{"id":4588,"date":"2024-08-04T14:55:47","date_gmt":"2024-08-04T14:55:47","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=4588"},"modified":"2024-08-04T14:55:47","modified_gmt":"2024-08-04T14:55:47","slug":"bairui-granules","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/es\/bairui-granulos\/","title":{"rendered":"Estudio de los componentes sangu\u00edneos de los gr\u00e1nulos de Bai Rui basado en la tecnolog\u00eda UHPLC-Q-TOF-MS\/MS"},"content":{"rendered":"<p>Estudio de los componentes sangu\u00edneos de los gr\u00e1nulos de Bai Rui basado en la tecnolog\u00eda UHPLC-Q-TOF-MS\/MS<\/p>\n<p>Estudio de los componentes sangu\u00edneos de los gr\u00e1nulos de Bai Rui basado en la tecnolog\u00eda UHPLC-Q-TOF-MS\/MS<br \/>\nLos gr\u00e1nulos de Bairui son un preparado granulado compuesto de hierba \u00fanica Bairui, que tiene efectos antibacterianos y antiinflamatorios, despeja el calor y desintoxica, y alivia la tos. Se utilizan habitualmente en la pr\u00e1ctica cl\u00ednica moderna para tratar la amigdalitis pedi\u00e1trica, la bronquitis y diversas infecciones respiratorias. Para ejercer sus efectos, los principios activos de la medicina tradicional china se transportan principalmente a la diana a trav\u00e9s de la sangre como medio (excluyendo la acci\u00f3n directa en el intestino y la medicaci\u00f3n externa). Por lo tanto, el an\u00e1lisis de los ingredientes activos en el cuerpo despu\u00e9s de la administraci\u00f3n oral de la medicina tradicional china es muy importante para el estudio de la base material de la eficacia de la medicina tradicional china. Nuestro grupo de investigaci\u00f3n ha utilizado anteriormente la tecnolog\u00eda de cromatograf\u00eda l\u00edquida-espectrometr\u00eda de masas para analizar sistem\u00e1ticamente la composici\u00f3n qu\u00edmica del extracto alcoh\u00f3lico de Atractylodes macrocephala, y ha descubierto que hay muchos ingredientes eficaces en Atractylodes macrocephala, como flavonoides, alcaloides y otros compuestos. Los estudios bibliogr\u00e1ficos anteriores se han centrado sobre todo en la composici\u00f3n qu\u00edmica y el control de calidad de hierbas individuales, y carecen de investigaciones sobre los componentes sangu\u00edneos y los procesos metab\u00f3licos de los gr\u00e1nulos de Atractylodes macrocephala in vivo, y la base farmacol\u00f3gica de la sustancia a\u00fan no est\u00e1 clara.<\/p>\n<p>La tecnolog\u00eda de espectrometr\u00eda de masas de tiempo de vuelo cuadrupolar, debido a su alta sensibilidad y resoluci\u00f3n, puede analizar de forma r\u00e1pida y eficiente los componentes qu\u00edmicos de la medicina tradicional china, y se ha utilizado ampliamente en la investigaci\u00f3n de la base de sustancias de la eficacia de la medicina tradicional china. Por lo tanto, sobre la base de investigaciones anteriores, nuestro grupo de investigaci\u00f3n sigue utilizando la tecnolog\u00eda de espectrometr\u00eda de masas de tiempo de vuelo cuadrupolar de cromatograf\u00eda l\u00edquida de ultra alto rendimiento (UHPLC-Q-TOF-MS\/MS) para analizar los componentes que entran en la sangre y el proceso metab\u00f3lico del gr\u00e1nulo Baisui, que proporciona una base de referencia para la investigaci\u00f3n b\u00e1sica de sustancias eficaces, y es de gran importancia para el control de calidad y el desarrollo y la utilizaci\u00f3n de medicinas tradicionales chinas patentadas y preparaciones simples.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4589\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-74.png\" alt=\"\" width=\"604\" height=\"791\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-74.png 604w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-74-550x720.png 550w\" sizes=\"(max-width: 604px) 100vw, 