{"id":7220,"date":"2024-08-06T19:04:29","date_gmt":"2024-08-06T19:04:29","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=7220"},"modified":"2024-08-06T19:04:29","modified_gmt":"2024-08-06T19:04:29","slug":"chinese-medicine-component-compatibility","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/da\/chinese-medicine-component-compatibility\/","title":{"rendered":"Udforskning af mekanismen for traditionel kinesisk medicins komponentkompatibilitet til forebyggelse og behandling af kronisk hjertesvigt baseret p\u00e5 netv\u00e6rksfarmakologi og eksperimentel validering for at n\u00e6re Qi, varme Yang, fremme blodcirkulationen og gavne vand"},"content":{"rendered":"<p>Udforskning af mekanismen for traditionel kinesisk medicins komponentkompatibilitet til forebyggelse og behandling af kronisk hjertesvigt baseret p\u00e5 netv\u00e6rksfarmakologi og eksperimentel validering for at n\u00e6re Qi, varme Yang, fremme blodcirkulationen og gavne vand<br \/>\nKronisk hjertesvigt (CHF) er et klinisk symptom for\u00e5rsaget af hjerteinsufficiens, n\u00e5r forskellige hjertesygdomme udvikler sig til det terminale stadie. De vigtigste kliniske manifestationer af CHF er v\u00e6skeretention, dyspn\u00f8 og h\u00e6velser i ansigtet. Sygdommen er progressiv med d\u00e5rlig prognose og h\u00f8j d\u00f8delighed, hvilket udg\u00f8r en alvorlig trussel mod menneskers livssikkerhed. Kronisk hjertesvigt er mere skadeligt for menneskers liv end tumorer, og diagnosticering og behandling af sygdommen er blevet et vigtigt emne for det medicinske samfund i det 21. \u00e5rhundrede. Med den hurtige udvikling af traditionel kinesisk medicin har forst\u00e5elsen af hjerte-kar-sygdomme n\u00e5et et nyt niveau. Recepternes kompatibilitet er en specifik manifestation af traditionel kinesisk medicins syndromdifferentiering og -behandling, som har unikke fordele i behandlingen. At forst\u00e5 den dybe videnskabelige konnotation af kompatibilitet er et problem, der skal l\u00f8ses p\u00e5 nuv\u00e6rende tidspunkt.<br \/>\nAkademiker Zhang Boli og hans ekspertteam har for f\u00f8rste gang klart foresl\u00e5et det teoretiske koncept for effektiv kompatibilitet af kinesiske medicinkomponenter ved at bruge metoder som biologisk kromatografi, netv\u00e6rksfarmakologi og polar segmenteringsscreening til at screene kinesiske medicinkomponenter. Den videnskabelige og reproducerbare kompatibilitet af kinesiske medicinkomponenter er dens fordel. Netv\u00e6rksfarmakologi bruger hovedsageligt netv\u00e6rket til at screene specifikke signalknudepunkter, der har en f\u00e6lles forbindelse mellem l\u00e6gemiddelaktive ingredienser og relaterede sygdomme, for at analysere og finde ud af, om l\u00e6gemiddelingredienser har terapeutiske virkninger p\u00e5 relaterede sygdomme og specifikke signalveje. Samtidig svarer de holistiske egenskaber ved netv\u00e6rksfarmakologi til det holistiske koncept for traditionel kinesisk medicin, hvilket ogs\u00e5 afspejler dets fordele inden for traditionel kinesisk medicin.<br \/>\nDenne unders\u00f8gelse screenede de aktive ingredienser i fire l\u00e6gemiddelkomponenter, herunder totale saponiner af Astragalus membranaceus, totale phenolsyrer af Salvia miltiorrhiza, vandekstrakt af Scutellaria baicalensis og cinnamaldehyd. M\u00e5lene for de aktive ingredienser, der interagerer med relaterede sygdomme, blev identificeret, og den mulige virkningsmekanisme for komponenter i traditionel kinesisk medicin til behandling af hjertesvigt blev afsl\u00f8ret gennem molekyl\u00e6r docking og eksperimentel verifikation.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7221\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-289.png\" alt=\"\" width=\"786\" height=\"235\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-289.png 786w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-289-768x230.png 768w\" sizes=\"(max-width: 786px) 100vw, 786px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7222\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-241.png\" alt=\"\" width=\"785\" height=\"196\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-241.