{"id":5231,"date":"2024-08-04T17:55:12","date_gmt":"2024-08-04T17:55:12","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=5231"},"modified":"2024-08-04T17:55:12","modified_gmt":"2024-08-04T17:55:12","slug":"bletilla-striata","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/hu\/bletilla-striata\/","title":{"rendered":"A Bai Ji Zhong k\u00e9miai \u00f6sszetev\u0151inek azonos\u00edt\u00e1sa \u00e9s a Staphylococcus aureus g\u00e1tl\u00e1si mechanizmus\u00e1nak vizsg\u00e1lata"},"content":{"rendered":"<p>A Bai Ji Zhong k\u00e9miai \u00f6sszetev\u0151inek azonos\u00edt\u00e1sa \u00e9s a Staphylococcus aureus g\u00e1tl\u00e1si mechanizmus\u00e1nak vizsg\u00e1lata<br \/>\nAz antibiotikumokat a 20. sz\u00e1zad \"csodaszereinek\" tartj\u00e1k. Az antibiotikumok t\u00falzott emberi felhaszn\u00e1l\u00e1sa miatt azonban a bakt\u00e9riumok rezisztenci\u00e1ja kialakult. V\u00e1rhat\u00f3an 2050-re a bakteri\u00e1lis fert\u0151z\u00e9sek \u00e1ltal az embereknek okozott glob\u00e1lis vagyoni vesztes\u00e9gek el\u00e9rik az $100 billi\u00f3 forintot. A Staphylococcus aureus egy gyakori, \u00e9lelmiszerrel terjed\u0151 patog\u00e9n bakt\u00e9rium, amely l\u00e9g\u00fati, em\u00e9szt\u0151rendszeri \u00e9s h\u00fagy\u00fati fert\u0151z\u00e9seket okozhat. Jelenleg a klinikai gyakorlatban haszn\u00e1lt antibakteri\u00e1lis gy\u00f3gyszerekkel olyan probl\u00e9m\u00e1k vannak, mint a korl\u00e1tozott szerkezeti t\u00edpusok, a gyakori toxikus mell\u00e9khat\u00e1sok \u00e9s a n\u00f6vekv\u0151 gy\u00f3gyszerrezisztencia. Ez\u00e9rt s\u00fcrg\u0151sen sz\u00fcks\u00e9g van \u00faj t\u00edpus\u00fa antibakteri\u00e1lis gy\u00f3gyszerek kifejleszt\u00e9s\u00e9re.<br \/>\nA term\u00e9szetes term\u00e9keket m\u00e9g mindig az \u00faj gy\u00f3gyszerek felfedez\u00e9s\u00e9nek kincsesb\u00e1ny\u00e1j\u00e1nak tekintik. Az amerikai \u00c9lelmiszer- \u00e9s Gy\u00f3gyszer\u00fcgyi Hivatal (FDA) szerint a klinikai gy\u00f3gyszerek t\u00f6bb mint fele term\u00e9szetes term\u00e9kekb\u0151l vagy azok szintetikus sz\u00e1rmaz\u00e9kaib\u00f3l sz\u00e1rmazik, \u00e9s mintegy 200 mikrobi\u00e1lis forr\u00e1sb\u00f3l sz\u00e1rmaz\u00f3 term\u00e9szetes antibiotikumot haszn\u00e1lnak k\u00f6zvetlen\u00fcl gy\u00f3gyszerk\u00e9nt.<br \/>\nA Baiji, m\u00e1s n\u00e9ven j\u00e1cint orchidea, j\u00e1cint baiji vagy Ulan, gum\u00f3it gyakran haszn\u00e1lj\u00e1k gy\u00f3gy\u00e1szati r\u00e9szekk\u00e9nt. \u00cdze \u00e9des, keser\u0171 \u00e9s fanyar, enyh\u00e9n hideg jelleg\u0171. Hat\u00e1sai: \u00f6sszeh\u00faz\u00f3, v\u00e9rz\u00e9scsillap\u00edt\u00f3, duzzanatcs\u00f6kkent\u0151 \u00e9s izomregener\u00e1l\u00f3. Gyakran haszn\u00e1lj\u00e1k felk\u00f6h\u00f6g\u00e9s \u00e9s v\u00e9rh\u00e1ny\u00e1s, k\u00fcls\u0151 v\u00e9rz\u00e9s, fek\u00e9lyek \u00e9s m\u00e9rgek, b\u0151rreped\u00e9s, fek\u00e9lyv\u00e9rz\u00e9s stb. kezel\u00e9s\u00e9re. F\u0151 \u00f6sszetev\u0151i k\u00f6z\u00e9 tartoznak a poliszacharidok, fenantr\u00e9n, fenantr\u00e9nkinon, dibenzol, triterpenoidok, lign\u00e1nok \u00e9s szerves savak. Farmakol\u00f3giai vizsg\u00e1latok kimutatt\u00e1k, hogy a Bai Ji k\u00fcl\u00f6nb\u00f6z\u0151 biol\u00f3giai aktivit\u00e1sokkal rendelkezik, mint p\u00e9ld\u00e1ul