{"id":4588,"date":"2024-08-04T14:55:47","date_gmt":"2024-08-04T14:55:47","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=4588"},"modified":"2024-08-04T14:55:47","modified_gmt":"2024-08-04T14:55:47","slug":"bairui-granules","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/da\/bairui-granules\/","title":{"rendered":"Unders\u00f8gelse af blodkomponenterne i Bai Rui-granulat baseret p\u00e5 UHPLC-Q-TOF-MS\/MS-teknologi"},"content":{"rendered":"<p>Unders\u00f8gelse af blodkomponenterne i Bai Rui-granulat baseret p\u00e5 UHPLC-Q-TOF-MS\/MS-teknologi<\/p>\n<p>Unders\u00f8gelse af blodkomponenterne i Bai Rui-granulat baseret p\u00e5 UHPLC-Q-TOF-MS\/MS-teknologi<br \/>\nBairui-granulat er et granulatpr\u00e6parat, der best\u00e5r af en enkelt urt, Bairui-gr\u00e6s, som virker antibakteriel og antiinflammatorisk, fjerner varme og afgiftende og lindrer hoste. De bruges ofte i moderne klinisk praksis til at behandle p\u00e6diatrisk tonsillitis, bronkitis og forskellige luftvejsinfektioner. De aktive ingredienser i traditionel kinesisk medicin transporteres for det meste til m\u00e5let gennem blod som et medium (undtagen direkte virkning i tarmen og ekstern medicinering) for at ud\u00f8ve deres virkning. Derfor er det meget vigtigt at analysere de aktive ingredienser i kroppen efter oral indtagelse af traditionel kinesisk medicin for at unders\u00f8ge det materielle grundlag for effekten af traditionel kinesisk medicin. Vores forskningsgruppe har tidligere brugt v\u00e6skekromatografi-massespektrometri-teknologi til systematisk at analysere den kemiske sammens\u00e6tning af alkoholekstraktet af Atractylodes macrocephala og fundet ud af, at der er mange effektive ingredienser i Atractylodes macrocephala, s\u00e5som flavonoider, alkaloider og andre forbindelser. Tidligere litteraturstudier har for det meste fokuseret p\u00e5 den kemiske sammens\u00e6tning og kvalitetskontrol af enkelte urter, der mangler forskning i blodkomponenter og metaboliske processer i Atractylodes macrocephala-granulat in vivo, og det farmakologiske stofgrundlag er endnu ikke klart.<\/p>\n<p>Quadrupol-time-of-flight-massespektrometri-teknologien kan p\u00e5 grund af sin h\u00f8je f\u00f8lsomhed og opl\u00f8sning hurtigt og effektivt analysere de kemiske komponenter i traditionel kinesisk medicin og er blevet brugt i vid udstr\u00e6kning i forskningen af stofgrundlaget for traditionel kinesisk medicins effektivitet. P\u00e5 baggrund af tidligere forskning forts\u00e6tter vores forskningsgruppe derfor med at bruge UHPLC-Q-TOF-MS\/MS-teknologien (ultra high performance liquid chromatography quadrupole time of flight mass spectrometry) til at analysere de blodindg\u00e5ende komponenter og den metaboliske proces i Baisui Granule, hvilket giver et referencegrundlag for den grundl\u00e6ggende forskning i effektive stoffer og er af stor betydning for kvalitetskontrollen og udviklingen og anvendelsen af traditionelle kinesiske patentl\u00e6gemidler og enkle pr\u00e6parater.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4589\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-74.png\" alt=\"\" width=\"604\" height=\"791\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-74.png 604w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-74-550x720.png 550w\" sizes=\"(max-width: 604px) 100vw, 604px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4590\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-64.png\" alt=\"\" width=\"601\" height=\"515\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4591\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-2.jpg\" alt=\"\" width=\"601\" height=\"286\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4592\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-6.jpg\" alt=\"\" width=\"601\" height=\"281\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4593\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-49.png\" alt=\"\" width=\"601\" height=\"462\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4594\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-45.png\" alt=\"\" width=\"601\" height=\"661\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4595\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-2.jpg\" alt=\"\" width=\"600\" height=\"651\" \/><br \/>\nDenne unders\u00f8gelse brugte UHPLC-Q-TOF-MS\/MS-teknologi til at analysere de absorberede blodkomponenter i Bairui-granulat. I alt 20 prototypekomponenter og 10 metabolitter blev p\u00e5vist fra rotteserum. De vigtigste komponenter, der analyseres i kroppen, er alkaloider som quercetin og sophocarpine samt flavonoider som kaempferol og resveratrol I; De vigtigste metaboliske produkter i kroppen er oxidation og glucuronidation af kaempferol og oxidation og hydrolyse af sophocarpine, hvilket indikerer, at alkaloider og flavonoider er de vigtigste komponenter, der kommer ind i kroppen og ogs\u00e5 kan v\u00e6re potentielle aktive ingredienser til l\u00e6gemiddeleffektivitet.<\/p>\n<p>Moderne farmakologisk forskning har vist, at flavonoider og alkaloider har farmakologiske funktioner som antiinflammatoriske, antibakterielle, antivirale og antioxidanter. Tidligere unders\u00f8gelser har rapporteret, at den antiinflammatoriske virkning af resveratrolderivater i Bai Rui Cao er relateret til deres effektive h\u00e6mning af intracellul\u00e6r produktion af reaktive oxygenarter og aktivering af p38 MAPK og aktivatorprotein 1. Som en naturlig flavonol har resveratrol en st\u00e6rk effekt i at h\u00e6mme inflammatorisk cellefunktion og undertrykke udtrykket af proinflammatoriske cytokiner og kemokiner. Bairuicao I kan h\u00e6mme udtrykket af inflammatoriske cytokiner TNF - \u03b1, IL-6, IL-1 \u03b2 osv. ved at virke p\u00e5 NF - \u03ba B- og MAPK-vejene og derved forbedre lunge\u00f8dem hos mus, der er inficeret med lungebet\u00e6ndelse. Alkaloider kan h\u00e6mme v\u00e6ksten af mikroorganismer som Escherichia coli og Staphylococcus aureus betydeligt. Sophocarpine har st\u00e6rke antiinflammatoriske og smertestillende virkninger og kan reducere inflammation ved at h\u00e6mme NF - \u03ba B-signalvejen. Oxymatrin kan ud\u00f8ve antiinflammatoriske virkninger ved at h\u00e6mme NF-\u03ba B-signalvejen og reducere udtrykket af de inflammatoriske faktorer IL-6 og IL-8.<\/p>\n<p>Sammenfattende belyste denne unders\u00f8gelse blodkomponenterne og metabolitterne i Bairui-granulat ved hj\u00e6lp af UHPLC-Q-TOFMS\/MS-teknologi. Disse forbindelser kan v\u00e6re t\u00e6t forbundet med de antiinflammatoriske og antibakterielle virkninger af Bairui-granulat, hvilket er af stor betydning for at afklare det materielle grundlag for traditionel kinesisk medicins effektivitet og forbedre kvalitetsstandarderne for traditionel kinesisk medicin. Det giver et referencegrundlag for yderligere forst\u00e5else af dets virkningsmekanisme og kliniske anvendelse.<\/p>","protected":false},"excerpt":{"rendered":"<p>Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology Bairui granules are a granular preparation composed of single herb Bairui grass, which has the effects of antibacterial and anti-inflammatory, clearing heat and detoxifying, and relieving cough. They are [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/da\/bairui-granules\/\" \/>\n<meta property=\"og:locale\" content=\"da_DK\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology Study on the Blood Components of Bai Rui Granules Based on UHPLC-Q-TOF-MS\/MS Technology Bairui granules are a granular preparation composed of single herb Bairui grass, which has the effects of antibacterial and anti-inflammatory, clearing heat and detoxifying, and relieving cough. 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