{"id":4566,"date":"2024-08-04T14:53:22","date_gmt":"2024-08-04T14:53:22","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=4566"},"modified":"2024-08-04T14:53:22","modified_gmt":"2024-08-04T14:53:22","slug":"callicarpa-nudiflora","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/fr\/callicarpa-nudiflora\/","title":{"rendered":"Exploration des composants actifs anti-H1N1 et des m\u00e9canismes des billes violettes nues sur la base de l'UPLC-Q-Exactive-Orbitrap-MS, de la pharmacologie de r\u00e9seau et de la validation exp\u00e9rimentale"},"content":{"rendered":"<p>Exploration des composants actifs anti-H1N1 et des m\u00e9canismes des billes violettes nues sur la base de l'UPLC-Q-Exactive-Orbitrap-MS, de la pharmacologie de r\u00e9seau et de la validation exp\u00e9rimentale<br \/>\nCallicarpa nudiflora Hook.&amp;Arn. est une feuille s\u00e9ch\u00e9e de la plante Callicarpa nudiflora Hook.&amp;Arn. de la famille des Verbenaceae. Les perles violettes nues sont principalement distribu\u00e9es \u00e0 Hainan, Guangxi, Guangdong et dans d'autres r\u00e9gions, la zone de production authentique \u00e9tant le district de Wuzhishan dans la province de Hainan. La fleur nue perle violette est le seul m\u00e9dicament traditionnel chinois nouvellement ajout\u00e9 dans l'\u00e9dition 2020 de la pharmacop\u00e9e de la R\u00e9publique populaire de Chine. Ses pr\u00e9parations unilat\u00e9rales, Naked Flower Purple Pearl Tablets et Naked Flower Purple Pearl Capsules, sont largement utilis\u00e9es pour traiter les h\u00e9morragies respiratoires et digestives et les inflammations infectieuses bact\u00e9riennes caus\u00e9es par une chaleur et une toxicit\u00e9 sanguines excessives. Les phytochimistes ont identifi\u00e9 plus de 300 compos\u00e9s dans les perles violettes nues, dont des ph\u00e9nylpropano\u00efdes, des flavono\u00efdes, des triterp\u00e9no\u00efdes, des diterp\u00e8nes, des irido\u00efdes, des huiles volatiles, etc. La recherche pharmacologique moderne a confirm\u00e9 que la fleur nue de perle violette a des activit\u00e9s anti-inflammatoires, antithrombotiques, antitumorales, antibact\u00e9riennes et h\u00e9patoprotectrices. Au cours du processus de s\u00e9lection des m\u00e9dicaments traditionnels chinois ayant une activit\u00e9 antivirale, il a \u00e9t\u00e9 constat\u00e9 que l'extrait de fleur nue de perle violette avait une bonne activit\u00e9 antivirale (comme le virus de la grippe H1N1, l'ent\u00e9rovirus 71, etc.) L'infection par le virus de la grippe A est une cause fr\u00e9quente de d\u00e9c\u00e8s li\u00e9s \u00e0 la pneumonie. Une infection s\u00e9v\u00e8re par le virus de la grippe A peut provoquer une infiltration pulmonaire bilat\u00e9rale et une hypox\u00e9mie, connues sous le nom de syndrome de d\u00e9tresse respiratoire aigu\u00eb, qui est l'une des principales causes de d\u00e9c\u00e8s provoqu\u00e9s par le virus de la grippe A. Cette exp\u00e9rience porte sur l'activit\u00e9 anti-H1N1 de la perle violette \u00e0 fleur nue. La composition chimique des parties efficaces de la fleur nue pourpre a \u00e9t\u00e9 identifi\u00e9e \u00e0 l'aide de la chromatographie liquide \u00e0 ultra-haute performance, de la spectrom\u00e9trie de masse \u00e0 champ \u00e9lectrostatique quadripolaire et le m\u00e9canisme anti-H1N1 de la fleur nue pourpre a \u00e9t\u00e9 pr\u00e9dit et v\u00e9rifi\u00e9 exp\u00e9rimentalement \u00e0 l'aide de la pharmacologie de r\u00e9seau. Le m\u00e9canisme d'action de la perle violette de fleur nue contre le H1N1 a fait l'objet d'une \u00e9tude pr\u00e9liminaire.