{"id":6820,"date":"2024-08-06T14:47:50","date_gmt":"2024-08-06T14:47:50","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=6820"},"modified":"2024-08-06T14:47:50","modified_gmt":"2024-08-06T14:47:50","slug":"corrugated-seeds","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/da\/corrugated-seeds\/","title":{"rendered":"Differentiel analyse af kemisk sammens\u00e6tning og verifikation af celleeksperimenter af b\u00f8lgepapfr\u00f8 og deres forfalskede produkter baseret p\u00e5 metabolomics"},"content":{"rendered":"<p>Differentiel analyse af kemisk sammens\u00e6tning og verifikation af celleeksperimenter af b\u00f8lgepapfr\u00f8 og deres forfalskede produkter baseret p\u00e5 metabolomics<br \/>\nKorrugerede muslinger er skaller af Arca subcrinata Lischke, Arca granosa Linnaeus eller Arca inflata Reeve, som tilh\u00f8rer muslingefamilien. De bruges ofte i traditionel kinesisk medicin til marine skaldyr og har den virkning, at de reducerer slim, fjerner blodstasis, bl\u00f8dg\u00f8r h\u00e5rdhed, spreder klumper og lindrer syre og smerte. B\u00f8lgede sten bruges i vid udstr\u00e6kning i klinisk praksis til behandling af mavesygdomme som gastro\u00f8sofageal refluks, akutte maves\u00e5r, kronisk gastritis og maves\u00e5r; Og behandling af kr\u00e6ft i skjoldbruskkirtlen, skjoldbruskkirtelknuder, tumorer, ulcer\u00f8s colitis, hypertension og andre sygdomme.<br \/>\nB\u00f8lgede muslinger er en r\u00e6kke originale medicinske urter, og der er ogs\u00e5 mange forfalskede produkter, hovedsageligt inklusive ribbede, ru dekorerede muslinger, knudemuslinger, b\u00e5dmuslinger, kuglemuslinger og beh\u00e5rede muslinger. Ligesom andre skaldyr i traditionel kinesisk medicin best\u00e5r den kemiske sammens\u00e6tning af b\u00f8lgede fr\u00f8 af to hovedkategorier: uorganiske og organiske komponenter. De vigtigste uorganiske komponenter er uorganiske salte, der hovedsageligt best\u00e5r af calciumcarbonat og uorganiske sporstoffer. If\u00f8lge 2020-udgaven af Pharmacopoeia of the People's Republic of China b\u00f8r indholdet af calciumcarbonat (CaCO3) ikke v\u00e6re mindre end 93,0%. Hovedkomponenterne i organisk materiale er proteiner, aminosyrer, polysaccharider osv. Organiske komponenter udg\u00f8r generelt ca. 0,3% til 5,0% af skallens t\u00f8rv\u00e6gt. P\u00e5 grund af det lave organiske indhold og den komplekse struktur samt begr\u00e6nsninger i forskningsmetoder og ideer er den overordnede farmakologiske stofbasisforskning af skaldyrs traditionelle kinesiske medicin relativt svag, hvilket resulterer i en mangel p\u00e5 specialiserede identifikations- og bestemmelsesmetoder for indholdet af funktionelle komponenter i de nuv\u00e6rende kvalitetsstandarder for skaldyrs traditionelle kinesiske medicin, hvilket g\u00f8r det vanskeligt at evaluere dens iboende kvalitet. Systematisk identifikation og analyse af de organiske komponenter ved hj\u00e6lp af moderne forskningsmetoder er en foruds\u00e6tning og et fundament for at belyse det materielle grundlag og forbedre kvalitetsstandarderne. Denne unders\u00f8gelse benyttede TM Wide Targeted Metabolomics-teknikken, som integrerer fordelene ved ikke-m\u00e5lrettede (quad bar time-of-flight massespektrometri, QTOF) og bredt m\u00e5lrettede metabolitdetektionsteknikker (kvantitativ multipel reaktionsoverv\u00e5gning, MRM). Denne teknik kombinerer non target (h\u00f8j opl\u00f8sning, bred d\u00e6kning) med wide target (h\u00f8j f\u00f8lsomhed, pr\u00e6cis kvantificering), hvilket g\u00f8r den velegnet til analyse af komplekse pr\u00f8ver. Identifikation af traditionelle kinesiske medicinsorter er n\u00f8glen til kvalitetskontrol af traditionel kinesisk medicin. Metabolomics-teknologi kan anvendes til kvalitetskontrol af traditionel kinesisk medicin med lignende metaboliske oplysninger. I de senere \u00e5r er metabolomics-teknologi blevet brugt i vid udstr\u00e6kning i sammenlignende unders\u00f8gelser af traditionel kinesisk medicinkvalitet. I denne unders\u00f8gelse blev wide target-teknologi derfor brugt til omfattende at analysere de metaboliske komponenter i b\u00f8lgede muslinger og deres forfalskede produkter, s\u00e5som den tykke ribbede musling, for at identificere deres differentierede metabolitter og s\u00f8ge efter potentielle kvalitetsmark\u00f8rer. Forskning har vist, at b\u00f8lgede sten har en betydelig terapeutisk effekt p\u00e5 kr\u00e6ft i skjoldbruskkirtlen. Denne unders\u00f8gelse valgte den humane skjoldbruskkirtelkr\u00e6ftcellelinje TPC-1, som er relateret til dens traditionelle effektivitet, for at unders\u00f8ge de farmakologiske virkninger af nogle differentierede metabolitter og l\u00e6gge grunden til forbedring af det farmakologiske stofgrundlag og kvalitetsstandarder for b\u00f8lgepapfr\u00f8.