{"id":6642,"date":"2024-08-06T12:49:34","date_gmt":"2024-08-06T12:49:34","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=6642"},"modified":"2024-08-06T12:49:34","modified_gmt":"2024-08-06T12:49:34","slug":"primitive-leeches","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/da\/primitive-leeches\/","title":{"rendered":"Unders\u00f8gelse af kvaliteten af forskellige primitive igler og deres forvekslede produkter"},"content":{"rendered":"<p>Unders\u00f8gelse af kvaliteten af forskellige primitive igler og deres forvekslede produkter<br \/>\nI 2020-udgaven af Folkerepublikken Kinas farmakop\u00e9, i det f\u00f8lgende ben\u00e6vnt den kinesiske farmakop\u00e9, hedder det, at igler er den t\u00f8rrede helhed af iglefamiliens dyr, s\u00e5som iglen Whitman pigra Whitman, iglen Hirudo nipponica Whitman eller pilebladets igle Whitman acranulata Whitman. Dens smag er salt, bitter og flad; der er et lille giftstof, som h\u00f8rer til levermeridianen. Den har den funktion at bryde blod og fremme cirkulation, fjerne blodstasis og eliminere stagnation. Det bruges ofte til blodstasis og meridianobstruktion, behandling af masser, slagtilf\u00e6lde hemiplegi og fald og skader. Unders\u00f8gelser har vist, at de farmakologiske virkninger af igler hovedsageligt omfatter antikoagulation, antitrombotiske, antitumor-, hypolipidemiske og antiinflammatoriske virkninger og har meget brede kliniske anvendelser, herunder behandling af trombose, hyperlipid\u00e6mi, hypertension, diabetes, prostatitis, kr\u00e6ft, \u00e5reknuder, infertilitet, skrumpelever og andre sygdomme. Hovedkomponenterne i igler er makromolekyl\u00e6re forbindelser, der hovedsageligt indeholder proteiner og 17 typer aminosyrer, herunder 8 essentielle aminosyrer for menneskekroppen. Det hydrolyserede aminosyreindhold er s\u00e5 h\u00f8jt som 49,4%; Derudover indeholder det ogs\u00e5 forskellige stoffer som hirudin, heparin, histamin, hirudin, glycolipider, sphenoider, steroider og carboxylestere.<br \/>\nEn litteraturgennemgang har vist, at den nuv\u00e6rende forskning i igler fokuserer p\u00e5 antikoagulerende mekanismer og bestemmelse af aminosyrer, og at der er begr\u00e6nsede omfattende unders\u00f8gelser af kvaliteten af forskellige primitive igler og deres blandinger. Identifikationsunders\u00f8gelser mellem forskellige primitive igler og deres blandinger er for det meste baseret p\u00e5 tr\u00e6kidentifikation i henhold til 2020-udgaven af den kinesiske farmakop\u00e9. Markedet for igler er dyrt og kaotisk, og traditionel udseendeidentifikation alene kan ikke hurtigt og effektivt evaluere deres kvalitet. Desuden kan identifikation af udseende ikke anvendes p\u00e5 igleekstrakter og -pr\u00e6parater, hvilket har visse begr\u00e6nsninger. Derfor er det af stor betydning at etablere en hurtig, videnskabelig og effektiv evalueringsmetode. Denne unders\u00f8gelse brugte HPLC til at etablere det karakteristiske spektrum og metoden til indholdsbestemmelse af igler. Denne metode giver en omfattende evaluering af igler og deres blandingsprodukter og udg\u00f8r et videnskabeligt grundlag for kvalitetsevalueringen af igler og deres blandingsprodukter.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6643\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-245.png\" alt=\"\" width=\"789\" height=\"378\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-245.png 789w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-245-768x368.png 768w\" sizes=\"(max-width: 789px) 100vw, 789px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6644\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-205.png\" alt=\"\" width=\"784\" height=\"412\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-205.png 784w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-205-768x404.png 768w\" sizes=\"(max-width: 784px) 100vw, 784px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6645\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-192.png\" alt=\"\" width=\"787\" height=\"714\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-192.png 787w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-192-768x697.png 768w\" sizes=\"(max-width: 787px) 100vw, 