gyullad\u00e1scs\u00f6kkent\u0151, fibr\u00f3zisellenes, tumorellenes \u00e9s immunszab\u00e1lyoz\u00f3 hat\u00e1s\u00fa, de kev\u00e9s jelent\u00e9s sz\u00f3l antibakteri\u00e1lis mechanizmus\u00e1r\u00f3l. Ez\u00e9rt ebben a k\u00eds\u00e9rletben a Staphylococcus aureus-t v\u00e1lasztottuk kutat\u00e1si t\u00e1rgynak, hogy megvizsg\u00e1ljuk a kivonat \u00e9s a monomer vegy\u00fclet antibakteri\u00e1lis aktivit\u00e1sa k\u00f6z\u00f6tti k\u00fcl\u00f6nbs\u00e9get. Az alkalikus foszfat\u00e1z (AKP), a DNS-sziv\u00e1rg\u00e1s m\u00e9rt\u00e9k\u00e9nek \u00e9s a bakteri\u00e1lis elektronmikroszk\u00f3pos morfol\u00f3gi\u00e1nak a bakt\u00e9riumoldatban t\u00f6rt\u00e9n\u0151 m\u00e9r\u00e9s\u00e9vel vizsg\u00e1lt\u00e1k a vegy\u00fclet hat\u00e1s\u00e1t a Staphylococcus aureus sejtmembr\u00e1nfal\u00e1ra, elm\u00e9leti alapot szolg\u00e1ltatva a Staphylococcus aureus \u00e1tfog\u00f3 felhaszn\u00e1l\u00e1s\u00e1hoz \u00e9s \u00faj antibakteri\u00e1lis szerek kifejleszt\u00e9s\u00e9hez.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5232\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-128.png\" alt=\"\" width=\"774\" height=\"262\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-128.png 774w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-128-768x260.png 768w\" sizes=\"(max-width: 774px) 100vw, 774px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5233\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-115.png\" alt=\"\" width=\"777\" height=\"302\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-115.png 777w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-115-768x299.png 768w\" sizes=\"(max-width: 777px) 100vw, 777px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5234\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-109.png\" alt=\"\" width=\"776\" height=\"269\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-109.png 776w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-109-768x266.png 768w\" sizes=\"(max-width: 776px) 100vw, 776px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5235\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-97.png\" alt=\"\" width=\"772\" height=\"282\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-97.png 772w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-97-768x281.png 768w\" sizes=\"(max-width: 772px) 100vw, 772px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5236\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-89.png\" alt=\"\" width=\"775\" height=\"209\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-89.png 775w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-89-768x207.png 768w\" sizes=\"(max-width: 775px) 100vw, 775px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5237\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-82.png\" alt=\"\" width=\"777\" height=\"207\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-82.png 777w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-82-768x205.png 768w\" sizes=\"(max-width: 777px) 100vw, 777px\" \/>Ez a k\u00eds\u00e9rlet az antibakteri\u00e1lis aktivit\u00e1sra \u00f6sszpontos\u00edt, \u00e9s kromatogr\u00e1fi\u00e1s elv\u00e1laszt\u00e1si technol\u00f3gi\u00e1t alkalmaz a Baiji hagyom\u00e1nyos k\u00ednai gy\u00f3gyszer k\u00e9miai \u00f6sszetev\u0151inek izol\u00e1l\u00e1s\u00e1ra \u00e9s tiszt\u00edt\u00e1s\u00e1ra. \u00d6sszesen 10 vegy\u00fcletet (1-10) izol\u00e1ltunk \u00e9s azonos\u00edtottunk, k\u00f6zt\u00fck 6 fenantr\u00e9nvegy\u00fcletet (1-6) \u00e9s 4 kum\u00e1rsav-anal\u00f3got (7-10). A kum\u00e1rsav-anal\u00f3gok els\u0151 \u00edzben t\u00f6rt\u00e9n\u0151 felfedez\u00e9se a Platycodon nemzets\u00e9g n\u00f6v\u00e9nyeiben fontos ir\u00e1nymutat\u00f3 jelent\u0151s\u00e9ggel b\u00edr az Orchidaceae csal\u00e1dba tartoz\u00f3 n\u00f6v\u00e9nyek gazdag k\u00e9miai \u00f6sszet\u00e9tel\u00e9t illet\u0151en.<br \/>\nA vegy\u00fcletek antibakteri\u00e1lis mechanizmus\u00e1nak felt\u00e1r\u00e1sa sor\u00e1n el\u0151sz\u00f6r a kivonatok \u00e9s a monomer vegy\u00fcletek antibakteri\u00e1lis aktivit\u00e1s\u00e1t vizsg\u00e1lt\u00e1k. A vizsg\u00e1lati eredm\u00e9nyek azt mutatt\u00e1k, hogy a vizsg\u00e1lt vegy\u00fcletek k\u00f6z\u00fcl a 6. vegy\u00fclet rendelkezett a legjobb antibakteri\u00e1lis aktivit\u00e1ssal a Staphylococcus aureus ellen (MIC0,01mh\/mL), \u00e9s az antibakteri\u00e1lis hat\u00e1s d\u00f3zisf\u00fcgg\u0151 volt. A SEM eredm\u00e9nyek azt mutatt\u00e1k, hogy a vegy\u00fclet k\u00e1ros\u00edtotta a bakt\u00e9rium sejtfal\u00e1t \u00e9s membr\u00e1nj\u00e1t, intracellul\u00e1ris anyagok sziv\u00e1rg\u00e1s\u00e1t okozva. Ezenk\u00edv\u00fcl az AKP enzimtartalom \u00e9s a PI szonda fluoreszcencia-intenzit\u00e1s\u00e1nak v\u00e1ltoz\u00e1sa tov\u00e1bb bizony\u00edtotta a 6. vegy\u00fclet bakt\u00e9rium membr\u00e1nok k\u00e1rosod\u00e1s\u00e1t. Klinikai alkalmaz\u00e1sban az Atractylodes macrocephala kivonata gyors\u00edthatja a sebgy\u00f3gyul\u00e1st \u00e9s megel\u0151zheti a fert\u0151z\u00e9seket, ami arra utal, hogy az Atractylodes macrocephala antibakteri\u00e1lis tulajdons\u00e1gai a 6. vegy\u00fclettel \u00e9s m\u00e1s fenantr\u00e9nsz\u00e1rmaz\u00e9kokkal hozhat\u00f3k \u00f6sszef\u00fcgg\u00e9sbe.<br \/>\nA fenantr\u00e9nvegy\u00fcletek a szerkezeti t\u00edpusok szempontj\u00e1b\u00f3l a kereskedelmi forgalomban kaphat\u00f3 antibiotikumokt\u00f3l (\u03b2-lakt\u00e1mok, makrolidok, kinolonok) teljesen elt\u00e9r\u0151 szerkezet\u0171 term\u00e9szetes term\u00e9kek. Ebben a tanulm\u00e1nyban a fenantr\u00e9nvegy\u00fcletek j\u00f3 antibakteri\u00e1lis hat\u00e1st mutattak, ami inspir\u00e1ci\u00f3t ny\u00fajt a jelenlegi antibakteri\u00e1lis gy\u00f3gyszerek b\u0151s\u00e9g\u00e9hez. Az \u00faj fenantr\u00e9n antibiotikumok kifejleszt\u00e9se v\u00e1rhat\u00f3an megoldja a gy\u00f3gyszerrezisztens bakt\u00e9riumok probl\u00e9m\u00e1j\u00e1t. Az irodalmi jelent\u00e9sek szerint m\u00e9g az azonos t\u00edpus\u00fa fenantr\u00e9nvegy\u00fcletek is k\u00fcl\u00f6nb\u00f6z\u0151 antibakteri\u00e1lis mechanizmusokat mutathatnak. P\u00e9ld\u00e1ul a blestricin els\u0151sorban a Staphylococcus n\u00f6veked\u00e9s\u00e9t g\u00e1tolja a bakteri\u00e1lis membr\u00e1npotenci\u00e1l \u00e9s integrit\u00e1s megzavar\u00e1s\u00e1val, m\u00edg az aristoloxazin C a Pseudomonas aeruginosa n\u00f6veked\u00e9s\u00e9t a sejtfal lebont\u00e1s\u00e1nak \u00e9s abl\u00e1ci\u00f3j\u00e1nak induk\u00e1l\u00e1s\u00e1val g\u00e1tolja. Szerkezetileg a fenantr\u00e9nvegy\u00fcletek az \u00e9l\u0151 