enterovir\u00fcs 71, vb. gibi). \u0130nfluenza A vir\u00fcs\u00fc enfeksiyonu, pn\u00f6moniye ba\u011fl\u0131 \u00f6l\u00fcmlerin yayg\u0131n bir nedenidir. \u0130nfluenza A vir\u00fcs\u00fc ile \u015fiddetli enfeksiyon, influenza A vir\u00fcs\u00fcn\u00fcn neden oldu\u011fu ana \u00f6l\u00fcm nedenlerinden biri olan akut solunum s\u0131k\u0131nt\u0131s\u0131 sendromu olarak bilinen bilateral akci\u011fer infiltrasyonuna ve hipoksemiye neden olabilir. Bu deney, \u00e7\u0131plak \u00e7i\u00e7ek mor boncu\u011funun anti H1N1 aktivitesine odaklanmaktad\u0131r. \u00c7\u0131plak \u00e7i\u00e7ek moru boncu\u011funun etkili k\u0131s\u0131mlar\u0131n\u0131n kimyasal bile\u015fimi ultra y\u00fcksek performansl\u0131 s\u0131v\u0131 kromatografisi kuadrupol elektrostatik alan orbitrap MS kullan\u0131larak tan\u0131mlanm\u0131\u015f ve \u00e7\u0131plak \u00e7i\u00e7ek moru boncu\u011funun anti H1N1 mekanizmas\u0131 a\u011f farmakolojisi kullan\u0131larak tahmin edilmi\u015f ve deneysel olarak do\u011frulanm\u0131\u015ft\u0131r. \u00c7\u0131plak \u00e7i\u00e7ek moru boncu\u011funun H1N1'e kar\u015f\u0131 etki mekanizmas\u0131 \u00f6n ara\u015ft\u0131rmaya tabi tutulmu\u015ftur.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4570\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-73.png\" alt=\"\" width=\"340\" height=\"709\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4571\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-63.png\" alt=\"\" width=\"340\" height=\"234\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4572\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-60.png\" alt=\"\" width=\"600\" height=\"621\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4573\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-50.png\" alt=\"\" width=\"600\" height=\"660\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4574\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-2.jpg\" alt=\"\" width=\"539\" height=\"748\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-2.jpg 539w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-2-519x720.jpg 519w\" sizes=\"(max-width: 539px) 100vw, 539px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4575\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-44.png\" alt=\"\" width=\"539\" height=\"272\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4576\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-42.png\" alt=\"\" width=\"600\" height=\"784\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-42.png 600w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-42-551x720.png 551w\" sizes=\"(max-width: 600px) 100vw, 600px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4577\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-36.png\" alt=\"\" width=\"600\" height=\"539\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4578\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-31.png\" alt=\"\" width=\"600\" height=\"304\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4579\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-27.png\" alt=\"\" width=\"600\" height=\"244\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4580\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-25.png\" alt=\"\" width=\"340\" height=\"219\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4581\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-21.png\" alt=\"\" width=\"340\" height=\"546\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4582\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-18.png\" alt=\"\" width=\"600\" height=\"271\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4583\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/14-15.png\" alt=\"\" width=\"600\" height=\"327\" \/>callicarpa