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-241-768x192.png 768w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7223\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-227.png\" alt=\"\" width=\"784\" height=\"331\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-227.png 784w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-227-768x324.png 768w\" sizes=\"(max-width: 784px) 100vw, 784px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7224\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-205.png\" alt=\"\" width=\"785\" height=\"896\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-205.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-205-768x877.png 768w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-205-631x720.png 631w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7225\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-185.png\" alt=\"\" width=\"778\" height=\"305\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-185.png 778w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-185-768x301.png 768w\" sizes=\"(max-width: 778px) 100vw, 778px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7226\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-169.png\" alt=\"\" width=\"788\" height=\"585\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-169.png 788w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-169-768x570.png 768w\" sizes=\"(max-width: 788px) 100vw, 788px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7227\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-154.png\" alt=\"\" width=\"785\" height=\"869\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-154.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-154-768x850.png 768w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-154-650x720.png 650w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7228\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-139.png\" alt=\"\" width=\"784\" height=\"909\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-139.png 784w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-139-768x890.png 768w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-139-621x720.png 621w\" sizes=\"(max-width: 784px) 100vw, 784px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7229\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-131.png\" alt=\"\" width=\"776\" height=\"623\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-131.png 776w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-131-768x617.png 768w\" sizes=\"(max-width: 776px) 100vw, 776px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7230\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-103.png\" alt=\"\" width=\"782\" height=\"909\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-103.png 782w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-103-768x893.png 768w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-103-619x720.png 619w\" sizes=\"(max-width: 782px) 100vw, 782px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7231\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-98.png\" alt=\"\" width=\"782\" height=\"281\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-98.png 782w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-98-768x276.png 768w\" sizes=\"(max-width: 782px) 100vw, 782px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7232\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-82.png\" alt=\"\" width=\"781\" height=\"221\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-82.png 781w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-82-768x217.png 768w\" sizes=\"(max-width: 781px) 100vw, 781px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7233\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-69.png\" alt=\"\" width=\"784\" height=\"247\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-69.png 784w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-69-768x242.png 768w\" sizes=\"(max-width: 784px) 100vw, 784px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7234\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/14-53.png\" alt=\"\" width=\"785\" height=\"126\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/14-53.