szervezetekben k\u00f6nnyen kinonokk\u00e1 alakulnak \u00e1t, ami f\u00e9lkinon szabadgy\u00f6k\u00f6k termel\u0151d\u00e9s\u00e9hez \u00e9s antibakteri\u00e1lis aktivit\u00e1s kialakul\u00e1s\u00e1hoz vezet. Ez arra utal, hogy tov\u00e1bb kell vizsg\u00e1lni a fenantr\u00e9nvegy\u00fcletek antibakteri\u00e1lis mechanizmus\u00e1t. \u00d6sszefoglalva, kutat\u00e1sunk el\u0151zetesen meger\u0151s\u00edtette a fenantr\u00e9n antibakteri\u00e1lis mechanizmus\u00e1t a bakteri\u00e1lis membr\u00e1nok megbont\u00e1s\u00e1val, k\u00eds\u00e9rleti adatokat szolg\u00e1ltatva a feh\u00e9r \u00e9s antibakteri\u00e1lis szerek farmakol\u00f3giai anyagalapj\u00e1hoz.<\/p>","protected":false},"excerpt":{"rendered":"<p>Identification of Chemical Components in Bai Ji Zhong and Study on the Inhibition Mechanism of Staphylococcus aureus Antibiotics are considered the most &#8220;miracle drugs&#8221; of the 20th century. However, due to the overuse of antibiotics by people, bacterial resistance has emerged. It is expected that by 2050, the global property losses caused by bacterial infections [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Identification of Chemical Components in Bai Ji Zhong and Study on the Inhibition Mechanism of Staphylococcus aureus - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/hu\/bletilla-striata\/\" \/>\n<meta property=\"og:locale\" content=\"hu_HU\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Identification of Chemical Components in Bai Ji Zhong and Study on the Inhibition Mechanism of Staphylococcus aureus - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Identification of Chemical Components in Bai Ji Zhong and Study on the Inhibition Mechanism of Staphylococcus aureus Antibiotics are considered the most &#8220;miracle drugs&#8221; of the 20th century. However, due to the overuse of antibiotics by people, bacterial resistance has emerged. It is expected that by 2050, the global property losses caused by bacterial infections [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/longchangextracts.com\/hu\/bletilla-striata\/\" \/>\n<meta property=\"og:site_name\" content=\"China Chemical Manufacturer\" \/>\n<meta property=\"article:published_time\" content=\"2024-08-04T17:55:12+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-128.png\" \/>\n<meta name=\"author\" content=\"longcha9\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Szerz\u0151:\" \/>\n\t<meta name=\"twitter:data1\" content=\"longcha9\" \/>\n\t<meta name=\"twitter:label2\" content=\"Becs\u00fclt olvas\u00e1si id\u0151\" \/>\n\t<meta name=\"twitter:data2\" content=\"5 perc\" \/>\n<script type=\"application\/ld+json\" class=\"yoast-schema-graph\">{\"@context\":\"https:\/\/schema.org\",\"@graph\":[{\"@type\":\"WebPage\",\"@id\":\"https:\/\/longchangextracts.com\/bletilla-striata\/\",\"url\":\"https:\/\/longchangextracts.com\/bletilla-striata\/\",\"name\":\"Identification of Chemical Components in Bai Ji Zhong and Study on the Inhibition Mechanism of Staphylococcus aureus - China Chemical