787px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6646\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-18.jpg\" alt=\"\" width=\"687\" height=\"274\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6647\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-155.png\" alt=\"\" width=\"780\" height=\"266\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-155.png 780w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-155-768x262.png 768w\" sizes=\"(max-width: 780px) 100vw, 780px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6648\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-141.png\" alt=\"\" width=\"780\" height=\"253\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-141.png 780w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-141-768x249.png 768w\" sizes=\"(max-width: 780px) 100vw, 780px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6649\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-129.png\" alt=\"\" width=\"787\" height=\"297\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-129.png 787w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-129-768x290.png 768w\" sizes=\"(max-width: 787px) 100vw, 787px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6650\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-117.png\" alt=\"\" width=\"783\" height=\"311\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-117.png 783w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-117-768x305.png 768w\" sizes=\"(max-width: 783px) 100vw, 783px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6651\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-109.png\" alt=\"\" width=\"786\" height=\"257\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-109.png 786w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-109-768x251.png 768w\" sizes=\"(max-width: 786px) 100vw, 786px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6652\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-87.png\" alt=\"\" width=\"783\" height=\"199\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-87.png 783w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-87-768x195.png 768w\" sizes=\"(max-width: 783px) 100vw, 783px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6653\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-79.png\" alt=\"\" width=\"785\" height=\"503\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-79.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-79-768x492.png 768w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-6654\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-62.png\" alt=\"\" width=\"785\" height=\"178\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-62.png 785w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-62-768x174.png 768w\" sizes=\"(max-width: 785px) 100vw, 785px\" \/><br \/>\nOptimering af kromatografiske forhold. P\u00e5 grundlag af etableringen af et karakteristisk spektrum anvendte denne unders\u00f8gelse den samme metode til at bestemme indholdet af to karakteristiske komponenter af igle, igleamin C-carboxylderivat og igleamin B. En diodearray-detektor blev brugt til at udf\u00f8re fuld b\u00f8lgel\u00e6ngdescanning af testopl\u00f8sningen i b\u00f8lgel\u00e6ngdeomr\u00e5det 200-400 nm. Resultaterne viste, at de kromatografiske toppe for hver hovedkomponent havde st\u00e6rk UV-absorption ved 254 nm b\u00f8lgel\u00e6ngde. Derfor blev de samme betingelser brugt til at analysere det karakteristiske spektrum og indholdet af iglepr\u00f8ver.<br \/>\nAnalyse af funktionskortets resultater. Blodiglen er den t\u00f8rrede hele krop af et dyr i iglefamilien, iglen Whitmania pigra Whitman. Dens medicinske egenskaber er flade, spindelformede. 