{"id":5562,"date":"2024-08-04T19:49:08","date_gmt":"2024-08-04T19:49:08","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=5562"},"modified":"2024-08-04T19:49:08","modified_gmt":"2024-08-04T19:49:08","slug":"qigui","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/hu\/qigui\/","title":{"rendered":"A tumorsejtek prolifer\u00e1ci\u00f3j\u00e1nak izol\u00e1l\u00e1sa, tiszt\u00edt\u00e1sa \u00e9s in vitro g\u00e1tl\u00e1sa Qigui poliszacharidok \u00e1ltal"},"content":{"rendered":"<p>A tumorsejtek prolifer\u00e1ci\u00f3j\u00e1nak izol\u00e1l\u00e1sa, tiszt\u00edt\u00e1sa \u00e9s in vitro g\u00e1tl\u00e1sa Qigui poliszacharidok \u00e1ltal<br \/>\nA Huangqi \u00e9s a Danggui kombin\u00e1ci\u00f3ja a klinikai gyakorlatban leggyakrabban haszn\u00e1lt \u00e9s legjellemz\u0151bb toniz\u00e1l\u00f3 qi \u00e9s t\u00e1pl\u00e1l\u00f3 v\u00e9r gy\u00f3gyszer. A hagyom\u00e1nyos k\u00ednai orvosl\u00e1s receptjeinek adatb\u00e1zis\u00e1ban a Huangqi \u00e9s a Danggui k\u00f6z\u00f6tti kompatibilit\u00e1s gyakoris\u00e1ga 2632 alkalommal fordul el\u0151. A Huangqi \u00e9s a Danggui 5:1 ar\u00e1nyban kombin\u00e1lva alkotja a Danggui Buxue Tangot, amely a qi felt\u00f6lt\u00e9s\u00e9re \u00e9s a v\u00e9r el\u0151\u00e1ll\u00edt\u00e1s\u00e1ra szolg\u00e1l\u00f3 j\u00f3l ismert formula. A hagyom\u00e1nyos k\u00ednai orvosl\u00e1s kutat\u00f3i sz\u00e9les k\u00f6rben kedvelik kifinomult formul\u00e1ja \u00e9s pontos ter\u00e1pi\u00e1s hat\u00e1sa miatt. A Qi Gui gy\u00f3gyszerk\u00e9sz\u00edtm\u00e9nyp\u00e1rok alapgy\u00f3gyszerk\u00e9sz\u00edtm\u00e9nyp\u00e1rokk\u00e9nt is haszn\u00e1lhat\u00f3k kombin\u00e1lt k\u00e9pletekben. Nincs olyan formula, mint a Huangqi Danggui Jianzhong Tang, Buzhong Yiqi Tang, Guipi Tang, Shengyu Tang, Buyang Huanwu Tang, amely ne haszn\u00e1lna Qi Gui gy\u00f3gyszerk\u00e9sz\u00edtm\u00e9nyp\u00e1rokat. A klinikai alkalmaz\u00e1sok \u00e9s kutat\u00e1sok legink\u00e1bb erre a gy\u00f3gyszerk\u00e9sz\u00edtm\u00e9nyp\u00e1rra \u00f6sszpontos\u00edtanak. A modern farmakol\u00f3giai kutat\u00e1sok kimutatt\u00e1k, hogy a Qigui gy\u00f3gyszer olyan hat\u00e1sokkal rendelkezik, mint a v\u00e9rk\u00e9pz\u00e9s el\u0151seg\u00edt\u00e9se, immunszab\u00e1lyoz\u00e1s, sz\u00edv- \u00e9s \u00e9rrendszeri v\u00e9delem \u00e9s daganatellenes hat\u00e1sok. A Qigui gy\u00f3gyszer jelent\u0151s daganatellenes hat\u00e1ssal rendelkezik, jelent\u0151s g\u00e1tl\u00f3 hat\u00e1st mutat a vastagb\u00e9lr\u00e1kra, t\u00fcd\u0151r\u00e1kra, leuk\u00e9mi\u00e1ra \u00e9s m\u00e1s r\u00e1kos megbeteged\u00e9sekre.<\/p>\n<p>A poliszacharidok b\u0151s\u00e9gesen el\u0151fordulnak a Qigui gy\u00f3gyn\u00f6v\u00e9nyekben, \u00e9s a Huangqi \u00e9s a Danggui gyakori makromolekul\u00e1ris hat\u00f3anyagai. Olyan hat\u00e1suk van, mint a v\u00e9rszeg\u00e9nys\u00e9g jav\u00edt\u00e1sa, \u00f6reged\u00e9sg\u00e1tl\u00e1s, fibr\u00f3zis \u00e9s daganatellenes hat\u00e1s. A poliszacharidok fontos hat\u00f3anyagok a Qi Gui gy\u00f3gy\u00e1szatban a v\u00e9rp\u00f3tl\u00f3 