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4570\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-73.png\" alt=\"\" width=\"340\" height=\"709\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4571\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-63.png\" alt=\"\" width=\"340\" height=\"234\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4572\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-60.png\" alt=\"\" width=\"600\" height=\"621\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4573\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-50.png\" alt=\"\" width=\"600\" height=\"660\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4574\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-2.jpg\" alt=\"\" width=\"539\" height=\"748\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-2.jpg 539w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-2-519x720.jpg 519w\" sizes=\"(max-width: 539px) 100vw, 539px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4575\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-44.png\" alt=\"\" width=\"539\" height=\"272\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4576\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-42.png\" alt=\"\" width=\"600\" height=\"784\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-42.png 600w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-42-551x720.png 551w\" sizes=\"(max-width: 600px) 100vw, 600px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4577\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-36.png\" alt=\"\" width=\"600\" height=\"539\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4578\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-31.png\" alt=\"\" width=\"600\" height=\"304\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4579\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-27.png\" alt=\"\" width=\"600\" height=\"244\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4580\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-25.png\" alt=\"\" width=\"340\" height=\"219\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4581\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-21.png\" alt=\"\" width=\"340\" height=\"546\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4582\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-18.png\" alt=\"\" width=\"600\" height=\"271\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4583\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/14-15.png\" alt=\"\" width=\"600\" height=\"327\" \/>callicarpa nudiflora<br \/>\nLe virus de la grippe A a d\u00e9velopp\u00e9 divers degr\u00e9s de r\u00e9sistance aux inhibiteurs du canal M2 et aux inhibiteurs de la NA couramment utilis\u00e9s. Par cons\u00e9quent, la recherche de nouveaux m\u00e9dicaments ou de nouvelles m\u00e9thodes de traitement contre la grippe A est devenue un probl\u00e8me urgent \u00e0 r\u00e9soudre. La m\u00e9decine traditionnelle chinoise a jou\u00e9 un r\u00f4le important dans le traitement clinique du virus de la grippe A. Le concept holistique de la th\u00e9orie de la m\u00e9decine traditionnelle chinoise r\u00e9gule syst\u00e9matiquement les patients comme un ensemble organique, tandis que la pharmacologie de r\u00e9seau explore l'interaction entre les fonctions biologiques de chaque n\u0153ud du r\u00e9seau et les maladies en construisant un r\u00e9seau de voies cibles des composants des m\u00e9dicaments, ce qui est coh\u00e9rent avec le concept holistique de la m\u00e9decine traditionnelle chinoise. Cette exp\u00e9rience a d'abord examin\u00e9 les principaux sites actifs anti-H1N1 du m\u00e9dicament traditionnel chinois Naked Flower Purple Pearl et a analys\u00e9 les sites pour identifier 34 composants chimiques. En combinant la litt\u00e9rature et les bases de donn\u00e9es, 67 cibles de m\u00e9dicaments et de maladies se chevauchant ont \u00e9t\u00e9 identifi\u00e9es. Gr\u00e2ce \u00e0 l'analyse d'enrichissement des cibles crois\u00e9es, nous supposons que le processus biologique important de l'EACN contre le H1N1 pourrait \u00eatre la r\u00e9gulation positive de la phosphorylation des prot\u00e9ines et la r\u00e9ponse au stress oxydatif. Les r\u00e9sultats de l'analyse d'enrichissement KEGG ont montr\u00e9 que 19 compos\u00e9s d'EACN agissent sur la voie du virus de la grippe A par l'interm\u00e9diaire de 11 cibles. Le m\u00e9dicament affecte le canal M2 du virus H1N1 en agissant sur PLG et PRSS1, et