nudiflora<br \/>\n\u0130nfluenza A vir\u00fcs\u00fc, yayg\u0131n olarak kullan\u0131lan M2 kanal inhibit\u00f6rlerine ve NA inhibit\u00f6rlerine kar\u015f\u0131 \u00e7e\u015fitli derecelerde diren\u00e7 geli\u015ftirmi\u015ftir. Bu nedenle, anti influenza A i\u00e7in yeni ila\u00e7lar veya tedavi y\u00f6ntemleri bulmak \u00e7\u00f6z\u00fclmesi gereken acil bir sorun haline gelmi\u015ftir. Geleneksel \u00c7in t\u0131bb\u0131, influenza A vir\u00fcs\u00fcn\u00fcn klinik tedavisinde \u00f6nemli bir rol oynam\u0131\u015ft\u0131r. Geleneksel \u00c7in t\u0131bb\u0131 teorisindeki b\u00fct\u00fcnsel kavram, hastalar\u0131 organik bir b\u00fct\u00fcn olarak sistematik bir \u015fekilde d\u00fczenlerken, a\u011f farmakolojisi, geleneksel \u00c7in t\u0131bb\u0131ndaki b\u00fct\u00fcnsel kavramla tutarl\u0131 olan bir ila\u00e7 bile\u015feni hedef yolu hastal\u0131k a\u011f\u0131 olu\u015fturarak a\u011fdaki her bir d\u00fc\u011f\u00fcm\u00fcn biyolojik i\u015flevleri ile hastal\u0131klar aras\u0131ndaki etkile\u015fimi ara\u015ft\u0131r\u0131r. Bu deney ilk olarak geleneksel \u00c7in ilac\u0131 \u00c7\u0131plak \u00c7i\u00e7ek Mor \u0130nci'nin ana anti H1N1 aktif b\u00f6lgelerini taram\u0131\u015f ve 34 kimyasal bile\u015feni tan\u0131mlamak i\u00e7in b\u00f6lgeleri analiz etmi\u015ftir. Literat\u00fcr ve veri tabanlar\u0131 birle\u015ftirilerek, ila\u00e7lar\u0131n ve hastal\u0131klar\u0131n 67 \u00f6rt\u00fc\u015fen hedefi belirlendi. \u00c7apraz hedeflerin zenginle\u015ftirme analizi yoluyla, EACN'nin H1N1'e kar\u015f\u0131 \u00f6nemli biyolojik s\u00fcrecinin protein fosforilasyonunun pozitif d\u00fczenlenmesi ve oksidatif strese yan\u0131t olabilece\u011fini tahmin ediyoruz. KEGG zenginle\u015ftirme analizi sonu\u00e7lar\u0131, EACN'deki 19 bile\u015fi\u011fin 11 hedef arac\u0131l\u0131\u011f\u0131yla influenza A vir\u00fcs yolu \u00fczerinde etkili oldu\u011funu g\u00f6stermi\u015ftir. \u0130la\u00e7, PLG ve PRSS1'e etki ederek H1N1 vir\u00fcs\u00fcn\u00fcn M2 kanal\u0131n\u0131 etkiler ve PLG arac\u0131l\u0131\u011f\u0131yla n\u00f6raminidaz (NA) yoluna etki ederek vir\u00fcs sal\u0131n\u0131m s\u00fcrecini de etkileyebilir. PLG ve PRSS1, EACN'nin do\u011frudan H1N1 \u00fczerinde etkili olmas\u0131 i\u00e7in kilit hedefler olabilir. EACN, d\u00f6k\u00fclme ve sal\u0131n\u0131m s\u00fcre\u00e7lerini etkileyerek H1N1'in \u00e7o\u011falmas\u0131n\u0131 engelleyebilir. \u0130la\u00e7 i\u00e7eri\u011fi hedef yolu hastal\u0131k a\u011f\u0131nda, RELA ve NF - \u03ba B1 en y\u00fcksek derece de\u011ferlerine sahip iki hedeftir. Bulunduklar\u0131 NF - \u03ba B sinyal yolu IL1 \u03b2, TNF - \u03b1, IL-6 gibi fakt\u00f6rlerin ifadesini destekleyebilir ve enflamatuar yan\u0131t\u0131 te\u015fvik edebilir, bu da EACN'nin NF - \u03ba B sinyal yolunu d\u00fczenlemek ve enflamasyonun v\u00fccuda verdi\u011fi zarar\u0131 azaltmak i\u00e7in RELA ve NF - \u03ba B1 gibi kilit hedefler \u00fczerinde etkili olabilece\u011fini d\u00fc\u015f\u00fcnd\u00fcrmektedir. A\u011f farmakolojisi taraf\u0131ndan \u00f6ng\u00f6r\u00fclen sonu\u00e7lara g\u00f6re, EACN T h\u00fccresi sinyal yolaklar\u0131n\u0131 d\u00fczenleyebilir, Th1 ve Th2 farkl\u0131la\u015fmas\u0131n\u0131 etkileyebilir ve ba\u011f\u0131\u015f\u0131kl\u0131k