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6821\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-31.jpg\" alt=\"\" width=\"800\" height=\"277\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-31.jpg 800w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-31-768x266.jpg 768w\" sizes=\"(max-width: 800px) 100vw, 800px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6822\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-29.jpg\" alt=\"\" width=\"700\" height=\"277\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6823\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-20.jpg\" alt=\"\" width=\"700\" height=\"365\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6824\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-181.png\" alt=\"\" width=\"700\" height=\"702\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-181.png 700w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-181-200x200.png 200w\" sizes=\"(max-width: 700px) 100vw, 700px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6825\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-165.png\" alt=\"\" width=\"800\" height=\"606\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-165.png 800w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-165-768x582.png 768w\" sizes=\"(max-width: 800px) 100vw, 800px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6826\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-150.png\" alt=\"\" width=\"700\" height=\"308\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6827\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-137.png\" alt=\"\" width=\"700\" height=\"370\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6828\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-125.png\" alt=\"\" width=\"800\" height=\"460\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-125.png 800w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-125-768x442.png 768w\" sizes=\"(max-width: 800px) 100vw, 800px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6829\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-117.png\" alt=\"\" width=\"700\" height=\"270\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6830\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-8.jpg\" alt=\"\" width=\"800\" height=\"395\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-8.jpg 800w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-8-768x379.jpg 768w\" sizes=\"(max-width: 800px) 100vw, 800px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6831\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-4.jpg\" alt=\"\" width=\"800\" height=\"226\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-4.jpg 800w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-4-768x217.jpg 768w\" sizes=\"(max-width: 800px) 100vw, 800px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6832\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-70.png\" alt=\"\" width=\"800\" height=\"790\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-70.png 800w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-70-768x758.png 768w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-70-729x720.png 729w\" sizes=\"(max-width: 800px) 100vw, 800px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6833\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-59.png\" alt=\"\" width=\"800\" height=\"846\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-59.png 800w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-59-768x812.png 768w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-59-681x720.png 681w\" sizes=\"(max-width: 800px) 100vw, 800px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6834\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/14-45.png\" alt=\"\" width=\"700\" height=\"280\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6835\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/15-34.png\" alt=\"\" width=\"765\" height=\"362\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6836\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/16-26.png\" alt=\"\" width=\"789\" height=\"344\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/16-26.png 789w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/16-26-768x335.png 768w\" sizes=\"(max-width: 789px) 100vw, 789px\" \/><br \/>\nForskningen i det farmakologiske stofgrundlag og virkningsmekanismen for b\u00f8lgede fr\u00f8 er svag. I denne unders\u00f8gelse blev der for f\u00f8rste gang brugt wide target metabolomics-teknologi til omfattende at analysere de metaboliske komponenter i b\u00f8lgepapfr\u00f8 og deres forfalskede produkter, og i alt 1208 metabolitter fra 22 kategorier blev opdaget. Hovedsageligt inklusive aminosyrer og deres metabolitter, benzen og dets derivater, heterocykliske forbindelser, organiske syrer og deres derivater, aldehyder, ketoner, estere, nukleotider og deres metabolitter osv. er det materielle grundlag forel\u00f8bigt blevet belyst.<br \/>\nI den tidlige fase sammenlignede forskningsgruppen traditionelle indikatorer som calciumcarbonatindhold, Ca2+indhold i afkog, vandopl\u00f8seligt ekstraktindhold, pH-v\u00e6rdi af vandekstrakt og totalt aminosyreindhold i b\u00f8lgepapfr\u00f8 og deres blandede produkter, og resultaterne viste ingen signifikante forskelle; Differentiel termisk analyse, r\u00f8ntgendiffraktion og r\u00f8ntgenfluorescens blev brugt til systematisk komparativ analyse, og resultaterne viste stadig ingen signifikante forskelle. Denne unders\u00f8gelse analyserede de metaboliske komponenter i sine autentiske og forfalskede produkter, herunder i alt 1083 metaboliske komponenter og 167 differentielle metabolitter, hvilket indikerer, at de organiske komponenter i hver pr\u00f8ve var de samme, men der var ogs\u00e5 forskelle. PCA og clustering heatmaps viste, at de tre autentiske originale pr\u00f8ver kunne grupperes sammen, mens de forfalskede produkter blev grupperet separat, hvilket indikerer, at den brede m\u00e5lmetaboliske analysemetode har god referencev\u00e6rdi til identifikation af autentiske og forfalskede skaldyr i traditionel kinesisk medicin.