{"id":3536,"date":"2024-08-02T14:40:15","date_gmt":"2024-08-02T14:40:15","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=3536"},"modified":"2024-08-02T14:40:15","modified_gmt":"2024-08-02T14:40:15","slug":"huaze-lan","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/tr\/huaze-lan\/","title":{"rendered":"Huaze Lan'daki endofitik fungus Septoriella phragmitis'in sekonder metabolitleri ve biyolojik aktiviteleri \u00fczerine \u00e7al\u0131\u015fma"},"content":{"rendered":"<p>Huaze Lan'daki endofitik fungus Septoriella phragmitis'in sekonder metabolitleri ve biyolojik aktiviteleri \u00fczerine \u00e7al\u0131\u015fma<\/p>\n<p>\u00c7ok say\u0131da endofitik mantar t\u00fcr\u00fc vard\u0131r ve bunlar\u0131n metabolitleri \u00e7e\u015fitlidir, bu da konak\u00e7\u0131n\u0131nkine benzer \u00e7e\u015fitli aktif maddeler \u00fcretebilir. Modern farmakolojik \u00e7al\u0131\u015fmalar, Huaze orkidesinden elde edilen endofitik mantar Septoriella phragmitis \u00f6z\u00fct\u00fcn\u00fcn antidepresan, anti-enflamatuar, ba\u011f\u0131\u015f\u0131kl\u0131k d\u00fczenleyici ve antioksidan gibi aktivitelere sahip oldu\u011funu g\u00f6stermi\u015ftir. Zhang ve arkada\u015flar\u0131, Hua Zelan'dan 8 endofitik mantar izole etmi\u015f ve fermantasyon suyunun etil asetat \u00f6z\u00fct\u00fc \u00fczerinde in vitro anti-t\u00fcm\u00f6r deneyleri ger\u00e7ekle\u015ftirmi\u015ftir, ancak bireysel bile\u015fikler \u00fczerinde ara\u015ft\u0131rma yap\u0131lmam\u0131\u015ft\u0131r. Ara\u015ft\u0131rma ekibi Huaze Lan'\u0131n k\u00f6klerinden bir endofitik mantar izole etmi\u015f ve su\u015f tan\u0131mlamas\u0131ndan sonra bunun Zhang Jianfen ve arkada\u015flar\u0131 taraf\u0131ndan izole edilen endofitik mantardan farkl\u0131 oldu\u011fu ve Septoriella phragmitis oldu\u011fu belirlenmi\u015ftir. \u015eu anda sekonder metabolitleri hakk\u0131nda bilgi veren bir literat\u00fcr bulunmamaktad\u0131r. Septoriella phragmatis endofitik mantar\u0131n\u0131n maddi temelini daha fazla incelemek i\u00e7in, bu \u00e7al\u0131\u015fma kimyasal bile\u015fenlerini izole edip tan\u0131mlad\u0131 ve anti diyabet ve anti-t\u00fcm\u00f6r aktivitelerini test ederek, olduk\u00e7a etkili ve d\u00fc\u015f\u00fck toksik anti diyabet \u00f6nc\u00fc bile\u015fi\u011fi bulmak ve bu t\u0131bbi mantar kayna\u011f\u0131n\u0131 geli\u015ftirmek ve kullanmak i\u00e7in bir referans sa\u011flad\u0131.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone  wp-image-3539\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/640.jpg\" alt=\"\" width=\"700\" height=\"324\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/640.jpg 854w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/640-768x355.jpg 768w\" sizes=\"(max-width: 700px) 100vw, 700px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-3540\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/640.webp\" alt=\"\" width=\"472\" height=\"364\" \/>Bu \u00e7al\u0131\u015fmada su\u015fun kimyasal bile\u015fimi ara\u015ft\u0131r\u0131lm\u0131\u015f ve 5 alkaloid, 4 fenol ve 1 benzofuran dahil olmak \u00fczere 10 bile\u015fik elde edilmi\u015f ve bunlar\u0131n t\u00fcm\u00fc ilk kez su\u015ftan izole edilmi\u015ftir. Ayr\u0131ca, mikroorganizmalar\u0131n Eupatorium adenophorum bitkisinin etken maddesi olan puerarini \u00fcretebildi\u011fi ilk kez ke\u015ffedilmi\u015ftir. Farmakolojik aktivite test sonu\u00e7lar\u0131, bile\u015fik 6 ve 7'nin s\u0131ras\u0131yla alfa glukozidaza kar\u015f\u0131 iyi inhibit\u00f6r aktiviteye sahip oldu\u011funu; Bile\u015fik 6, 7 ve 9'un iyi PTP1B inhibit\u00f6r aktivitesi sergiledi\u011fini ve aktivitelerinin pozitif ila\u00e7 sodyum ortovanadattan daha \u00fcst\u00fcn oldu\u011funu; Bile\u015fik 5 ve 6'n\u0131n di\u011fer bile\u015fiklere k\u0131yasla mide kanseri h\u00fccre hatt\u0131 HGC-27'ye kar\u015f\u0131 belirli inhibit\u00f6r aktivite sergiledi\u011fini g\u00f6stermi\u015ftir. Daha ileri molek\u00fcler yerle\u015ftirme deneyleri, 6 ve 7 numaral\u0131 bile\u015fiklerin hidrojen ba\u011f\u0131, hidrofobiklik, konjugasyon vb. gibi \u00e7e\u015fitli etkile\u015fimler yoluyla \u03b1-glukozidaz veya PTP1B hedef proteinlerinin amino asit kal\u0131nt\u0131lar\u0131yla etkile\u015fime girebilece\u011fini g\u00f6stermi\u015ftir. \u015eu anda, hi\u00e7bir literat\u00fcr Septoriella phragmatis mantar\u0131n\u0131n sekonder metabolitlerini rapor etmemi\u015ftir. Bu \u00e7al\u0131\u015fma, bu t\u00fcr\u00fcn ikincil metabolitlerini ilk kez rapor etmi\u015ftir ve bulunan baz\u0131 bile\u015fikler diyabete kar\u015f\u0131 \u00e7ift hedefli inhibit\u00f6r aktiviteye sahiptir. Ara\u015ft\u0131rma sonu\u00e7lar\u0131 2024 y\u0131l\u0131nda Natural Product Research and Development dergisinin 6. say\u0131s\u0131nda yay\u0131mlanm\u0131\u015ft\u0131r.<\/p>\n<p>&nbsp;<\/p>\n<p>&nbsp;<\/p>\n<p>&nbsp;<\/p>","protected":false},"excerpt":{"rendered":"<p>Study on the secondary metabolites and biological activities of the endophytic fungus Septoriella phragmitis in Huaze Lan There are abundant species of endophytic fungi, and their metabolites are diverse, which may produce various active substances similar to those of the host. Modern pharmacological studies have shown that the extract of the endophytic fungus Septoriella phragmitis [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Study on the secondary metabolites and biological activities of the endophytic fungus Septoriella phragmitis in Huaze Lan - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/tr\/huaze-lan\/\" \/>\n<meta property=\"og:locale\" content=\"tr_TR\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Study on the secondary metabolites and biological activities of the endophytic fungus Septoriella phragmitis in Huaze Lan - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Study on the secondary metabolites and biological activities of the endophytic fungus Septoriella phragmitis in Huaze Lan There are abundant species of endophytic fungi, and their metabolites are diverse, which may produce various active substances similar to those of the host. 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