d\u00fczenleyici etkiler g\u00f6sterebilir. Bu nedenle, bu \u00e7al\u0131\u015fmada EACN'nin H1N1 proliferasyonu \u00fczerindeki inhibit\u00f6r etkisini, anti-enflamatuar etkisini ve ba\u011f\u0131\u015f\u0131kl\u0131k d\u00fczenleyici etkisini do\u011frulamak i\u00e7in hayvan deneyleri yap\u0131lm\u0131\u015ft\u0131r. Deneysel sonu\u00e7lar, EACN'nin H1N1 enfeksiyonunun neden oldu\u011fu kilo kayb\u0131n\u0131 ve akci\u011fer indeksi art\u0131\u015f\u0131n\u0131 iyile\u015ftirebilece\u011fini, fare akci\u011fer dokusundaki viral y\u00fck\u00fc azaltabilece\u011fini, fare akci\u011fer dokusundaki patolojik hasar\u0131 hafifletebilece\u011fini, periferik kan serumundaki TNF - \u03b1, IFN - \u03b3, IL-1 \u03b2 seviyelerini d\u00fc\u015f\u00fcrebilece\u011fini ve serum antikor IgG seviyesini art\u0131rabilece\u011fini g\u00f6stermi\u015ftir. Bu \u00e7al\u0131\u015fmada ilk olarak Naked Purple Pearl'\u00fcn H1N1'e kar\u015f\u0131 aktif ekstraksiyon b\u00f6lgelerini taramak i\u00e7in in vitro deneyler kullan\u0131lm\u0131\u015f ve UPLC-Q-Hexactive-Orbitrap-MS ve a\u011f farmakolojisi kullan\u0131larak EACN'nin H1N1'e kar\u015f\u0131 aktif bile\u015fenleri tahmin edilmi\u015ftir. Tahmin edilen sonu\u00e7lar hayvan deneyleri ile do\u011frulanm\u0131\u015f ve quercetin, myricetin, luteolin, kaempferol, quercetin, apigenin ve acacetin dahil olmak \u00fczere H1N1'e kar\u015f\u0131 EACN'nin potansiyel aktif bile\u015fenleri taranm\u0131\u015ft\u0131r. Naked Purple Pearl'\u00fcn do\u011frudan vir\u00fcs inhibisyonu, anti-enflamatuar etkiler ve ba\u011f\u0131\u015f\u0131kl\u0131k d\u00fczenlemesi gibi \u00e7oklu yollar arac\u0131l\u0131\u011f\u0131yla anti H1N1 etkileri g\u00f6sterebilece\u011fi ilk olarak g\u00f6sterilmi\u015ftir. Sonraki deneylerde, se\u00e7ilen monomerik bile\u015fikleri do\u011frulamak ve EACN'nin anti H1N1 etkisinin mekanizmas\u0131n\u0131 mRNA ve protein seviyelerinde daha fazla ara\u015ft\u0131rmak i\u00e7in in vitro ve in vivo deneyler yap\u0131lmas\u0131 gerekmektedir.<\/p>","protected":false},"excerpt":{"rendered":"<p>Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation The traditional Chinese medicine, Callicarpa nudiflora Hook.&amp;Arn., is a dried leaf of the plant Callicarpa nudiflora Hook.&amp;Arn. in the family Verbenaceae. Naked Purple Beads are mainly distributed in Hainan, Guangxi, Guangdong and other regions, with [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/tr\/callicarpa-nudiflora\/\" \/>\n<meta property=\"og:locale\" content=\"tr_TR\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation The traditional Chinese medicine, Callicarpa nudiflora Hook.&amp;Arn., is a dried leaf of the plant Callicarpa nudiflora Hook.&amp;Arn. in the family Verbenaceae. 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\u00c7in Kimya \u00dcreticisi","robots":{"index":"index","follow":"follow","max-snippet":"max-snippet:-1","max-image-preview":"max-image-preview:large","max-video-preview":"max-video-preview:-1"},"canonical":"https:\/\/longchangextracts.com\/tr\/callicarpa-nudiflora\/","og_locale":"tr_TR","og_type":"article","og_title":"Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation - China Chemical Manufacturer","og_description":"Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation The traditional Chinese medicine, Callicarpa nudiflora Hook.&amp;Arn., is a dried leaf of the plant Callicarpa nudiflora Hook.&amp;Arn. in the family Verbenaceae. 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