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/14-53-768x123.png 768w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7235\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/15-40.png\" alt=\"\" width=\"783\" height=\"87\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/15-40.png 783w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/15-40-768x85.png 768w\" sizes=\"(max-width: 783px) 100vw, 783px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7236\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/16-28.png\" alt=\"\" width=\"778\" height=\"493\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/16-28.png 778w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/16-28-768x487.png 768w\" sizes=\"(max-width: 778px) 100vw, 778px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7237\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/17-23.png\" alt=\"\" width=\"785\" height=\"390\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/17-23.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/17-23-768x382.png 768w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7238\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/18-16.png\" alt=\"\" width=\"784\" height=\"173\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/18-16.png 784w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/18-16-768x169.png 768w\" sizes=\"(max-width: 784px) 100vw, 784px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7239\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/19-13.png\" alt=\"\" width=\"783\" height=\"376\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/19-13.png 783w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/19-13-768x369.png 768w\" sizes=\"(max-width: 783px) 100vw, 783px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-7240\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/20-10.png\" alt=\"\" width=\"346\" height=\"220\" \/><br \/>\nCHF er ikke eksplicit n\u00e6vnt i klassisk kinesisk medicinsk litteratur. Baseret p\u00e5 dets kliniske manifestationer kan det klassificeres som \"hjerteobstruktion\", \"hjertebanken\", \"brystobstruktion\", \"hjertebanken\", \"\u00f8dem\" og andre sygdomssyndromer. I behandlingen af CHF kombinerer traditionel kinesisk medicin syndromdifferentiering og holistiske koncepter. \"Expert Consensus on Integrated Traditional Chinese and Western Medicine Diagnosis and Treatment of Chronic Heart Failure\" p\u00e5peger, at kernepatogenesen ved hjertesvigt er mangel, blodstase og vand. At supplere mangel og styrke fundamentet er n\u00f8glen til behandling af denne sygdom. P\u00e5 grundlag af supplering af mangel er det ogs\u00e5 vigtigt at fremme blodcirkulationen og fjerne stasis, fremme diurese og reducere h\u00e6velse. Derfor er det tilr\u00e5deligt at etablere behandlingsmetoden til toning af qi og opvarmning af yang, fremme af blodcirkulationen og fremme af diurese. Forskningsgruppens forel\u00f8bige forskning viste ogs\u00e5, at patogenesen af CHF er baseret p\u00e5 manglen p\u00e5 Zong Qi med blodstasis, slim uklarhed og vandretention som kriterier, som er syndromerne ved mangel i roden og overskud i overskuddet. Baseret p\u00e5 Mate-analyse er effektiviteten af tonificerende qi, opvarmning af yang, fremme af blodcirkulation og diureseformel til behandling af kronisk hjertesvigt blevet bekr\u00e6ftet. Forskning har vist, at klinisk modificerede formler med virkningerne af tonifying qi, opvarmning af yang, fremme af blodcirkulationen og fremme af diurese har vist sig at have en god terapeutisk effekt p\u00e5 patienter med kronisk hjertesvigt og diuretisk resistens. De kan effektivt forbedre patienternes hjertefunktion og tyder p\u00e5, at de kan forbedre patienternes prognose.<br \/>\nDe fire komponenter, der er opn\u00e5et gennem screening, nemlig totale saponiner af Astragalus membranaceus, totale phenolsyrer af Salvia miltiorrhiza, vandekstrakt af Scutellaria baicalensis og cinnamaldehyd, er repr\u00e6sentative l\u00e6gemidler til at n\u00e6re qi, opvarme yang, fremme blodcirkulationen og gavne vand. Moderne farmakologiske unders\u00f8gelser har ogs\u00e5 vist, at totale saponiner af Astragalus membranaceus kan h\u00e6mme ventrikul\u00e6r remodellering og forbedre hjertefunktionen hos CHF-rotter, og dens virkningsstyrke er dosisafh\u00e6ngig; Danshen total phenolsyre kan forbedre intracellul\u00e6r calciumcirkulation og forbedre myokardial diastolisk og systolisk funktion. Vandekstraktet af Platycodon grandiflorus kan ud\u00f8ve virkninger mod hjertesvigt ved at \u00e6ndre de metaboliske forstyrrelser hos rotter med hjertesvigt. Cinnamaldehyd kan effektivt forbedre rottehjertefunktionen, h\u00e6mme frigivelsen af inflammatoriske faktorer og dermed ud\u00f8ve en beskyttende virkning p\u00e5 hjertet.