hat\u00e1s kifejt\u00e9s\u00e9ben. A nem poliszacharid komponensekkel \u00f6sszehasonl\u00edtva a Danggui Buxue Tang poliszacharid komponense er\u0151sebb v\u00e9rp\u00f3tl\u00f3 hat\u00e1ssal rendelkezik, amely jelent\u0151sen el\u0151seg\u00edti a csontvel\u0151 v\u00e9rk\u00e9pz\u0151d\u00e9st, gyors\u00edtja a v\u00e9rsejtek differenci\u00e1l\u00f3d\u00e1s\u00e1t \u00e9s \u00e9r\u00e9s\u00e9t, \u00e9s n\u00f6veli a perif\u00e9ri\u00e1s v\u00f6r\u00f6sv\u00e9rtestek sz\u00e1m\u00e1t v\u00e9rhi\u00e1nyos egerekben. S\u0151t, a Danggui poliszacharidok k\u00fcl\u00f6n\u00f6sen jelent\u0151s v\u00e9rp\u00f3tl\u00f3 hat\u00e1ssal rendelkeznek. A Qigui poliszacharidok fokozhatj\u00e1k az immunrendszer \u00e9s az antioxid\u00e1ns funkci\u00f3kat is, szab\u00e1lyozhatj\u00e1k az \u00f6reged\u0151 sejtciklust \u00e9s a telomer\u00e1z aktivit\u00e1st, k\u00e9sleltethetik a sejtek \u00f6reged\u00e9s\u00e9t, \u00e9s enyh\u00edthetik az oxidat\u00edv k\u00e1rosod\u00e1st az \u00f6reged\u0151 modell egerek vesesz\u00f6vet\u00e9ben. Ezenk\u00edv\u00fcl a Qigui poliszacharidok v\u00e9d\u0151 hat\u00e1ssal vannak a CCl4 \u00e1ltal kiv\u00e1ltott m\u00e1jfibr\u00f3zis-k\u00e1rosod\u00e1sra \u00e9s a ciklofoszfamid \u00e1ltal kiv\u00e1ltott l\u00e9p- \u00e9s t\u00edmuszk\u00e1rosod\u00e1sra. A poliszacharidok a Qigui gy\u00f3gyszer daganatellenes hat\u00e1s\u00e1nak egyik f\u0151 hat\u00f3anyaga, \u00e9s a Huangqi \u00e9s a Danggui poliszacharidjai, amelyek a Qigui gy\u00f3gyszert alkotj\u00e1k, jelent\u0151s g\u00e1tl\u00f3 hat\u00e1ssal vannak a k\u00fcl\u00f6nb\u00f6z\u0151 daganatokra. Az Astragalus poliszacharid jelent\u0151s hat\u00e1ssal van a t\u00fcd\u0151r\u00e1kra, mellr\u00e1kra, melanom\u00e1ra stb. Tumorellenes szerepet j\u00e1tszhat az\u00e1ltal, hogy k\u00f6zvetlen\u00fcl g\u00e1tolja a tumorsejtek prolifer\u00e1ci\u00f3j\u00e1t, apopt\u00f3zist \u00e9s ciklusmeg\u00e1ll\u00e1st induk\u00e1l, aktiv\u00e1lja az immunrendszert \u00e9s szab\u00e1lyozza a gyullad\u00e1sos mikrok\u00f6rnyezetet. Az Angelica poliszacharidok kiemelked\u0151 hat\u00e1ssal vannak a leuk\u00e9mi\u00e1ra, melanom\u00e1ra, vastagb\u00e9lr\u00e1kra, m\u00e1jr\u00e1kra stb. Daganatellenes hat\u00e1st fejthetnek ki a tumorsejtek prolifer\u00e1ci\u00f3j\u00e1nak g\u00e1tl\u00e1s\u00e1val, az apopt\u00f3zis induk\u00e1l\u00e1s\u00e1val, az immunit\u00e1s fokoz\u00e1s\u00e1val, az autof\u00e1gia szab\u00e1lyoz\u00e1s\u00e1val, valamint a tumorsejtek inv\u00e1zi\u00f3j\u00e1nak \u00e9s migr\u00e1ci\u00f3j\u00e1nak g\u00e1tl\u00e1s\u00e1val. Hazai \u00e9s k\u00fclf\u00f6ldi tud\u00f3sok kiterjedt \u00e9s m\u00e9lyrehat\u00f3 kutat\u00e1sokat v\u00e9geztek a Qigui gy\u00f3gyn\u00f6v\u00e9nyp\u00e1rt alkot\u00f3 Huangqi \u00e9s Danggui gy\u00f3gyn\u00f6v\u00e9nyek poliszacharidszerkezet\u00e9vel kapcsolatban. Jelenleg 34 homog\u00e9n poliszacharidot izol\u00e1ltak az Astragalus membranaceusb\u00f3l \u00e9s 39 homog\u00e9n poliszacharidot az Angelica sinensisb\u0151l. E poliszacharidok els\u0151dleges