Manufacturer\",\"isPartOf\":{\"@id\":\"https:\/\/longchangextracts.com\/#website\"},\"primaryImageOfPage\":{\"@id\":\"https:\/\/longchangextracts.com\/bletilla-striata\/#primaryimage\"},\"image\":{\"@id\":\"https:\/\/longchangextracts.com\/bletilla-striata\/#primaryimage\"},\"thumbnailUrl\":\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-128.png\",\"datePublished\":\"2024-08-04T17:55:12+00:00\",\"dateModified\":\"2024-08-04T17:55:12+00:00\",\"author\":{\"@id\":\"https:\/\/longchangextracts.com\/#\/schema\/person\/80933ac6926ad63fea74ec33f8d04869\"},\"breadcrumb\":{\"@id\":\"https:\/\/longchangextracts.com\/bletilla-striata\/#breadcrumb\"},\"inLanguage\":\"hu\",\"potentialAction\":[{\"@type\":\"ReadAction\",\"target\":[\"https:\/\/longchangextracts.com\/bletilla-striata\/\"]}]},{\"@type\":\"ImageObject\",\"inLanguage\":\"hu\",\"@id\":\"https:\/\/longchangextracts.com\/bletilla-striata\/#primaryimage\",\"url\":\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-128.png\",\"contentUrl\":\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-128.png\"},{\"@type\":\"BreadcrumbList\",\"@id\":\"https:\/\/longchangextracts.com\/bletilla-striata\/#breadcrumb\",\"itemListElement\":[{\"@type\":\"ListItem\",\"position\":1,\"name\":\"Home\",\"item\":\"https:\/\/longchangextracts.com\/\"},{\"@type\":\"ListItem\",\"position\":2,\"name\":\"Identification of Chemical Components in Bai Ji Zhong and Study on the Inhibition Mechanism of Staphylococcus aureus\"}]},{\"@type\":\"WebSite\",\"@id\":\"https:\/\/longchangextracts.com\/#website\",\"url\":\"https:\/\/longchangextracts.com\/\",\"name\":\"China Chemical Manufacturer\",\"description\":\"\",\"potentialAction\":[{\"@type\":\"SearchAction\",\"target\":{\"@type\":\"EntryPoint\",\"urlTemplate\":\"https:\/\/longchangextracts.com\/?s={search_term_string}\"},\"query-input\":\"required name=search_term_string\"}],\"inLanguage\":\"hu\"},{\"@type\":\"Person\",\"@id\":\"https:\/\/longchangextracts.com\/#\/schema\/person\/80933ac6926ad63fea74ec33f8d04869\",\"name\":\"longcha9\",\"image\":{\"@type\":\"ImageObject\",\"inLanguage\":\"hu\",\"@id\":\"https:\/\/longchangextracts.com\/#\/schema\/person\/image\/\",\"url\":\"https:\/\/secure.gravatar.com\/avatar\/c1e84ee0759373263198c58e8f338f80?s=96&d=mm&r=g\",\"contentUrl\":\"https:\/\/secure.gravatar.com\/avatar\/c1e84ee0759373263198c58e8f338f80?s=96&d=mm&r=g\",\"caption\":\"longcha9\"}}]}<\/script>\n<!-- \/ Yoast SEO plugin. -->","yoast_head_json":{"title":"Azonos\u00edt\u00e1sa k\u00e9miai \u00f6sszetev\u0151k Bai Ji Zhong \u00e9s tanulm\u00e1nyozza a g\u00e1tl\u00e1si mechanizmusa Staphylococcus aureus - K\u00edna Chemical Manufacturer","robots":{"index":"index","follow":"follow","max-snippet":"max-snippet:-1","max-image-preview":"max-image-preview:large","max-video-preview":"max-video-preview:-1"},"canonical":"https:\/\/longchangextracts.com\/hu\/bletilla-striata\/","og_locale":"hu_HU","og_type":"article","og_title":"Identification of Chemical Components in Bai Ji Zhong and Study on the Inhibition Mechanism of Staphylococcus aureus - China Chemical Manufacturer","og_description":"Identification of Chemical Components in Bai Ji Zhong and Study on the Inhibition Mechanism of Staphylococcus aureus Antibiotics are considered the most &#8220;miracle drugs&#8221; of the 20th century. However, due to the overuse of antibiotics by people, bacterial resistance has emerged. 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