{"id":5071,"date":"2024-08-04T17:11:23","date_gmt":"2024-08-04T17:11:23","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=5071"},"modified":"2024-08-04T17:11:23","modified_gmt":"2024-08-04T17:11:23","slug":"chinese-herbs","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/hu\/chinese-herbs\/","title":{"rendered":"A k\u00ednai gy\u00f3gyn\u00f6v\u00e9nyek \u00e9s hat\u00f3anyagok kutat\u00e1si el\u0151rehalad\u00e1sa a diab\u00e9tesz hat\u00e1s c\u00e9lpontjain\u00e1l"},"content":{"rendered":"<p>A k\u00ednai gy\u00f3gyn\u00f6v\u00e9nyek \u00e9s hat\u00f3anyagok kutat\u00e1si el\u0151rehalad\u00e1sa a diab\u00e9tesz hat\u00e1s c\u00e9lpontjain\u00e1l<br \/>\nA cukorbetegs\u00e9g (DM) az inzulin hi\u00e1nya vagy el\u00e9gtelen szekr\u00e9ci\u00f3ja \u00e1ltal okozott anyagcserezavar, amelyet hiperglik\u00e9mia jellemez, \u00e9s amelynek 90%~95% r\u00e9sze a 2-es t\u00edpus\u00fa cukorbetegs\u00e9g. A Nemzetk\u00f6zi Diab\u00e9tesz Sz\u00f6vets\u00e9g (IDF) legfrissebb adatai szerint 2021-ben a DM sz\u00e1ma a vil\u00e1gon el\u00e9ri az 537 milli\u00f3t, ami 2045-ben v\u00e1rhat\u00f3an meghaladja a 783 milli\u00f3t (12,2%), K\u00edn\u00e1ban pedig v\u00e1rhat\u00f3an meghaladja a 175 milli\u00f3t 2045-ben. A DM a tumorok \u00e9s a sz\u00edv- \u00e9s \u00e9rrendszeri betegs\u00e9gek ut\u00e1n a harmadik legs\u00falyosabb, az emberi eg\u00e9szs\u00e9get vesz\u00e9lyeztet\u0151 kr\u00f3nikus betegs\u00e9gg\u00e9 v\u00e1lt a vil\u00e1gon. A magas v\u00e9rcukorszint okozta k\u00fcl\u00f6nb\u00f6z\u0151 akut \u00e9s kr\u00f3nikus sz\u00f6v\u0151dm\u00e9nyek k\u00e1ros\u00edthatj\u00e1k az emberi sz\u00f6veteket, szerveket stb. Ez\u00e9rt s\u00fcrg\u0151sen akt\u00edv int\u00e9zked\u00e9seket kell tenni a megel\u0151z\u00e9s \u00e9s a korai kezel\u00e9s \u00e9rdek\u00e9ben.<br \/>\nJelenleg nincs olyan gy\u00f3gyszerr\u0151l sz\u00f3l\u00f3 jelent\u00e9s, amely a klinikai gyakorlatban teljesen meggy\u00f3gy\u00edtan\u00e1 a DM-et. A v\u00e9rcukorszint szab\u00e1lyoz\u00e1s\u00e1ra sokf\u00e9le nyugati gy\u00f3gyszert haszn\u00e1lnak, bele\u00e9rtve az inzulint \u00e9s anal\u00f3gjait, szulfonilure\u00e1kat, biguanidokat, gliptideket, tiazolidindionokat, alfa-gl\u00fckozid\u00e1z-g\u00e1tl\u00f3kat, dipeptidil-peptid\u00e1z-g\u00e1tl\u00f3kat, n\u00e1trium-gl\u00fck\u00f3z-kotranszporter 2 g\u00e1tl\u00f3kat, gl\u00fckagonszer\u0171 peptid-1 receptor agonist\u00e1kat stb. B\u00e1r gyorsan \u00e9s hat\u00e9konyan szab\u00e1lyozhatj\u00e1k a cukrot, hossz\u00fa t\u00e1v\u00fa alkalmaz\u00e1suk k\u00f6nnyen egy sor probl\u00e9m\u00e1t okozhat, p\u00e9ld\u00e1ul hipoglik\u00e9mi\u00e1t, gyomor-b\u00e9lrendszeri reakci\u00f3kat \u00e9s sz\u00edv- \u00e9s \u00e9rrendszeri betegs\u00e9geket. A hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szat \u00e9s hat\u00f3anyagainak sz\u0171r\u00e9s\u00e9vel, valamint a farmakol\u00f3giai hat\u00e1sok tanulm\u00e1nyoz\u00e1s\u00e1val folyamatosan felt\u00e1rt\u00e1k a hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szat t\u00f6bbkomponens\u0171 \u00e9s t\u00f6bb c\u00e9lpontra gyakorolt hat\u00e1s\u00e1nak jellemz\u0151it, ami az enyhe hat\u00e9konys\u00e1g, a minim\u00e1lis toxikus mell\u00e9khat\u00e1sok \u00e9s az \u00e1ltal\u00e1nos szab\u00e1lyoz\u00e1s el\u0151nyeit mutatja a DM kezel\u00e9s\u00e9ben. Ugyanakkor a DM k\u00fcl\u00f6nb\u00f6z\u0151 sz\u00f6v\u0151dm\u00e9nyeinek