{"id":6930,"date":"2024-08-06T17:59:26","date_gmt":"2024-08-06T17:59:26","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=6930"},"modified":"2024-08-06T17:59:26","modified_gmt":"2024-08-06T17:59:26","slug":"polar-actinomycetes","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/hu\/polar-actinomycetes\/","title":{"rendered":"A pol\u00e1ris aktinomicit\u00e1k m\u00e1sodlagos anyagcsereterm\u00e9keinek \u00e9s farmakol\u00f3giai aktivit\u00e1sainak kutat\u00e1s\u00e1ban el\u00e9rt eredm\u00e9nyek"},"content":{"rendered":"<p>A pol\u00e1ris aktinomicit\u00e1k m\u00e1sodlagos anyagcsereterm\u00e9keinek \u00e9s farmakol\u00f3giai aktivit\u00e1sainak kutat\u00e1s\u00e1ban el\u00e9rt eredm\u00e9nyek<br \/>\nAz aktinomicita az aktinobakt\u00e9riumok t\u00f6rzs\u00e9be tartoz\u00f3, Gram-pozit\u00edv bakt\u00e9rium. Az aktinomic\u00e9t\u00e1kb\u00f3l sz\u00e1rmaz\u00f3 m\u00e1sodlagos metabolitok a mikroorganizmusokb\u00f3l sz\u00e1rmaz\u00f3 m\u00e1sodlagos metabolitok mintegy 45%-j\u00e9t teszik ki, \u00e9s sz\u00e1mos biol\u00f3giai aktivit\u00e1st mutatnak, bele\u00e9rtve a daganatellenes, antibakteri\u00e1lis, gyullad\u00e1scs\u00f6kkent\u0151, v\u00edrusellenes \u00e9s angiogenetikai hat\u00e1st. Az aktinomicit\u00e1kb\u00f3l sz\u00e1rmaz\u00f3 antibiotikumok teszik ki a bejelentett term\u00e9szetes antibiotikumok 70% r\u00e9sz\u00e9t, \u00e9s n\u00e9h\u00e1nyat, p\u00e9ld\u00e1ul a vankomicint \u00e9s az azitromicint sz\u00e9les k\u00f6rben haszn\u00e1lj\u00e1k a klinikai gyakorlatban. Az aktinobakt\u00e9riumokat mindig is a mikrobi\u00e1lis forr\u00e1sokb\u00f3l sz\u00e1rmaz\u00f3 \u00fajonnan akt\u00edv m\u00e1sodlagos metabolitok j\u00f3 forr\u00e1s\u00e1nak tekintett\u00e9k.<br \/>\nA sarkvid\u00e9kek \u00e1ltal\u00e1ban az \u00c9szaki \u00e9s a D\u00e9li-sarkot \u00e9s azok alr\u00e9gi\u00f3it foglalj\u00e1k magukban, amelyeket alacsony h\u0151m\u00e9rs\u00e9klet, sarki napf\u00e9ny \u00e9s er\u0151s ultraibolya sug\u00e1rz\u00e1s jellemez. A sarkvid\u00e9ki mikroorganizmusok egyedi g\u00e9nszab\u00e1lyoz\u00e1st \u00e9s anyagcsere-funkci\u00f3kat fejlesztettek ki a sz\u00e9ls\u0151s\u00e9ges sarkvid\u00e9ki k\u00f6r\u00fclm\u00e9nyekhez val\u00f3 alkalmazkod\u00e1s \u00e9rdek\u00e9ben, \u00e9s \u00edgy k\u00e9pesek szerkezetileg \u00fajszer\u0171 m\u00e1sodlagos anyagcsereterm\u00e9kek el\u0151\u00e1ll\u00edt\u00e1s\u00e1ra. Az elm\u00falt \u00e9vekben a kutat\u00f3k sz\u00e1mos szerkezetileg egyed\u00fcl\u00e1ll\u00f3 \u00e9s nagy aktivit\u00e1s\u00fa m\u00e1sodlagos anyagcsereterm\u00e9ket fedeztek fel a pol\u00e1ris aktinomicit\u00e1kb\u00f3l. Ez a cikk a pol\u00e1ris aktinomyc\u00e9t\u00e1k m\u00e1sodlagos metabolitjaival \u00e9s farmakol\u00f3giai aktivit\u00e1s\u00e1val kapcsolatos kutat\u00e1si eredm\u00e9nyeket tekinti \u00e1t 1999 \u00e9s 2021 k\u00f6z\u00f6tt. K\u00e9miai szerkezett\u00edpusaik szerint peptidek, alkaloidok, terp\u00e9nek, makrolidok, poliketonok, makrolakt\u00e1mok \u00e9s egy\u00e9b kateg\u00f3ri\u00e1kba sorolhat\u00f3k. Ez a cikk \u00f6sszefoglalja az elm\u00falt \u00e9vekben \u00fajonnan felfedezett pol\u00e1ris aktinomicit\u00e1kb\u00f3l sz\u00e1rmaz\u00f3 m\u00e1sodlagos metabolitokat (l\u00e1sd az 1. t\u00e1bl\u00e1zatot), amelyek alapot ny\u00fajthatnak a pol\u00e1ris aktinomicita er\u0151forr\u00e1sok jobb fejleszt\u00e9s\u00e9hez \u00e9s felhaszn\u00e1l\u00e1s\u00e1hoz.