szerkezet\u00e9t, bele\u00e9rtve a molekulat\u00f6meget, a monoszacharid-\u00f6sszet\u00e9telt, a cukormarad\u00e9kok \u00f6sszet\u00e9tel\u00e9t, a glikozidos k\u00f6t\u00e9s konfigur\u00e1ci\u00f3j\u00e1t \u00e9s a kapcsol\u00f3d\u00e1si szekvenci\u00e1t, elemezt\u00e9k. A Qigui poliszacharidok jelenlegi kutat\u00e1sa azonban t\u00f6bbnyire az extrakci\u00f3s folyamat optimaliz\u00e1l\u00e1s\u00e1ra ir\u00e1nyul, \u00e9s kev\u00e9s jelent\u00e9s sz\u00f3l a Qigui homog\u00e9n poliszacharidok kapcsol\u00f3d\u00f3 kutat\u00e1sair\u00f3l. A Qigui-drogok daganatellenes aktivit\u00e1s\u00e1r\u00f3l nem k\u00e9sz\u00fclt szisztematikus tanulm\u00e1ny a poliszacharidokr\u00f3l. Nem k\u00e9sz\u00fcltek jelent\u00e9sek arr\u00f3l, hogy a Qigui gy\u00f3gyszer jelent\u0151s g\u00e1tl\u00f3 hat\u00e1ssal van-e a tumorsejtek prolifer\u00e1ci\u00f3j\u00e1ra az \u00faj szerkezeti poliszacharidban. A kor\u00e1bbi kutat\u00e1sok \u00e9s a vonatkoz\u00f3 irodalmi jelent\u00e9sek alapj\u00e1n ez a tanulm\u00e1ny hatf\u00e9le Astragalus poliszacharidot izol\u00e1lt az Astragalus membranaceus gy\u00f3gyp\u00e1rokb\u00f3l, \u00e9s kiv\u00e1lasztott egyetlen gy\u00f3gyn\u00f6v\u00e9ny Angelica poliszacharidokat vagy Astragalus membranaceus poliszacharidokat, amelyek jelent\u0151s g\u00e1tl\u00f3 hat\u00e1ssal voltak az emberi vastagb\u00e9lr\u00e1ksejtekre HCT116, t\u00fcd\u0151r\u00e1ksejtekre A549 \u00e9s leuk\u00e9mi\u00e1s sejtekre K562. Az Astragalus membranaceus poliszacharidok prolifer\u00e1ci\u00f3t g\u00e1tl\u00f3 \u00e9s apopt\u00f3zist induk\u00e1l\u00f3 hat\u00e1s\u00e1t vizsg\u00e1lt\u00e1k h\u00e1romf\u00e9le tumorsejtre, \u00e9s meg\u00e1llap\u00edtott\u00e1k, hogy k\u00e9tf\u00e9le Astragalus membranaceus poliszacharid jelent\u0151sen g\u00e1tolja a HCT116 \u00e9s A549 sejtek prolifer\u00e1ci\u00f3j\u00e1t \u00e9s apopt\u00f3zist induk\u00e1l. Ez a tanulm\u00e1ny tudom\u00e1nyos alapot ny\u00fajt az \"Astragalus membranaceus poliszacharidokon\" \u00e9s az \"Astragalus membranaceus Angelica gy\u00f3gyp\u00e1ron\" alapul\u00f3, potenci\u00e1lis tumorellenes aktivit\u00e1ssal rendelkez\u0151 eg\u00e9szs\u00e9g\u00fcgyi term\u00e9kek kifejleszt\u00e9s\u00e9hez \u00e9s tov\u00e1bbi alkalmaz\u00e1s\u00e1hoz.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5563\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-156.png\" alt=\"\" width=\"647\" height=\"314\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5564\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-143.png\" alt=\"\" width=\"658\" height=\"253\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5565\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-135.png\" alt=\"\" width=\"659\" height=\"462\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5566\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-121.png\" alt=\"\" width=\"653\" height=\"280\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-121.png 653w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-121-650x280.png 650w\" sizes=\"(max-width: 