megel\u0151z\u00e9s\u00e9re \u00e9s kezel\u00e9s\u00e9re is alkalmas. Az elm\u00falt \u00e9vekben a DM kezel\u00e9s\u00e9re szolg\u00e1l\u00f3 \u00faj gy\u00f3gyszerek kifejleszt\u00e9se els\u0151sorban az effektor c\u00e9lpontokon alapult, bele\u00e9rtve az alfa-gl\u00fckozid\u00e1zt, az alfa-amil\u00e1zt, a dipeptidil-peptid\u00e1z-4-et (DPP-4), a gl\u00fckokin\u00e1zt (GK), n\u00e1trium-gl\u00fck\u00f3z-kotranszporter 2 (SGLT2), m\u00e1trix-metalloprotein\u00e1zok (MMP), feh\u00e9rje-tirozin-foszfat\u00e1z 1B (PTP1B), ald\u00f3z-redukt\u00e1z (AR), peroxisz\u00f3ma-prolifer\u00e1tor aktiv\u00e1lt receptor (peroxisz\u00f3ma-prolifer\u00e1tor aktiv\u00e1lt receptor). \u00e9letet aktiv\u00e1l\u00f3 receptorok (PPAR), adenozin-monofoszf\u00e1t aktiv\u00e1lt feh\u00e9rje-kin\u00e1z (AMPK) \u00fatvonal, ATP-\u00e9rz\u00e9keny k\u00e1liumcsatorna, A hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szat \u00e9s hat\u00f3anyagainak sz\u0171r\u00e9se a DM kezel\u00e9s\u00e9re a specifikus c\u00e9lpontok \u00e9s \u00fatvonalak, p\u00e9ld\u00e1ul a KATP c\u00e9lba v\u00e9tel\u00e9vel jav\u00edthatja a gy\u00f3gyszerhat\u00e1s szelektivit\u00e1s\u00e1t \u00e9s cs\u00f6kkentheti vagy minimaliz\u00e1lhatja a toxikus mell\u00e9khat\u00e1sokat; Ugyanakkor a hat\u00f3anyagok hat\u00e1smechanizmus\u00e1t is megvil\u00e1g\u00edthatja, \u00e9s referencia-m\u00f3dszereket \u00e9s \u00f6tleteket biztos\u00edthat a hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szat tov\u00e1bbi fejleszt\u00e9s\u00e9hez \u00e9s felhaszn\u00e1l\u00e1s\u00e1hoz. Ez\u00e9rt ez a cikk rendszerezi \u00e9s \u00f6sszefoglalja a hagyom\u00e1nyos k\u00ednai orvosl\u00e1s \u00e9s a hat\u00f3anyagok DM c\u00e9lpontokra \u00e9s \u00fatvonalakra gyakorolt hat\u00e1saival kapcsolatos relev\u00e1ns irodalmat itthon \u00e9s k\u00fclf\u00f6ld\u00f6n, annak \u00e9rdek\u00e9ben, hogy referenci\u00e1t ny\u00fajtson a hagyom\u00e1nyos k\u00ednai orvosl\u00e1s tanulm\u00e1nyoz\u00e1s\u00e1hoz a DM \u00e9s sz\u00f6v\u0151dm\u00e9nyeinek kezel\u00e9s\u00e9ben.<\/p>\n<p>&nbsp;<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5072\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-116.png\" alt=\"\" width=\"773\" height=\"256\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-116.png 773w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-116-768x254.png 768w\" sizes=\"(max-width: 773px) 100vw, 773px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5073\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-102.png\" alt=\"\" width=\"773\" height=\"231\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-102.png 773w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-102-768x230.png 768w\" sizes=\"(max-width: 773px) 100vw, 773px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5074\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-96.png\" alt=\"\" width=\"782\" height=\"462\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-96.png 782w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-96-768x454.png 768w\" sizes=\"(max-width: 782px) 100vw, 782px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5075\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-85.png\" alt=\"\" width=\"782\" height=\"342\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-85.png 782w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-85-768x336.png 