{"id":5377,"date":"2024-08-04T18:38:02","date_gmt":"2024-08-04T18:38:02","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=5377"},"modified":"2024-08-04T18:38:02","modified_gmt":"2024-08-04T18:38:02","slug":"lamiophlomis","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/hu\/lamiophlomis\/","title":{"rendered":"Az Angelica sinensisb\u0151l sz\u00e1rmaz\u00f3 \u00f6sszes flavonoid kulcskomponens\u00e9nek felt\u00e1r\u00e1sa az anti-reumatoid artritiszben a spektr\u00e1lis hat\u00e1skapcsolat \u00e9s a komponensek ki\u00fct\u00e9se alapj\u00e1n"},"content":{"rendered":"<p>Az Angelica sinensisb\u0151l sz\u00e1rmaz\u00f3 \u00f6sszes flavonoid kulcskomponens\u00e9nek felt\u00e1r\u00e1sa az anti-reumatoid artritiszben a spektr\u00e1lis hat\u00e1skapcsolat \u00e9s a komponensek ki\u00fct\u00e9se alapj\u00e1n<br \/>\nA Lamiophlomis Herba (LH), egy hagyom\u00e1nyos k\u00ednai gy\u00f3gyszer, a Lamiaceae csal\u00e1dba tartoz\u00f3 Lamiophlomis rotata (Benth.) Kudo n\u00f6v\u00e9ny sz\u00e1r\u00edtott f\u00f6ld feletti r\u00e9sze. A tibetiek \u00e1ltal\u00e1nosan haszn\u00e1lt gy\u00f3gyn\u00f6v\u00e9ny, amelyet hagyom\u00e1nyos k\u00ednai gy\u00f3gyszerk\u00e9nt is gyakran alkalmaznak. A K\u00ednai N\u00e9pk\u00f6zt\u00e1rsas\u00e1g gy\u00f3gyszerk\u00f6nyv\u00e9nek 2020-as kiad\u00e1sa szerint a v\u00e9rkering\u00e9st el\u0151seg\u00edt\u0151, v\u00e9rz\u00e9scsillap\u00edt\u00f3, sz\u00e9l\u0171z\u0151 \u00e9s f\u00e1jdalomcsillap\u00edt\u00f3 hat\u00e1s\u00fa. Haszn\u00e1lhat\u00f3 es\u00e9sek okozta s\u00e9r\u00fcl\u00e9sek, reuma \u00e9s s\u00e1rgav\u00edz-betegs\u00e9g kezel\u00e9s\u00e9re. Tibeti gy\u00f3gy\u00e1szati neve \"Daba\" \u00e9s \"Dabuba\", amelyeket olyan tibeti orvosi m\u0171vekben jegyeztek fel, mint a \"Yue Wang Yao Jian\", \"Four Medical Classics\", \"Jing Zhu Ben Cao\" stb. Alkalmaz\u00e1s\u00e1nak t\u00f6rt\u00e9nete eddig 1200 \u00e9vre ny\u00falik vissza; a \"Jingzhu Bencao\" feljegyzi, hogy \"a Du Yi Wei megszil\u00e1rd\u00edtja az esszenci\u00e1t \u00e9s elvezeti a s\u00e1rga vizet\", ami azt jelzi, hogy a Du Yi Wei haszn\u00e1lhat\u00f3 a \"s\u00e1rga v\u00edz betegs\u00e9g\" kezel\u00e9s\u00e9re. A klinikai megnyilv\u00e1nul\u00e1sok alapj\u00e1n a tibeti orvosl\u00e1sban feljegyzett \"s\u00e1rga v\u00edz betegs\u00e9g\" a hagyom\u00e1nyos k\u00ednai orvosl\u00e1sban a \"bi szindr\u00f3m\u00e1hoz\" sorolhat\u00f3. A \"bi szindr\u00f3m\u00e1b\u00f3l\" kialakult \"csont bi\" \u00e9s \"li jie betegs\u00e9g\" szorosabban kapcsol\u00f3dik a modern orvostudom\u00e1nyban a \"reumatoid artritisz (RA)\" klinikai jellemz\u0151ihez. Ez\u00e9rt a Du Yi Wei alkalmas az RA kezel\u00e9s\u00e9re, \u00e9s a megl\u00e9v\u0151 kutat\u00e1sok azt is kimutatt\u00e1k, hogy a Du Yi Wei RA-ellenes hat\u00e1ssal rendelkezik.