653px) 100vw, 653px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5567\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-107.png\" alt=\"\" width=\"657\" height=\"173\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5568\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-100.png\" alt=\"\" width=\"656\" height=\"357\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5569\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-91.png\" alt=\"\" width=\"654\" height=\"324\" \/>A poliszacharidok t\u00f6bb monoszacharid egys\u00e9gb\u0151l \u00e1llnak, amelyeket glikozidos k\u00f6t\u00e9sek k\u00f6tnek \u00f6ssze, \u00e9s a term\u00e9szetben az egyik legelterjedtebb \u00e9s legfontosabb biol\u00f3giai polimerek k\u00f6z\u00e9 tartoznak. A shiitake gomba poliszacharidok daganatellenes hat\u00e1s\u00e1r\u00f3l sz\u00f3l\u00f3 els\u0151, 1969-ben a Nature foly\u00f3iratban megjelent besz\u00e1mol\u00f3 \u00f3ta a poliszacharidok gy\u00f3gyszerk\u00e9nt val\u00f3 kutat\u00e1sa \u00e9s alkalmaz\u00e1sa sz\u00e9les k\u00f6r\u0171 figyelmet keltett a hazai \u00e9s k\u00fclf\u00f6ldi tud\u00f3sok k\u00f6r\u00e9ben. A hagyom\u00e1nyos k\u00ednai orvosl\u00e1s poliszacharidjai kiemelked\u0151 farmakol\u00f3giai aktivit\u00e1ssal rendelkeznek az immunszab\u00e1lyoz\u00e1s, a daganatellenes, a cukorbetegs\u00e9g elleni, az oxid\u00e1ci\u00f3 elleni, a v\u00edrusellenes, a sz\u00edv- \u00e9s \u00e9rrendszeri v\u00e9delem \u00e9s a neuroprotekt\u00edv tev\u00e9kenys\u00e9gek ter\u00e9n, \u00e9s az ut\u00f3bbi \u00e9vekben a hagyom\u00e1nyos k\u00ednai orvosl\u00e1s hat\u00f3anyagainak kutat\u00e1si ter\u00fclet\u00e9n forr\u00f3 pontok. Jelenleg a hagyom\u00e1nyos k\u00ednai gy\u00f3gyszerekb\u0151l, p\u00e9ld\u00e1ul a Ganoderma lucidumb\u00f3l, a ginzengb\u0151l, az astragalusb\u00f3l, az Angelica sinensisb\u0151l \u00e9s a farkasbogy\u00f3b\u00f3l t\u00f6bb sz\u00e1z, jelent\u0151s farmakol\u00f3giai hat\u00e1ssal rendelkez\u0151, nagy tisztas\u00e1g\u00fa \"akt\u00edv poliszacharidot\" nyertek.<br \/>\nAz egy \u00f6sszetev\u0151b\u0151l \u00e1ll\u00f3 poliszacharidokkal \u00f6sszehasonl\u00edtva az \u00f6sszetett poliszacharidok k\u00e9pesek egyes\u00edteni a k\u00fcl\u00f6nb\u00f6z\u0151 egy \u00f6sszetev\u0151b\u0151l \u00e1ll\u00f3 poliszacharidok biol\u00f3giai aktivit\u00e1s\u00e1t, hogy szinergikus hat\u00e1st \u00e9rjenek el. Ezenk\u00edv\u00fcl a vegyes poliszacharidokat befoly\u00e1solj\u00e1k a gy\u00f3gy\u00e1szati anyagok forr\u00e1sa, a feldolgoz\u00e1si technik\u00e1k, a kompatibilit\u00e1si hat\u00e1sok \u00e9s az extrakci\u00f3s m\u00f3dszerek, \u00e9s tisztas\u00e1guk \u00e9s szerkezeti jellemz\u0151ik elt\u00e9rnek az egyn\u00f6v\u00e9nyes poliszacharidok\u00e9t\u00f3l. A hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szatban haszn\u00e1lt \u00f6sszetett poliszacharidok hat\u00e9kony \u00e9s teljes elk\u00fcl\u00f6n\u00edt\u00e9se \u00e9s tiszt\u00edt\u00e1sa az egyn\u00f6v\u00e9ny\u0171 poliszacharidok kutat\u00e1s\u00e1n alapulva, valamint