768w\" sizes=\"(max-width: 782px) 100vw, 782px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5076\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-78.png\" alt=\"\" width=\"784\" height=\"236\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-78.png 784w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-78-768x231.png 768w\" sizes=\"(max-width: 784px) 100vw, 784px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-5077\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-70.png\" alt=\"\" width=\"780\" height=\"362\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-70.png 780w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-70-768x356.png 768w\" sizes=\"(max-width: 780px) 100vw, 780px\" \/><\/p>\n<p>Ez a cikk \u00f6sszefoglalja a hagyom\u00e1nyos k\u00ednai orvosl\u00e1st \u00e9s a DM kezel\u00e9s\u00e9re szolg\u00e1l\u00f3 hat\u00f3anyagokat olyan effektor c\u00e9lpontokkal, mint az \u03b1 - gl\u00fckozid\u00e1z, \u03b1 - amil\u00e1z, DPP-4, GK, PTP1B, SGLT2, PPAR, stb. Meg\u00e1llap\u00edtott\u00e1k, hogy a k\u00fcl\u00f6nb\u00f6z\u0151 term\u00e9szetes term\u00e9kek k\u00fcl\u00f6nb\u00f6z\u0151 k\u00e9miai szerkezet\u0171ek, \u00e9s kompetit\u00edv, nem kompetit\u00edv \u00e9s vegyes m\u00f3dszerekkel k\u00e9pesek g\u00e1tolni vagy aktiv\u00e1lni az effektor c\u00e9lpontokat. Farmakol\u00f3giai aktivit\u00e1suk is elt\u00e9r\u0151.<\/p>\n<p>A vonatkoz\u00f3 hazai \u00e9s k\u00fclf\u00f6ldi kutat\u00e1si eredm\u00e9nyek \u00e1ttekint\u00e9se sor\u00e1n meg\u00e1llap\u00edtott\u00e1k, hogy a hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szat k\u00fcl\u00f6nb\u00f6z\u0151 hipoglik\u00e9mi\u00e1s hat\u00f3anyagokat, p\u00e9ld\u00e1ul alkaloidokat, flavonoidokat, terp\u00e9neket \u00e9s poliszacharidokat tartalmaz. Az enzimekre, receptorokra, ioncsatorn\u00e1kra stb. hatva szab\u00e1lyozza az inzulinszekr\u00e9ci\u00f3t, fokozza az inzulin\u00e9rz\u00e9kenys\u00e9get \u00e9s kezeli a DM-et. Szinergikus \u00e9s kieg\u00e9sz\u00edt\u0151 hipoglik\u00e9mi\u00e1s mechanizmusainak k\u00f6sz\u00f6nhet\u0151en cs\u00f6kkenti a toxicit\u00e1st \u00e9s n\u00f6veli a hat\u00e9konys\u00e1got. A klinikai gyakorlatban jelenleg haszn\u00e1lt k\u00e9miai gy\u00f3gyszerekkel \u00f6sszehasonl\u00edtva hat\u00e1sai enyh\u00e9bbek \u00e9s biztons\u00e1gosabbak. Ez\u00e9rt a c\u00e9lhat\u00e1sokra hat\u00f3 term\u00e9szetes term\u00e9kekb\u0151l sz\u00e1rmaz\u00f3 hat\u00f3anyagok kinyer\u00e9se a DM innovat\u00edv gy\u00f3gyszerfejleszt\u00e9s\u00e9nek egyik f\u0151 f\u00f3kuszpontj\u00e1v\u00e1 v\u00e1lt K\u00edn\u00e1ban.<\/p>\n<p>Jelenleg a DM hagyom\u00e1nyos k\u00ednai orvosl\u00e1ssal t\u00f6rt\u00e9n\u0151 kezel\u00e9s\u00e9nek kutat\u00e1sa bizonyos el\u0151rehalad\u00e1st \u00e9rt el, de m\u00e9g mindig a felt\u00e1r\u00f3 szakaszban van. A j\u00f6v\u0151ben m\u00e9lyrehat\u00f3an vizsg\u00e1lhatjuk ezeket a k\u00e9rd\u00e9seket: sok, a DM kezel\u00e9s\u00e9re haszn\u00e1lt gy\u00f3gyn\u00f6v\u00e9ny \u00e9s hat\u00f3anyag csak egyetlen c\u00e9lpontra hat, \u00e9s a t\u00f6bb c\u00e9lpontot \u00e9s t\u00f6bb \u00fatvonalat \u00e9rint\u0151 hagyom\u00e1nyos k\u00ednai orvosl\u00e1ssal t\u00f6rt\u00e9n\u0151 kezel\u00e9s el\u0151nyei m\u00e9g nem teljesen tiszt\u00e1zottak, \u00e9s a specifikus hat\u00e1smechanizmus m\u00e9g jav\u00edt\u00e1sra szorul. A kutat\u00e1sok meg\u00e1llap\u00edtott\u00e1k, hogy