peut \u00e9galement affecter le processus de lib\u00e9ration du virus en agissant sur la voie de la neuraminidase (NA) par l'interm\u00e9diaire de PLG. PLG et PRSS1 peuvent \u00eatre des cibles cl\u00e9s pour l'action directe de l'EACN sur le virus H1N1. L'EACN peut inhiber la prolif\u00e9ration du H1N1 en affectant ses processus d'excr\u00e9tion et de lib\u00e9ration. Dans le r\u00e9seau de maladies de la voie des ingr\u00e9dients m\u00e9dicamenteux, RELA et NF - \u03ba B1 sont les deux cibles ayant les valeurs de degr\u00e9 les plus \u00e9lev\u00e9es. La voie de signalisation NF - \u03ba B dans laquelle elles se trouvent peut promouvoir l'expression de facteurs tels que IL1 \u03b2, TNF - \u03b1, IL-6, et favoriser la r\u00e9ponse inflammatoire, ce qui sugg\u00e8re que l'EACN peut agir sur des cibles cl\u00e9s telles que RELA et NF - \u03ba B1 pour r\u00e9guler la voie de signalisation NF - \u03ba B et r\u00e9duire les dommages caus\u00e9s par l'inflammation \u00e0 l'organisme. Selon les r\u00e9sultats pr\u00e9dits par la pharmacologie des r\u00e9seaux, l'EACN peut r\u00e9guler les voies de signalisation des cellules T, affecter la diff\u00e9renciation Th1 et Th2 et exercer des effets r\u00e9gulateurs sur le syst\u00e8me immunitaire. Par cons\u00e9quent, cette \u00e9tude a men\u00e9 des exp\u00e9riences sur des animaux pour v\u00e9rifier l'effet inhibiteur, l'effet anti-inflammatoire et l'effet r\u00e9gulateur immunitaire de l'EACN sur la prolif\u00e9ration du virus H1N1. Les r\u00e9sultats exp\u00e9rimentaux ont montr\u00e9 que l'EACN peut am\u00e9liorer la perte de poids et l'augmentation de l'indice pulmonaire caus\u00e9es par l'infection H1N1, r\u00e9duire la charge virale dans le tissu pulmonaire de la souris, att\u00e9nuer les dommages pathologiques dans le tissu pulmonaire de la souris, r\u00e9duire les niveaux de TNF - \u03b1, IFN - \u03b3, IL-1 \u03b2 dans le s\u00e9rum du sang p\u00e9riph\u00e9rique et augmenter le niveau d'anticorps IgG dans le s\u00e9rum. Cette \u00e9tude a d'abord utilis\u00e9 des exp\u00e9riences in vitro pour cribler les sites d'extraction actifs de Naked Purple Pearl contre le H1N1, et a pr\u00e9dit les ingr\u00e9dients actifs d'EACN contre le H1N1 en utilisant l'UPLC-Q-Hexactive-Orbitrap-MS et la pharmacologie de r\u00e9seau. Les r\u00e9sultats pr\u00e9dits ont \u00e9t\u00e9 v\u00e9rifi\u00e9s par des exp\u00e9riences sur les animaux, et les ingr\u00e9dients actifs potentiels de l'EACN contre le H1N1 ont \u00e9t\u00e9 s\u00e9lectionn\u00e9s, y compris la querc\u00e9tine, la myric\u00e9tine, la lut\u00e9oline, le kaempf\u00e9rol, la querc\u00e9tine, l'apig\u00e9nine et l'ac\u00e9tine. Il a \u00e9t\u00e9 d\u00e9montr\u00e9 de mani\u00e8re pr\u00e9liminaire que le Naked Purple Pearl peut exercer des effets anti-H1N1 par de multiples voies telles que l'inhibition directe du virus, les effets anti-inflammatoires et la r\u00e9gulation immunitaire. Dans des exp\u00e9riences ult\u00e9rieures, il est n\u00e9cessaire de mener des exp\u00e9riences in vitro et in vivo pour valider les compos\u00e9s monom\u00e8res s\u00e9lectionn\u00e9s et \u00e9tudier plus en d\u00e9tail le m\u00e9canisme de l'effet anti H1N1 de l'EACN au niveau de l'ARNm et de la prot\u00e9ine.<\/p>","protected":false},"excerpt":{"rendered":"<p>Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation The traditional Chinese medicine, Callicarpa nudiflora Hook.&amp;Arn., is a dried leaf of the plant Callicarpa nudiflora Hook.&amp;Arn. in the family Verbenaceae. Naked Purple Beads are mainly distributed in Hainan, Guangxi, Guangdong and other regions, with [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/fr\/callicarpa-nudiflora\/\" \/>\n<meta property=\"og:locale\" content=\"fr_FR\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation The traditional Chinese medicine, Callicarpa nudiflora Hook.&amp;Arn., is a dried leaf of the plant Callicarpa nudiflora Hook.&amp;Arn. in the family Verbenaceae. 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