{"id":4566,"date":"2024-08-04T14:53:22","date_gmt":"2024-08-04T14:53:22","guid":{"rendered":"https:\/\/longchangextracts.com\/?p=4566"},"modified":"2024-08-04T14:53:22","modified_gmt":"2024-08-04T14:53:22","slug":"callicarpa-nudiflora","status":"publish","type":"post","link":"https:\/\/longchangextracts.com\/da\/callicarpa-nudiflora\/","title":{"rendered":"Udforskning af de aktive anti-H1N1-komponenter og -mekanismer i n\u00f8gne lilla perler baseret p\u00e5 UPLC-Q-Exactive-Orbitrap-MS, netv\u00e6rksfarmakologi og eksperimentel validering"},"content":{"rendered":"<p>Udforskning af de aktive anti-H1N1-komponenter og -mekanismer i n\u00f8gne lilla perler baseret p\u00e5 UPLC-Q-Exactive-Orbitrap-MS, netv\u00e6rksfarmakologi og eksperimentel validering<br \/>\nDen traditionelle kinesiske medicin, Callicarpa nudiflora Hook.&amp;Arn., er et t\u00f8rret blad af planten Callicarpa nudiflora Hook.&amp;Arn. i familien Verbenaceae. Naked Purple Beads distribueres hovedsageligt i Hainan, Guangxi, Guangdong og andre regioner, og det autentiske produktionsomr\u00e5de er Wuzhishan-distriktet i Hainan-provinsen. Naked Flower Purple Pearl er den eneste nyligt tilf\u00f8jede traditionelle kinesiske medicin i 2020-udgaven af Pharmacopoeia of the People's Republic of China. Dens ensidige pr\u00e6parater, Naked Flower Purple Pearl Tablets og Naked Flower Purple Pearl Capsules, bruges i vid udstr\u00e6kning til at behandle bl\u00f8dninger i luftvejene og ford\u00f8jelsessystemet og bakteriel infekti\u00f8s inflammation for\u00e5rsaget af overdreven blodvarme og toksicitet. Fytokemikere har identificeret over 300 forbindelser fra n\u00f8gne lilla perler, herunder phenylpropanoider, flavonoider, triterpenoider, diterpener, iridoider, flygtige olier og meget mere. Moderne farmakologisk forskning har bekr\u00e6ftet, at den n\u00f8gne blomsterlilla perle har antiinflammatoriske, antitrombotiske, antitumorale, antibakterielle og hepatobeskyttende aktiviteter. I processen med at screene traditionel kinesisk medicin med antiviral aktivitet blev det konstateret, at ekstraktet af n\u00f8gen blomst lilla perle har god antiviral aktivitet (s\u00e5som H1N1 influenzavirus, enterovirus 71 osv.). Influenza A-virusinfektion er en almindelig \u00e5rsag til lungebet\u00e6ndelsesrelaterede d\u00f8dsfald. Alvorlig infektion med influenza A-virus kan for\u00e5rsage bilateral lungeinfiltration og hypox\u00e6mi, kendt som akut respiratorisk distress syndrom, som er en af de vigtigste d\u00f8ds\u00e5rsager for\u00e5rsaget af influenza A-virus. Dette eksperiment fokuserer p\u00e5 anti-H1N1-aktiviteten af den n\u00f8gne blomsterlilla perle. Den kemiske sammens\u00e6tning af de effektive dele af den n\u00f8gne blomsterlilla perle blev identificeret ved hj\u00e6lp af ultrah\u00f8jtydende v\u00e6skekromatografi quadrupol elektrostatisk felt orbitrap MS, og anti H1N1-mekanismen for den n\u00f8gne blomsterlilla perle blev forudsagt og eksperimentelt verificeret ved hj\u00e6lp af netv\u00e6rksfarmakologi. Virkningsmekanismen for den n\u00f8gne blomsterperle mod H1N1 blev forel\u00f8bigt udforsket.<\/p>\n<p><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4570\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/1-73.png\" alt=\"\" width=\"340\" height=\"709\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4571\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/2-63.png\" alt=\"\" width=\"340\" height=\"234\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4572\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/3-60.png\" alt=\"\" width=\"600\" height=\"621\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4573\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/4-50.png\" alt=\"\" width=\"600\" height=\"660\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4574\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-2.jpg\" alt=\"\" width=\"539\" height=\"748\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-2.jpg 539w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/5-2-519x720.jpg 519w\" sizes=\"(max-width: 539px) 100vw, 