<br \/>\nAz RA egy autoimmun betegs\u00e9g, amelyet kr\u00f3nikus \u00e9s t\u00f6bbsz\u00f6r\u00f6s \u00edz\u00fcleti gyullad\u00e1sok jellemeznek. Patol\u00f3giai jellemz\u0151i k\u00f6z\u00e9 tartozik a synovialis sejtek tumorszer\u0171 burj\u00e1nz\u00e1sa \u00e9s az \u00e9rhom\u00e1lyok kialakul\u00e1sa, a fibroblasztszer\u0171 synoviocit\u00e1k (FLS) a f\u0151 effektor sejtek. Az RA patogenezise jelenleg m\u00e9g mindig nem tiszt\u00e1zott. El\u0151fordul\u00e1si ar\u00e1nya \u00e9s rokkants\u00e1gi ar\u00e1nya magas, \u00e9s \u00e1ltal\u00e1ban l\u00e1tens. A betegs\u00e9g k\u00e9s\u0151i st\u00e1dium\u00e1ban k\u00fcl\u00f6nb\u00f6z\u0151 m\u00e9rt\u00e9k\u0171 irreverzibilis rokkants\u00e1ghoz vezethet, amely az Eg\u00e9szs\u00e9g\u00fcgyi Vil\u00e1gszervezet \u00e1ltal meghat\u00e1rozott modern refrakter betegs\u00e9g. A klinikai gyakorlatban az RA kezel\u00e9s\u00e9re \u00e1ltal\u00e1nosan haszn\u00e1lt k\u00e9miai gy\u00f3gyszerek k\u00f6z\u00e9 tartoznak a nem szteroid gyullad\u00e1scs\u00f6kkent\u0151k, az immunszuppressz\u00e1nsok, a gl\u00fckokortikoidok \u00e9s a biol\u00f3gikumok. Az els\u0151 h\u00e1rom k\u00e9miai gy\u00f3gyszer jelent\u0151s mell\u00e9khat\u00e1sokkal j\u00e1r, m\u00edg a biol\u00f3giai szerek dr\u00e1ga \u00e1ra korl\u00e1tozza hossz\u00fa t\u00e1v\u00fa alkalmaz\u00e1sukat. Ez\u00e9rt k\u00fcl\u00f6n\u00f6sen sz\u00fcks\u00e9ges \u00faj, alacsony mell\u00e9khat\u00e1sokkal \u00e9s stabil ter\u00e1pi\u00e1s hat\u00e1ssal rendelkez\u0151 klinikai RA-ellenes gy\u00f3gyszerek kifejleszt\u00e9se.<br \/>\nA kutat\u00f3csoport el\u0151sz\u00f6r alkalmazta a h\u00e1l\u00f3zati farmakol\u00f3gi\u00e1t a Du Yi Wei farmakol\u00f3giai hat\u00f3anyag-alapj\u00e1nak \u00e9s hat\u00e1smechanizmus\u00e1nak felt\u00e1r\u00e1s\u00e1ra az RA kezel\u00e9s\u00e9ben. Meg\u00e1llap\u00edtott\u00e1k, hogy a Du Yi Wei RA-ra gyakorolt ter\u00e1pi\u00e1s hat\u00e1sa 23 \u00f6sszetev\u0151j\u00e9hez kapcsol\u00f3dik, amelyek k\u00f6z\u00fcl a flavonoidok k\u00f6zel 40%-t tesznek ki, ami azt jelzi, hogy a flavonoidok fontos szerepet j\u00e1tszanak a Du Yi Wei RA-ellenes folyamat\u00e1ban, k\u00fcl\u00f6n\u00f6sen a luteolin; \u00c9s azt javasolj\u00e1k, hogy a Du Yi Wei RA-ellenes hat\u00e1s\u00e1nak f\u0151 mechanizmusa a PI3K Akt jel\u00e1tviteli \u00fatvonal g\u00e1tl\u00e1s\u00e1val a szinovi\u00e1lis sejtek apopt\u00f3zis\u00e1nak kiv\u00e1lt\u00e1sa lehet. Ek\u00f6zben a Du Yi Wei anti-RA hat\u00e1s\u00e1t \u00e9s farmakol\u00f3giai anyag\u00e1nak alapj\u00e1t patk\u00e1ny adjuv\u00e1ns artritisz modellen kereszt\u00fcl vizsg\u00e1lt\u00e1k, \u00e9s az eredm\u00e9nyek azt mutatt\u00e1k, hogy a Du Yi Wei \u00f6sszes flavonoidja j\u00f3 anti-RA hat\u00e1ssal rendelkezik. A Du Yi Wei \u00f6sszes flavonoidja lehet az egyik f\u0151 farmakol\u00f3giai anyag az anti RA hat\u00e1s\u00e9rt, de a Du Yi Wei \u00f6sszes flavonoidj\u00e1nak kulcsfontoss\u00e1g\u00fa anti RA \u00f6sszetev\u0151i m\u00e9g mindig nem tiszt\u00e1zottak \u00e9s tov\u00e1bbi kutat\u00e1st ig\u00e9nyelnek. Ez\u00e9rt e tanulm\u00e1ny c\u00e9lja az Angelica sinensis \u00f6sszes flavonoidj\u00e1ban l\u00e9v\u0151 kulcsfontoss\u00e1g\u00fa RA-ellenes komponensek felt\u00e1r\u00e1sa spektr\u00e1lis hat\u00e1skapcsolatok \u00e9s komponens knockout technik\u00e1k seg\u00edts\u00e9g\u00e9vel, azzal a c\u00e9llal, hogy elm\u00e9leti alapot \u00e9s hivatkoz\u00e1si alapot biztos\u00edtson az Angelica sinensis klinikai alkalmaz\u00e1s\u00e1hoz az RA kezel\u00e9s\u00e9ben.