a gyullad\u00e1s okozta immunv\u00e1lasz inzulinrezisztenci\u00e1t v\u00e1lthat ki, ami a DM kialakul\u00e1s\u00e1hoz vezet. A gyullad\u00e1s \u00e9s az inzulinrezisztencia mechanizmus\u00e1nak tov\u00e1bbi tiszt\u00e1z\u00e1sa hat\u00e9kony eszk\u00f6z\u00f6ket biztos\u00edthat a DM kezel\u00e9s\u00e9hez. A hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szati formul\u00e1k \u00f6sszetetts\u00e9ge, t\u00f6bbf\u00e9le hat\u00e1sc\u00e9lja \u00e9s a hat\u00e1smechanizmus felt\u00e1r\u00e1s\u00e1nak neh\u00e9zs\u00e9gei megnehez\u00edtik a kutat\u00e1sukat. A DM kezel\u00e9s\u00e9vel kapcsolatos kutat\u00e1sok t\u00f6bbnyire az egyes k\u00ednai gy\u00f3gyszerkivonatokkal \u00e9s hat\u00f3anyagaikkal v\u00e9gzett in vitro alapk\u00eds\u00e9rleteken alapulnak. Ez\u00e9rt a j\u00f6v\u0151beni munk\u00e1ban a DM kezel\u00e9s\u00e9re szolg\u00e1l\u00f3 hagyom\u00e1nyos k\u00ednai gy\u00f3gyszerk\u00e9sz\u00edtm\u00e9nyek \u00e9s \u00f6sszetev\u0151ik kutat\u00e1sa lehet a f\u0151 feladat. Ezen t\u00falmen\u0151en a hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szat \u00e9s hat\u00f3anyagai a DM kezel\u00e9se \u00e9rdek\u00e9ben a kapcsol\u00f3d\u00f3 jel\u00e1tviteli \u00fatvonalakat is szab\u00e1lyozhatj\u00e1k effektor c\u00e9lpontokon kereszt\u00fcl. Az\u00e1ltal, hogy \u00e1tfog\u00f3an felt\u00e1rja az \"\u00f6sszetev\u0151k betegs\u00e9g c\u00e9lpontok \u00fatvonalai\" k\u00f6z\u00f6tti kapcsolatot k\u00fcl\u00f6nb\u00f6z\u0151 modern tudom\u00e1nyos technol\u00f3gi\u00e1kon kereszt\u00fcl, ez alapot ny\u00fajt a DM kezel\u00e9s\u00e9re szolg\u00e1l\u00f3 jobb hagyom\u00e1nyos k\u00ednai gy\u00f3gy\u00e1szat tov\u00e1bbi kutat\u00e1s\u00e1hoz \u00e9s fejleszt\u00e9s\u00e9hez.<\/p>\n<p>\u00dagy v\u00e9lem, hogy a technol\u00f3gia fejl\u0151d\u00e9s\u00e9vel \u00e9s a kutat\u00e1s elm\u00e9ly\u00edt\u00e9s\u00e9vel a hagyom\u00e1nyos k\u00ednai orvosl\u00e1s hat\u00e1smechanizmusa a DM kezel\u00e9s\u00e9ben vil\u00e1gosabb\u00e1 v\u00e1lik, \u00e9s t\u00f6bb biztons\u00e1gos \u00e9s hat\u00e9kony term\u00e9szetes gy\u00f3gyszert \u00e9s hat\u00f3anyagot fedeznek fel a DM kezel\u00e9s\u00e9re.<\/p>","protected":false},"excerpt":{"rendered":"<p>Research progress of Chinese herbs and active ingredients acting on diabetes effect targets Diabetes (DM) is a metabolic disorder caused by insulin deficiency or insufficient secretion, and is characterized by hyperglycemia, of which type 2 diabetes accounts for 90%~95%. According to the latest data of International diabetes Federation (IDF) in 2021, the number of DM [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Research progress of Chinese herbs and active ingredients acting on diabetes effect targets - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/hu\/chinese-herbs\/\" \/>\n<meta property=\"og:locale\" content=\"hu_HU\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Research progress of Chinese herbs and active ingredients acting on diabetes effect targets - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Research progress of Chinese herbs and active ingredients acting on diabetes effect targets Diabetes (DM) is a metabolic disorder caused by insulin deficiency or insufficient secretion, and is characterized by hyperglycemia, of which type 2 diabetes accounts for 90%~95%. 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