szerkezeti alapjaik \u00e9s hat\u00e1smechanizmusuk tiszt\u00e1z\u00e1sa az ut\u00f3bbi \u00e9vekben a k\u00ednai gy\u00f3gy\u00e1szati hat\u00f3anyagok tanulm\u00e1nyoz\u00e1s\u00e1nak egyik forr\u00f3 pontj\u00e1v\u00e1 \u00e9s neh\u00e9zs\u00e9g\u00e9v\u00e9 v\u00e1lt. A hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szati formul\u00e1kb\u00f3l, p\u00e9ld\u00e1ul a Sijunzi Tangb\u00f3l nyert egys\u00e9ges poliszacharidszerkezet elt\u00e9r az egyes gy\u00f3gyn\u00f6v\u00e9ny-poliszacharidok\u00e9t\u00f3l. A kutat\u00e1sok azt tal\u00e1lt\u00e1k, hogy a Qigui gy\u00f3gyszer jelent\u0151s daganatellenes aktivit\u00e1ssal rendelkezik a poliszacharidokkal szemben, de a Qigui poliszacharidok szerkezeti alapja \u00e9s hat\u00e1smechanizmusa a daganatellenes kezel\u00e9sben m\u00e9g mindig nem vil\u00e1gos. Nem sz\u00e1moltak be arr\u00f3l, hogy a Qigui gy\u00f3gyszerben l\u00e9v\u0151 poliszacharid komponensek szerkezete \u00e9s aktivit\u00e1sa k\u00fcl\u00f6nb\u00f6zik-e az egyes gy\u00f3gyn\u00f6v\u00e9nyek\u00e9t\u0151l. Ebben a tanulm\u00e1nyban az Astragalus membranaceusb\u00f3l izol\u00e1lt\u00e1k az Astragalus membranaceus teljes poliszacharidjait (AAPS), \u00e9s vizsg\u00e1lt\u00e1k a tumorsejtek prolifer\u00e1ci\u00f3j\u00e1t g\u00e1tl\u00f3 hat\u00e1sukat. Meg\u00e1llap\u00edtott\u00e1k, hogy az AAPS jelent\u0151s g\u00e1tl\u00f3 hat\u00e1ssal van a vastagb\u00e9lr\u00e1ksejtek prolifer\u00e1ci\u00f3j\u00e1ra. Az AAPS tov\u00e1bbi elv\u00e1laszt\u00e1sa \u00e9s tiszt\u00edt\u00e1sa ut\u00e1n meg\u00e1llap\u00edtott\u00e1k, hogy a Qigui poliszacharidok k\u00e9t t\u00edpusa, az AAPS-1a \u00e9s az AAPS-3a jelent\u0151sen g\u00e1tolja a HCT116 hum\u00e1n vastagb\u00e9lr\u00e1k-sejtvonal \u00e9s az A549 t\u00fcd\u0151r\u00e1k-sejtvonal prolifer\u00e1ci\u00f3j\u00e1t, \u00e9s apopt\u00f3zist induk\u00e1l. Az el\u0151zetes szerkezeti elemz\u00e9s azt mutatja, hogy az AAPS-1a \u00e9s az AAPS-3a a Qigui homog\u00e9n poliszacharidjai, amelyek molekulat\u00f6mege 7,3 \u00d7 105, illetve 8,5 \u00d7 104 Da. \u00d6sszefoglalva, az AAPS-1a \u00e9s az AAPS-3a akt\u00edv Qigui homog\u00e9n poliszacharidok, amelyek potenci\u00e1lis daganatellenes hat\u00e1ssal rendelkeznek. Ez a tanulm\u00e1ny kutat\u00e1si alapot ny\u00fajt a Qigui poliszacharidok daganatellenes anyagalapj\u00e1nak \u00e9s szerkezet-hat\u00e1s kapcsolat\u00e1nak k\u00e9s\u0151bbi vizsg\u00e1lat\u00e1hoz, \u00e9s fontos m\u00f3dszereket, \u00f6tleteket \u00e9s k\u00eds\u00e9rleti bizony\u00edt\u00e9kokat szolg\u00e1ltat a hagyom\u00e1nyos k\u00ednai gy\u00f3gyszerk\u00e9sz\u00edtm\u00e9nyek makromolekul\u00e1ris anyagalapj\u00e1nak kutat\u00e1s\u00e1hoz.<\/p>","protected":false},"excerpt":{"rendered":"<p>Isolation, purification, and in vitro inhibition of tumor cell proliferation by Qigui polysaccharides The combination of Huangqi and Danggui is the most commonly used and representative tonifying qi and nourishing blood medicine in clinical practice. 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