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5378\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-140.png\" alt=\"\" width=\"662\" height=\"337\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5379\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-127.png\" alt=\"\" width=\"656\" height=\"217\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5380\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-120.png\" alt=\"\" width=\"655\" height=\"333\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5381\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-108.png\" alt=\"\" width=\"651\" height=\"329\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5382\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-97.png\" alt=\"\" width=\"327\" height=\"453\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5383\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-90.png\" alt=\"\" width=\"333\" height=\"281\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5384\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-80.png\" alt=\"\" width=\"653\" height=\"230\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-80.png 653w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-80-650x230.png 650w\" sizes=\"(max-width: 653px) 100vw, 653px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5385\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-75.png\" alt=\"\" width=\"643\" height=\"237\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5386\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-68.png\" alt=\"\" width=\"650\" height=\"299\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5387\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-56.png\" alt=\"\" width=\"658\" height=\"192\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5388\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-50.png\" alt=\"\" width=\"321\" height=\"214\" \/><\/p>\n<p>Megbesz\u00e9l\u00e9s \u00e9s k\u00f6vetkeztet\u00e9s<br \/>\nAz Angelica sinensisben tal\u00e1lhat\u00f3 \u00f6sszes flavonoidok ujjlenyomat\u00e1nak el\u0151zetes vizsg\u00e1lat\u00e1t nagy teljes\u00edtm\u00e9ny\u0171 folyad\u00e9kkromatogr\u00e1fi\u00e1s di\u00f3dasoros detektorral (HPLC-DAD) v\u00e9gezt\u00fck. Az Angelica sinensis \u00f6sszes flavonoidmint\u00e1k egyes t\u00e9teleinek ujjlenyomat-spektrumai \u00e9s a meg\u00e1llap\u00edtott kontroll-ujjlenyomat-spektrumok k\u00f6z\u00f6tti hasonl\u00f3s\u00e1g nagyobb volt, mint 0,9, ami azt jelzi, hogy az Angelica sinensis \u00f6sszes flavonoidmint\u00e1k k\u00fcl\u00f6nb\u00f6z\u0151 t\u00e9teleiben tal\u00e1lhat\u00f3 k\u00e9miai komponensek konzisztensek voltak. A kutat\u00f3csoport megvizsg\u00e1lta az Angelica sinensisben l\u00e9v\u0151 \u00f6sszes flavonoidok k\u00fcl\u00f6nb\u00f6z\u0151 koncentr\u00e1ci\u00f3inak \u00e9s bead\u00e1si idej\u00e9nek hat\u00e1s\u00e1t az FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9re