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6988\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-270.png\" alt=\"\" width=\"783\" height=\"655\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-270.png 783w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-270-768x642.png 768w\" sizes=\"(max-width: 783px) 100vw, 783px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6989\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-221.png\" alt=\"\" width=\"786\" height=\"452\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-221.png 786w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-221-768x442.png 768w\" sizes=\"(max-width: 786px) 100vw, 786px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6990\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-208.png\" alt=\"\" width=\"785\" height=\"241\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-208.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-208-768x236.png 768w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6991\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-188.png\" alt=\"\" width=\"782\" height=\"246\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-188.png 782w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-188-768x242.png 768w\" sizes=\"(max-width: 782px) 100vw, 782px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6992\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-171.png\" alt=\"\" width=\"785\" height=\"327\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-171.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-171-768x320.png 768w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6993\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-156.png\" alt=\"\" width=\"786\" height=\"453\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-156.png 786w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-156-768x443.png 768w\" sizes=\"(max-width: 786px) 100vw, 786px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6994\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-143.png\" alt=\"\" width=\"785\" height=\"174\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-143.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-143-768x170.png 768w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6995\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-130.png\" alt=\"\" width=\"785\" height=\"337\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-130.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-130-768x330.png 768w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6996\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-122.png\" alt=\"\" width=\"786\" height=\"223\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-122.png 786w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-122-768x218.png 768w\" sizes=\"(max-width: 786px) 100vw, 786px\" \/>1999 \u00e9s 2021 k\u00f6z\u00f6tt 104 m\u00e1sodlagos metabolitot jelentettek be pol\u00e1ris aktinomyc\u00e9t\u00e1kb\u00f3l hazai \u00e9s nemzetk\u00f6zi szinten egyar\u00e1nt, amelyek k\u00f6z\u00fcl 44 (42,3%) \u00faj vegy\u00fclet volt. Az \u00faj m\u00e1sodlagos metabolitok \u00f6sszefoglal\u00f3j\u00e1t az 1. t\u00e1bl\u00e1zat tartalmazza. A pol\u00e1ris aktinomyc\u00e9t\u00e1k m\u00e1sodlagos metabolitjainak nagy r\u00e9sz\u00e9t a Streptomyces nemzets\u00e9gb\u0151l izol\u00e1lt\u00e1k (74,5%), m\u00edg kis h\u00e1nyadukat az \u00e1l-Nocardia nemzets\u00e9gb\u0151l (14,2%), a termofil Bacillus nemzets\u00e9gb\u0151l (2,8%), a Nocardia-szer\u0171 nemzets\u00e9gb\u0151l (0,9%) \u00e9s egy\u00e9b