<br \/>\nDenne unders\u00f8gelse viste, at de fire komponentm\u00e5l med h\u00f8j grad af krydsning med sygdomsm\u00e5l er AKT1, TNF, PPAR, CASP3, BCL2L1, HIF1A, MTOR, IL6 osv. Forskning har vist, at AKT opn\u00e5r signalregulering ved at h\u00e6mme pro-apoptotiske proteiner eller transkriptionsfaktorer og derved reducere kardiomyocyt-apoptose. Aktivering af AKT i myokardieceller kan h\u00e6mme celleapoptose, lindre myokardieinfarkt efter I\/R-skade og beskytte hjertefunktionen. Samtidig deltager AKT1 i processer som celleapoptose og ventrikul\u00e6r remodellering ved at regulere n\u00f8gleekspressionen af transformerende v\u00e6kstfaktor - \u03b2 (TGF - \u03b2 1). AKT regulerer myokardiecelleapoptose og spiller en rolle i at reducere inflammation ved at aktivere AKT\/mTOR-stien. De klassiske apoptosefaktorer Bcl-2 og Caspase-3 er downstream-faktorer for AKT\/mTOR. Forskning har vist, at NFkB kan aktiveres i de tidlige stadier af myokardieskade og fremkalde ekspression af kemokiner og adh\u00e6sionsmolekyler, hvilket f\u00f8rer til myokardieinflammation og -skade.<br \/>\nHuangqis samlede saponiner er hovedsageligt beriget i calciumsignalvejen, cGMPPKG, PI3K Akt, cAMP-signalvejen osv. Tidligere eksperimenter har vist, at totale saponiner af Astragalus membranaceus kan lindre oxidativ stress i rotte myokardium, h\u00e6mme kardiomyocytapoptose og forbedre hjertefunktionen ved at regulere AKL \/ p38MAPK-vejen. Huangqi IV-glykosid kan h\u00e6mme blodpladeaggregering og spille en rolle i forebyggelsen af vaskul\u00e6r restenose, hvilket yderligere tyder p\u00e5, at det traditionelle kinesiske medicinprincip om \"qi-cirkulation f\u00f8rer til blodcirkulation\" er rimeligt. Danshens samlede phenolsyrer er hovedsageligt beriget i PI3K Akt-signalvejen, og unders\u00f8gelser har vist, at Danshen phenolic acid A lindrer lipopolysaccharid-induceret apoptose og oxidativ stress i H9c2-kardiomyocytter ved at aktivere AKT\/mTOR\/4EBP1-vejen. Vandekstraktet af Scutellaria baicalensis er beriget i MAPK-signalvejen, calciumsignalvejen osv. Unders\u00f8gelser har vist, at Scutellaria baicalensis-ekstrakt kan aktivere MAPK-signalvejen, h\u00e6mme celleapoptose og beskytte mod myokardieskade. Cinnamaldehyd er beriget med Toll-lignende receptorer, TNF-signalveje osv. Cinnamaldehyd kan reducere ROS-indholdet i myokardiev\u00e6v, lindre myokardiecelle-autofagi og beskytte myokardiet, hvilket delvist bekr\u00e6fter netv\u00e6rksforudsigelsesresultaterne i denne unders\u00f8gelse.<br \/>\nSammenfattende brugte denne unders\u00f8gelse netv\u00e6rksfarmakologiske metoder til at screene de aktive ingrediensm\u00e5l, der svarer til CHF-sygdom i Huangqi samlede saponiner, Danshen samlede fenoliske syrer, Tangzi vandekstrakt og cinnamaldehyd, og opn\u00e5ede krydsende m\u00e5l. M\u00e5lene med h\u00f8je v\u00e6rdier var AKT1, TNF, INS, IL1B, PTGS2, PPAR, CASP3, MTOR osv. De involverede n\u00f8gleveje er PI3K Akt, MAPK, Toll like receptor-signalvej, calciumsignalvej, cGMP PKG osv., som er relateret til flere biologiske processer s\u00e5som cellecyklus, apoptose, autofagi, oxidativ stress og inflammatorisk respons og er potentielle mekanismer til behandling af hjertesvigt. Denne unders\u00f8gelse brugte netv\u00e6rksfarmakologisk molekyl\u00e6r docking-teknologi til at forudsige det materielle grundlag og virkningsmekanismen for HGDT-komponenter i behandlingen af hjertesvigt og verificerede eksperimentelt netv\u00e6rksforudsigelsesresultaterne og lagde grunden til unders\u00f8gelsen af mekanismen for traditionelle kinesiske medicinkomponenter i behandlingen af hjertesvigt.<\/p>","protected":false},"excerpt":{"rendered":"<p>Exploring the Mechanism of Traditional Chinese Medicine Component Compatibility for the Prevention and Treatment of Chronic Heart Failure Based on Network Pharmacology and Experimental Validation to Nourish Qi, Warm Yang, Promote Blood Circulation and Benefit Water Chronic heart failure (CHF) is a clinical symptom caused by cardiac insufficiency when various heart diseases develop to the [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - 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