604px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4590\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-64.png\" alt=\"\" width=\"601\" height=\"515\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4591\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-2.jpg\" alt=\"\" width=\"601\" height=\"286\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4592\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-6.jpg\" alt=\"\" width=\"601\" height=\"281\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4593\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-49.png\" alt=\"\" width=\"601\" height=\"462\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4594\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-45.png\" alt=\"\" width=\"601\" height=\"661\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4595\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-2.jpg\" alt=\"\" width=\"600\" height=\"651\" \/><br \/>\nEn este estudio se utiliz\u00f3 la tecnolog\u00eda UHPLC-Q-TOF-MS\/MS para analizar los componentes sangu\u00edneos absorbidos de los gr\u00e1nulos de Bairui. Se detectaron un total de 20 componentes prototipo y 10 metabolitos del suero de rata. Los principales componentes analizados en el organismo son alcaloides como la quercetina y la sofocarpina, as\u00ed como flavonoides como el kaempferol y el resveratrol I; Los principales productos metab\u00f3licos en el organismo son la oxidaci\u00f3n y glucuronidaci\u00f3n del kaempferol y la oxidaci\u00f3n e hidr\u00f3lisis de la sofocarpina, lo que indica que los alcaloides y flavonoides son los principales componentes que entran en el organismo y tambi\u00e9n pueden ser potenciales principios activos para la eficacia del f\u00e1rmaco.<\/p>\n<p>La investigaci\u00f3n farmacol\u00f3gica moderna ha demostrado que los flavonoides y alcaloides tienen funciones farmacol\u00f3gicas como antiinflamatorias, antibacterianas, antivirales y antioxidantes. Estudios anteriores han informado de que el efecto antiinflamatorio de los derivados del resveratrol en Bai Rui Cao est\u00e1 relacionado con su eficaz inhibici\u00f3n de la producci\u00f3n intracelular de especies reactivas del ox\u00edgeno y la activaci\u00f3n de p38 MAPK y la prote\u00edna activadora 1. Como flavonol natural, el resveratrol tiene un fuerte efecto en la inhibici\u00f3n de la funci\u00f3n de las c\u00e9lulas inflamatorias y la supresi\u00f3n de la expresi\u00f3n de citoquinas proinflamatorias y quimioquinas. Bairuicao I puede inhibir la expresi\u00f3n de citoquinas inflamatorias TNF - \u03b1, IL-6, IL-1 \u03b2, etc, actuando sobre el NF - \u03ba B y v\u00edas MAPK, mejorando as\u00ed el edema pulmonar en ratones infectados con neumon\u00eda. Los alcaloides pueden inhibir significativamente el crecimiento de microorganismos como Escherichia coli y Staphylococcus aureus. La sofocarpina tiene fuertes efectos antiinflamatorios y analg\u00e9sicos y puede reducir la inflamaci\u00f3n inhibiendo la v\u00eda de se\u00f1alizaci\u00f3n NF - \u03ba B. La oximatrina puede ejercer efectos antiinflamatorios inhibiendo la v\u00eda de se\u00f1alizaci\u00f3n NF - \u03ba B y reduciendo la expresi\u00f3n de los factores inflamatorios IL-6 e IL-8.<\/p>\n<p>En resumen, este estudio dilucid\u00f3 los componentes sangu\u00edneos y los metabolitos de los gr\u00e1nulos de Bairui mediante la tecnolog\u00eda UHPLC-Q-TOFMS\/MS. Estos compuestos pueden estar estrechamente relacionados con los efectos antiinflamatorios y antibacterianos de los gr\u00e1nulos de Bairui, lo que es de gran importancia para aclarar la base material de la eficacia de la medicina tradicional china y mejorar los est\u00e1ndares de calidad de la medicina tradicional china. Proporciona una base de referencia para comprender mejor su mecanismo de acci\u00f3n y su aplicaci\u00f3n cl\u00ednica.<\/p>","protected":false},"excerpt":{"rendered":"<p>Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology Bairui granules are a granular preparation composed of single herb Bairui grass, which has the effects of antibacterial and anti-inflammatory, clearing heat and detoxifying, and relieving cough. They are [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/es\/bairui-granulos\/\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology Bairui granules are a granular preparation composed of single herb Bairui grass, which has the effects of antibacterial and anti-inflammatory, clearing heat and detoxifying, and relieving cough. 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