nemzets\u00e9gekb\u0151l (7,7%) (8. \u00e1bra, balra). A k\u00e9miai szerkezett\u00edpusok oszt\u00e1lyoz\u00e1sa szerint a 104 m\u00e1sodlagos metabolit k\u00f6z\u00fcl 21 (20,2%) peptidvegy\u00fclet, 9 (8,7%) alkaloid, 11 (10,6%) terp\u00e9n, 15 (14,4%) makrolid, 19 (18,3%) poliketon, 6 (5,8%) makrolakt\u00e1m \u00e9s 23 (22,1%) egy\u00e9b t\u00edpus\u00fa vegy\u00fclet. A f\u0151 szerkezeti t\u00edpusok a peptidek, poliketonok, makrolidok stb. (8. \u00e1bra, jobbra). K\u00f6z\u00fcl\u00fck a nagyon ritka szerkezet\u0171 m\u00e1sodlagos metabolitok k\u00f6z\u00e9 tartoznak a nitroporozin A (29) \u00e9s B (30), az antartin (41), a gephyromycin (41) stb. 60), a szalinikinonok G-I (72-74) stb. A 104 m\u00e1sodlagos metabolit legt\u00f6bbje j\u00f3 farmakol\u00f3giai aktivit\u00e1ssal rendelkezik, p\u00e9ld\u00e1ul antibakteri\u00e1lis, gombaellenes, v\u00edrusellenes \u00e9s citotoxikus hat\u00e1s\u00fa. Els\u0151sorban tumorellenes aktivit\u00e1s jellemzi, amely g\u00e1tl\u00f3 hat\u00e1ssal van a leuk\u00e9mi\u00e1ra, vastagb\u00e9lr\u00e1kra, epiderm\u00e1lis r\u00e1kra, myel\u00f3m\u00e1ra, m\u00e9hnyakr\u00e1kra, eml\u0151r\u00e1kra, melanom\u00e1ra, gyomorr\u00e1kra \u00e9s m\u00e1s tumorsejtekre. Egyes vegy\u00fcletek jelent\u0151s aktivit\u00e1ssal rendelkeznek, p\u00e9ld\u00e1ul a C-1027 kromof\u00f3r-V jelent\u0151s citotoxicit\u00e1ssal, a szalinikinonok G \uff5e H jelent\u0151s antibakteri\u00e1lis aktivit\u00e1ssal, \u00e9s az N - (2-hidroxifeny1) -2-fenazinamin (NHP) jelent\u0151s gombaellenes \u00e9s citotoxicit\u00e1ssal rendelkezik. Ezenk\u00edv\u00fcl egyes vegy\u00fcletek szelekt\u00edv g\u00e1tl\u00f3 hat\u00e1ssal is rendelkeznek. A k\u00f6vetkez\u0151 az antibakteri\u00e1lis aktivit\u00e1s, bele\u00e9rtve az antibakteri\u00e1lis \u00e9s gombaellenes aktivit\u00e1st, amely g\u00e1tl\u00f3 hat\u00e1ssal van a Candida albicans, Escherichia coli, Pseudomonas aeruginosa, Staphylococcus aureus, Bacillus subtilis, Proteus mirabilis, Bacillus cereus, Bacillus subtilis \u00e9s Micrococcus luteus eset\u00e9ben. N\u00e9h\u00e1nynak olyan hat\u00e1sai vannak, mint az angiogenezis elleni, antioxid\u00e1ns, a sejtek lipidszintj\u00e9nek cs\u00f6kkent\u00e9se, a melaninszint\u00e9zis g\u00e1tl\u00e1sa \u00e9s a glutamin aktivit\u00e1s. Tov\u00e1bbi kutat\u00e1s \u00e9s fejleszt\u00e9s indokolt az olyan \u00faj szerkezet\u0171, ak\u00e1r ritka v\u00e1zszerkezet\u0171 \u00e9s jelent\u0151s aktivit\u00e1s\u00fa m\u00e1sodlagos metabolitok eset\u00e9ben, mint a nitrosporozin A (29) \u00e9s B (30), antagonista (41), gephyromycin (60) \u00e9s a szalinequin G-I (72-74).<br \/>\n\u00d6sszefoglalva, a pol\u00e1ris aktinomicit\u00e1k b\u0151s\u00e9ges forr\u00e1sokkal rendelkeznek, a kutat\u00e1sok k\u00f6z\u00e9ppontj\u00e1ban a Streptomyces \u00e1ll. M\u00e1s ritka fajok sz\u00e9lesk\u00f6r\u0171 fejleszt\u00e9si kil\u00e1t\u00e1sokkal rendelkeznek. A pol\u00e1ris aktinomicit\u00e1k \u00e1ltal termelt m\u00e1sodlagos metabolitok k\u00e9miai szerkezeti t\u00edpusai v\u00e1ltozatosak, \u00e9s sokuk j\u00f3 biol\u00f3giai aktivit\u00e1ssal, k\u00fcl\u00f6n\u00f6sen daganatellenes aktivit\u00e1ssal rendelkezik, ami nagy \u00e9rt\u00e9ket k\u00e9pvisel a gy\u00f3gyszerfejleszt\u00e9s szempontj\u00e1b\u00f3l. A metabolitok bioszintetikus \u00fatjainak, akt\u00edv mechanizmusainak \u00e9s klinikai szempontjainak kutat\u00e1s\u00e1t azonban nem v\u00e9gezt\u00e9k el sz\u00e9les k\u00f6rben, \u00e9s a pol\u00e1ris aktinomicit\u00e1kb\u00f3l