a korai szakaszban. Ennek alapj\u00e1n a CCK-8 m\u00f3dszerrel 64 \u03bc g\/ml koncentr\u00e1ci\u00f3ban 48 \u00f3r\u00e1n kereszt\u00fcl kezelt\u00e9k az FLS sejteket, hogy megvizsg\u00e1lj\u00e1k az Angelica sinensisben l\u00e9v\u0151 \u00f6sszes flavonoidok k\u00fcl\u00f6nb\u00f6z\u0151 t\u00e9teleinek az FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9re gyakorolt hat\u00e1s\u00e1t. Az eredm\u00e9nyek azt mutatt\u00e1k, hogy az Angelica sinensisben tal\u00e1lhat\u00f3 \u00f6sszes flavonoidok mind a 13 t\u00e9tele jelent\u0151sen g\u00e1tolni tudta az FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9t. Az Angelica sinensisben l\u00e9v\u0151 \u00f6sszes flavonoidok ujjlenyomat-spektruma \u00e9s a sejthat\u00e9konys\u00e1gi k\u00eds\u00e9rletek eredm\u00e9nyei alapj\u00e1n sz\u00fcrke rel\u00e1ci\u00f3s anal\u00edzist \u00e9s r\u00e9szleges legkisebb n\u00e9gyzetek (PLS) regresszi\u00f3anal\u00edzist alkalmaztunk az Angelica sinensisben l\u00e9v\u0151 \u00f6sszes flavonoidok spektrum-hat\u00e1s kapcsolat\u00e1nak meg\u00e1llap\u00edt\u00e1s\u00e1ra az RA ellen. Az eredm\u00e9nyek azt mutatt\u00e1k, hogy az Angelica sinensis \u00f6sszes flavonoidj\u00e1ban a verbaszkozid \u00e9s a verbaszkozid komponensei jelent\u0151s szerepet j\u00e1tszottak az RA elleni hat\u00e9konys\u00e1gban. A v\u00e9konyr\u00e9teg-kromatogr\u00e1fia alapj\u00e1n az Angelica sinensis \u00f6sszes flavonoidj\u00e1nak magas verbaszkozid-tartalm\u00e1t hat\u00e9konyan kiiktatt\u00e1k, \u00e9s az egyes mint\u00e1k FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9re gyakorolt hat\u00e1s\u00e1t CCK-8 m\u00f3dszerrel hat\u00e1rozt\u00e1k meg. Az eredm\u00e9nyek azt mutatt\u00e1k, hogy a teljes komponens \u00e9s a c\u00e9lkomponens mint\u00e1k jelent\u0151sen g\u00e1tolni tudt\u00e1k az FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9t, m\u00edg a negat\u00edv c\u00e9lkomponens minta nem gyakorolt jelent\u0151s g\u00e1tl\u00f3 hat\u00e1st az FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9re. Ugyanakkor \u00f6sszehasonl\u00edtottuk a verbaszkozid \u00e9s a verbaszkozid ekvimol\u00e1ris mennyis\u00e9g\u00e9nek az RA-FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9re gyakorolt hat\u00e1s\u00e1t. Az eredm\u00e9nyek azt mutatt\u00e1k, hogy mind a verbaszkozid, mind a verbaszkozid szignifik\u00e1nsan g\u00e1tolni tudta az FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9t, de a verbaszkozid csoport \u00e9s a verbaszkozid csoport k\u00f6z\u00f6tt nem volt szignifik\u00e1ns k\u00fcl\u00f6nbs\u00e9g.<br \/>\n\u00d6sszefoglalva, e vizsg\u00e1lat eredm\u00e9nyei azt mutatj\u00e1k, hogy a verbaszkozid \u00e9s a verbaszkozid \u00f6sszetev\u0151i jelent\u0151s szerepet j\u00e1tszanak az Angelica sinensis \u00f6sszes flavonoidj\u00e1nak RA-ellenes hat\u00e9konys\u00e1g\u00e1ban. Az Angelica sinensisben l\u00e9v\u0151 \u00f6sszes flavonoidok ujjlenyomat-elemz\u00e9s\u00e9vel kombin\u00e1lva a verbaszkozid tartalma jelent\u0151sen magasabb, mint a verbaszkozid\u00e9, ami azt jelzi, hogy a verbaszkozid (C21H20O11) az Angelica sinensisben l\u00e9v\u0151 \u00f6sszes flavonoidok kulcsfontoss\u00e1g\u00fa \u00f6sszetev\u0151je az anti RA szempontj\u00e1b\u00f3l. Ez tudom\u00e1nyos alapot ny\u00fajthat a Du Yi Wei-b\u0151l sz\u00e1rmaz\u00f3 \u00f6sszes flavonoidok klinikai alkalmaz\u00e1s\u00e1hoz az RA kezel\u00e9s\u00e9ben. Az ozmanthus glikozidok sz\u00e9les k\u00f6rben jelen vannak k\u00fcl\u00f6nb\u00f6z\u0151 gy\u00f3gyn\u00f6v\u00e9nyekben, \u00e9s jelent\u0151s hat\u00e1ssal rendelkeznek gyullad\u00e1scs\u00f6kkent\u0151, antioxid\u00e1ns, r\u00e1kellenes \u00e9s hipoglik\u00e9mi\u00e1s szempontb\u00f3l, minim\u00e1lis toxikus mell\u00e9khat\u00e1sokkal. B\u00e1r a verbaszkozid komponensei viszonylag gyakoriak, a verbaszkozid RA-ellenes hat\u00e1sair\u00f3l jelenleg nincs elegend\u0151 irodalom. Ebben a tanulm\u00e1nyban a CCK-8 m\u00f3dszert haszn\u00e1lt\u00e1k a verbaszkozid RA-FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9re gyakorolt hat\u00e1s\u00e1nak vizsg\u00e1lat\u00e1ra, \u00e9s egy\u00e9rtelm\u0171en kimutatt\u00e1k, hogy a verbaszkozid g\u00e1tl\u00f3 hat\u00e1ssal van az FLS sejtek \u00e9letk\u00e9pess\u00e9g\u00e9re. Ezt k\u00f6vet\u0151en egy patk\u00e1ny artritisz modellt lehet l\u00e9trehozni az in vivo hat\u00e9konys\u00e1g ellen\u0151rz\u00e9s\u00e9re, \u00e9s a hat\u00e1smechanizmusa megmagyar\u00e1zhat\u00f3, ami t\u00f6bb hivatkoz\u00e1st \u00e9s alapot biztos\u00edt az Angelica sinensis teljes flavonoidjainak klinikai alkalmaz\u00e1s\u00e1hoz az RA kezel\u00e9s\u00e9ben.<\/p>","protected":false},"excerpt":{"rendered":"<p>Az Angelica sinensisb\u0151l sz\u00e1rmaz\u00f3 \u00f6sszes flavonoid kulcskomponens\u00e9nek felt\u00e1r\u00e1sa a reum\u00e1s \u00edz\u00fcleti gyullad\u00e1s ellen\u00e9ben spektr\u00e1lis hat\u00e1skapcsolat \u00e9s komponens-kies\u00e9s alapj\u00e1n A Lamiophlomis Herba (LH), egy hagyom\u00e1nyos k\u00ednai gy\u00f3gyszer, a Lamiophlomis rotata (Benth.) Kudo, a Lamiaceae csal\u00e1dba tartoz\u00f3 n\u00f6v\u00e9ny sz\u00e1r\u00edtott f\u00f6ld feletti r\u00e9sze. A tibetiek \u00e9s a [...]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Exploring the key components of total flavonoids from Angelica sinensis in anti rheumatoid arthritis based on spectral effect relationship and component knockout - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/hu\/lamiophlomis\/\" \/>\n<meta property=\"og:locale\" content=\"hu_HU\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Exploring the key components of total flavonoids from Angelica sinensis in anti rheumatoid arthritis based on spectral effect relationship and component knockout - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Exploring the key components of total flavonoids from Angelica sinensis in anti rheumatoid arthritis based on spectral effect relationship and component knockout Lamiophlomis Herba (LH), a traditional Chinese medicine, is the dried aboveground part of Lamiophlomis rotata (Benth.) Kudo, a plant in the family Lamiaceae. 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