2020-udgaven af den kinesiske farmakop\u00e9 kontrollerer kun dens kvalitet gennem fugt, totalt askeindhold, surheds- og alkalinitetstest og antitrombinaktivitet og har endnu ikke foretaget differentieret karakterisering mellem forskellige substrater. I denne unders\u00f8gelse blev HPLC-karakteristika for hirudo med forskellig oprindelse og dens forfalskninger etableret. Gennem sammenligning af referencestoffer blev det bekr\u00e6ftet, at hirudo indeholder fem komponenter: uracil, hypoxanthin, xanthin, hirudin C-carboxylderivater, hirudin B. If\u00f8lge litteraturrapporter har de ovenn\u00e6vnte pteridinforbindelser lignende strukturer med l\u00e6gemidler mod blodpladeaggregering s\u00e5som clopidogrel, og det antages, at disse komponenter kan v\u00e6re de aktive komponenter i hirudo for at spille antiplatelet-aggregering. De farmakologiske virkninger af hirudo, der er rapporteret mere om, er hovedsageligt antikoagulerende, antitrombotiske og antiaterosklerotiske virkninger. Derudover er der antitumor-, antiinflammatoriske, antifibrose- og lipidemiske aktiviteter, som indikerer, at de udvalgte karakteristiske toppe i denne unders\u00f8gelse er relateret til Det er af stor betydning at afklare de funktionelle stoffer i igler, der spiller farmakologiske aktiviteter og fremmer den sekund\u00e6re forskning og udvikling af l\u00e6gemidler. Samtidig kan den etablerede metode identificere forskellige primitive igler og deres blandingsprodukter. Det n\u00e6ste skridt er at forts\u00e6tte forskningen i anvendelsen af denne metode i ekstrakter og pr\u00e6parater, hvilket giver reference til udvikling og anvendelse af medicinske materialer fra igler.<br \/>\nAnalyse af resultater af indholdsbestemmelse. Baseret p\u00e5 unders\u00f8gelsen af karakteristiske kort bestemte denne unders\u00f8gelse kvantitativt fem komponenter i igler, herunder tre nukleosidforbindelser, uracil, hypoxanthin og to sphenoidforbindelser, leechamin C-carboxylderivater og leechamin B. If\u00f8lge eksisterende litteraturrapporter kan nukleosidforbindelser og sphenoidforbindelser bruges som indikatorer for kvalitetsevaluering af igler. Fors\u00f8gsresultaterne viste, at der var visse forskelle i indholdet af uracil og hypoxanthin blandt forskellige primitive igler og deres blandinger. Det gennemsnitlige indhold af uracil og hypoxanthin var i f\u00f8lgende r\u00e6kkef\u00f8lge: igle &gt; blodigle &gt; pileblad &gt; philippinsk igle; det gennemsnitlige indhold af xanthin er som f\u00f8lger: igle&gt;leech&gt;filippinsk igle&gt;pilblad igle; Det gennemsnitlige indhold af C-carboxylderivater af igleamin er som f\u00f8lger: blad igle&gt;leech&gt;leech&gt;filippinsk igle; Det gennemsnitlige indhold af igleamin B er som f\u00f8lger: blad igle&gt;leech&gt;leech&gt;filippinsk igle. Den filippinske igle indeholder ikke igleamin B, og indholdet af hypoxanthin er betydeligt lavere end de tre andre substrater. Derfor kan bestemmelse af indholdet af ovenn\u00e6vnte komponenter bruges til at skelne mellem vandblodigler (inklusive igler, igler og bladblodigler) og medicinske igler (filippinske igler); Derudover bruger PLS-DA-analyse topomr\u00e5derne af 8 karakteristiske toppe i pr\u00f8ven som variabler, og topomr\u00e5derne af karakteristiske toppe er t\u00e6t forbundet med indholdet af deres tilsvarende indikatorkomponenter. Kombineret med PLS-DA-analyseresultaterne i \"2.4.5\" er VIP-v\u00e6rdierne for de karakteristiske toppe, der svarer til hypoxanthin og xanthin, st\u00f8rre end 1, og pilebladet igle indeholder ikke xanthin. Det gennemsnitlige indhold af de tre andre primitive xanthiner viser ogs\u00e5 betydelige forskelle, hvilket yderligere indikerer, at valget af disse fem komponenter som indikatorer for indholdsbestemmelse har en vis videnskabelig validitet.<br \/>\nDen metode, som vores forskningsinstitut har etableret, er n\u00f8jagtig, f\u00f8lsom og har god specificitet. Den kan samtidig analysere de karakteristiske spektre og evaluere indholdet af medicinske iglematerialer. Den kan bruges som en kvalitetsevalueringsmetode for forskellige primitive igler og deres blandinger, hvilket giver en reference til kvalitetsevalueringen af medicinske iglematerialer.<\/p>","protected":false},"excerpt":{"rendered":"<p>Study on the Quality of Different Primitive Leeches and Their Confused Products The 2020 edition of the Pharmacopoeia of the People&#8217;s Republic of China, hereinafter referred to as the Chinese Pharmacopoeia, stipulates that leeches are the dried whole of the leech family animals, such as the leech Whitman pigra Whitman, leech Hirudo nipponica Whitman, or [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Study on the Quality of Different Primitive Leeches and Their Confused Products - 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