izol\u00e1lt m\u00e1sodlagos metabolitok t\u00f6bbs\u00e9ge ismert vegy\u00fclet. A bioinformatikai technol\u00f3gia fejl\u0151d\u00e9s\u00e9vel t\u00f6bb pol\u00e1ris aktinomicet\u00e1k genomszekvenci\u00e1j\u00e1t nyert\u00e9k szekven\u00e1l\u00e1ssal, \u00e9s egyre t\u00f6bb pol\u00e1ris aktinomiceta BGC-t fedeztek fel \u00e9s jelentettek be, p\u00e9ld\u00e1ul PKS, NRPS g\u00e9nek, halog\u00e9nezett enzim g\u00e9nek, terp\u00e9n \u00e9s oligoszacharid sz\u00e1rmaz\u00e9kkal kapcsolatos g\u00e9nek stb. L\u00e1that\u00f3, hogy a pol\u00e1ris aktinomicit\u00e1k er\u0151s potenci\u00e1llal rendelkeznek az akt\u00edv m\u00e1sodlagos metabolitok szint\u00e9zis\u00e9ben \u00e9s a pol\u00e1ris k\u00f6rnyezethez val\u00f3 alkalmazkod\u00e1sban, ami gazdagabb \u00e9s v\u00e1ltozatosabb forr\u00e1sokat biztos\u00edt \u00faj vegy\u00fcletekhez az \u00faj gy\u00f3gyszerek fejleszt\u00e9s\u00e9hez. Ugyanakkor az \u00faj m\u00e1sodlagos metabolitok bioszintetikus \u00fatjai k\u00f6nnyebben megfejthet\u0151k lesznek, \u00e9s tov\u00e1bbi kutat\u00e1sra \u00e9s fejleszt\u00e9sre \u00e9rdemesek. B\u00e1r a pol\u00e1ris aktinomyc\u00e9t\u00e1kb\u00f3l izol\u00e1lt vegy\u00fcletek t\u00f6bbs\u00e9ge jelenleg ismert, az \u00faj vegy\u00fcletek bioszint\u00e9zis\u00e9\u00e9rt felel\u0151s \"csendes g\u00e9nek\" nem felt\u00e9tlen\u00fcl fejez\u0151dnek ki a ferment\u00e1ci\u00f3 sor\u00e1n. Ez\u00e9rt a t\u00f6rzsekben a \"csendes g\u00e9nek\" kifejez\u0151d\u00e9s\u00e9t a ferment\u00e1ci\u00f3s k\u00f6r\u00fclm\u00e9nyek optimaliz\u00e1l\u00e1s\u00e1val, mikrobi\u00e1lis ko-kult\u00far\u00e1val \u00e9s m\u00e1s m\u00f3dszerekkel lehet serkenteni. G\u00e9nb\u00e1ny\u00e1szattal, aktivit\u00e1ssz\u0171r\u00e9ssel \u00e9s m\u00e1s m\u00f3dszerekkel kombin\u00e1lva a vegy\u00fcletizol\u00e1l\u00e1s ir\u00e1ny\u00edthat\u00f3, hogy akt\u00edvabb, \u00faj szerkezet\u0171 m\u00e1sodlagos metabolitokat izol\u00e1ljanak a pol\u00e1ris aktinomyc\u00e9ta er\u0151forr\u00e1sokb\u00f3l. A relev\u00e1ns hat\u00e1smechanizmusok tov\u00e1bbi tanulm\u00e1nyoz\u00e1s\u00e1val, a klinikai kutat\u00e1si er\u0151fesz\u00edt\u00e9sek n\u00f6vel\u00e9s\u00e9vel \u00e9s az innovat\u00edv gy\u00f3gyszerek kifejleszt\u00e9s\u00e9nek megalapoz\u00e1s\u00e1val.<\/p>","protected":false},"excerpt":{"rendered":"<p>Research progress on secondary metabolites and pharmacological activities of polar actinomycetes Actinomycete belongs to the phylum Actinobacteria and is a Gram positive bacterium. The secondary metabolites derived from actinomycetes account for about 45% of the secondary metabolites derived from microorganisms, and exhibit a range of biological activities, including anti-tumor, antibacterial, anti-inflammatory, antiviral, and anti angiogenic [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Research progress on secondary metabolites and pharmacological activities of polar actinomycetes - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/hu\/polar-actinomycetes\/\" \/>\n<meta property=\"og:locale\" content=\"hu_HU\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Research progress on secondary metabolites and pharmacological activities of polar actinomycetes - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Research progress on secondary metabolites and pharmacological activities of polar actinomycetes Actinomycete belongs to the phylum Actinobacteria and is a Gram positive bacterium. 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