<br \/>\nDette eksperiment p\u00e5viste 72 nukleotider og deres metabolitter, herunder N6 isopentenyl adenosin, adenosin osv. Nukleosidstoffer spiller en vigtig rolle for effekten af l\u00e6gemidler til dyr. Moderne forskning har vist, at nukleosidkomponenter har virkninger som afslappende glat bronkialmuskulatur, antihistaminer, antiastma, antibakteriel, antiblodpladeaggregering, beroligende centralnervesystem og antikonvulsivt middel. Blandt dem er N6 isopentenyl adenosin et potentielt nyt l\u00e6gemiddel mod kr\u00e6ft. Forskning har vist, at efter behandling med 10 \u03bc mol\/L N6-isopentenyladenosin h\u00e6mmes den klonogene aktivitet i 8 humane epiteliale kr\u00e6ftcellelinjer fuldst\u00e6ndigt. Adenosin kan h\u00e6mme spredningen af mavekr\u00e6ft MGC-803-celler og fremme apoptose, mens endoplasmatisk retikulumstress kan v\u00e6re involveret i adenosininduceret apoptose. Cellevalideringseksperimenter har vist, at N6-isopentenyladenosin kan fremme celleapoptose og h\u00e6mme celleproliferation ved at blokere cellecyklussen i S- og G2-faserne. Og N6-isopentenyladenosin er markant opreguleret i det autentiske produkt, hvilket forventes at fungere som en potentiel kvalitetsmark\u00f8r til at skelne mellem \u00e6gte og forfalskede b\u00f8lgepapprodukter. Det tyder p\u00e5, at nukleosidstoffer kan v\u00e6re en vigtig komponent i det farmakologiske stofgrundlag for \"at fordrive slim og fjerne blodstasis, bl\u00f8dg\u00f8re h\u00e5rdhed og sprede knuder\" i b\u00f8lgepapfr\u00f8.<br \/>\nDette eksperiment p\u00e5viste 237 aminosyrer og deres metabolitter, herunder 134 sm\u00e5 peptider, herunder 12 cykliske dipeptider (CDP'er). Moderne forskning har vist, at CDP'er har universel biologisk aktivitet og st\u00e6rke antitumoreffekter med h\u00e6mmende effekter p\u00e5 v\u00e6ksten af forskellige kr\u00e6ftceller. Eksperimenter med celleproliferation viste, at cyklisk tyrosin ikke havde nogen signifikant h\u00e6mmende effekt p\u00e5 proliferationen af TPC-1-celler, og der b\u00f8r foretages yderligere unders\u00f8gelser i fremtiden.<br \/>\nDer er 40 metabolitter i de autentiske produkter, men ikke i de forfalskede produkter. Blandt dem har \u00f8stradiolbenzoat en h\u00e6mmende effekt p\u00e5 forekomsten af brystkr\u00e6ft, og dens virkningsmekanisme er relateret til reguleringen af \u00f8strogenreceptoren ER \u03b1 og Er \u03b2. HC-toksin har en signifikant antiproliferationseffekt p\u00e5 humane brystkr\u00e6ftceller T47D. Farnesylthiosalicylsyre er en RAS- og mTOR-h\u00e6mmer (mammalian rapamycin target protein), som kan h\u00e6mme v\u00e6ksten og spredningen af tumorceller. Disse tre stoffer forventes at fungere som potentielle kvalitetsmark\u00f8rer for b\u00f8lgepapmaterialer.<br \/>\nP\u00e5 grund af det svage forskningsgrundlag for skaldyrs traditionelle kinesiske medicin og manglen p\u00e5 referencematerialer og databaser er den kvalitative analyse af dens stoffer vanskelig. Under den differentielle metabolitanalyse fandt man ud af, at nogle metabolitter, s\u00e5som ginkgolid og oxalsyre, hovedsageligt findes i planter. Der er behov for yderligere udforskning for at bestemme deres sande kilder. Efterf\u00f8lgende b\u00f8r de p\u00e5viste komponenter bekr\u00e6ftes med referencestandarder for at forbedre den kvalitative n\u00f8jagtighed.<\/p>","protected":false},"excerpt":{"rendered":"<p>Differential analysis of chemical composition and cell experiment verification of corrugated seeds and their counterfeit products based on metabolomics Corrugated clams are shells of the Arca subcrinata Lischke, Arca granosa Linnaeus, or Arca inflata Reeve, which belong to the family of clams. They are commonly used traditional Chinese medicine for marine shellfish and have the [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Differential analysis of chemical composition and cell experiment verification of corrugated seeds and their counterfeit products based on metabolomics - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/da\/corrugated-seeds\/\" \/>\n<meta property=\"og:locale\" content=\"da_DK\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Differential analysis of chemical composition and cell experiment verification of corrugated seeds and their counterfeit products based on metabolomics - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Differential analysis of chemical composition and cell experiment verification of corrugated seeds and their counterfeit products based on metabolomics Corrugated clams are shells of the Arca subcrinata Lischke, Arca granosa Linnaeus, or Arca inflata Reeve, which belong to the family of clams. 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