539px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4575\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/6-44.png\" alt=\"\" width=\"539\" height=\"272\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4576\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-42.png\" alt=\"\" width=\"600\" height=\"784\" srcset=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-42.png 600w, https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/7-42-551x720.png 551w\" sizes=\"(max-width: 600px) 100vw, 600px\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4577\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/8-36.png\" alt=\"\" width=\"600\" height=\"539\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4578\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/9-31.png\" alt=\"\" width=\"600\" height=\"304\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4579\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/10-27.png\" alt=\"\" width=\"600\" height=\"244\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4580\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/11-25.png\" alt=\"\" width=\"340\" height=\"219\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4581\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/12-21.png\" alt=\"\" width=\"340\" height=\"546\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4582\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/13-18.png\" alt=\"\" width=\"600\" height=\"271\" \/><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-4583\" src=\"https:\/\/longchangextracts.com\/wp-content\/uploads\/2024\/08\/14-15.png\" alt=\"\" width=\"600\" height=\"327\" \/>callicarpa nudiflora<br \/>\nInfluenza A-virus har udviklet varierende grader af resistens over for almindeligt anvendte M2-kanalh\u00e6mmere og NA-h\u00e6mmere. Derfor er det blevet et presserende problem at finde nye l\u00e6gemidler eller behandlingsmetoder mod influenza A. Traditionel kinesisk medicin har spillet en vigtig rolle i den kliniske behandling af influenza A-virus. Det holistiske koncept i traditionel kinesisk medicinteori regulerer systematisk patienter som en organisk helhed, mens netv\u00e6rksfarmakologi udforsker samspillet mellem de biologiske funktioner i hver node i netv\u00e6rket og sygdomme ved at konstruere et l\u00e6gemiddelkomponentm\u00e5lvejssygdomsnetv\u00e6rk, hvilket er i overensstemmelse med det holistiske koncept i traditionel kinesisk medicin. Dette eksperiment screenede f\u00f8rst de vigtigste anti-H1N1-aktive steder i den traditionelle kinesiske medicin Naked Flower Purple Pearl og analyserede stederne for at identificere 34 kemiske komponenter. Ved at kombinere litteratur og databaser blev der identificeret 67 overlappende m\u00e5l for l\u00e6gemidler og sygdomme. Gennem berigelsesanalyse af krydsende m\u00e5l spekulerer vi i, at den vigtige biologiske proces med EACN mod H1N1 kan v\u00e6re den positive regulering af proteinfosforylering og respons p\u00e5 oxidativ stress. Resultaterne af KEGG-berigelsesanalysen viste, at 19 forbindelser i EACN virker p\u00e5 influenza A-virusvejen gennem 11 m\u00e5l. L\u00e6gemidlet p\u00e5virker M2-kanalen i H1N1-virus ved at virke p\u00e5 PLG og PRSS1 og kan ogs\u00e5 p\u00e5virke virusfrigivelsesprocessen ved at virke p\u00e5 neuraminidase (NA)-vejen gennem PLG. PLG og PRSS1 kan v\u00e6re vigtige m\u00e5l for EACN, s\u00e5 de kan virke direkte p\u00e5 H1N1. EACN kan h\u00e6mme spredningen af H1N1 ved at p\u00e5virke dens udskillelses- og frig\u00f8relsesprocesser. I sygdomsnetv\u00e6rket for l\u00e6gemiddelingredienser er RELA og NF - \u03ba B1 de to m\u00e5l med de h\u00f8jeste gradv\u00e6rdier. NF-\u03ba B-signalvejen, hvor de er placeret, kan fremme udtrykket af faktorer som IL1 \u03b2, TNF - \u03b1, IL-6 og fremme inflammatorisk respons, hvilket tyder p\u00e5, at EACN kan virke p\u00e5 vigtige m\u00e5l som RELA og NF-\u03ba B1 for at regulere NF-\u03ba B-signalvejen og reducere bet\u00e6ndelsesskader i kroppen. I henhold til de resultater, der forudsiges af netv\u00e6rksfarmakologi, kan EACN regulere T-cellesignalveje, p\u00e5virke Th1- og Th2-differentiering og ud\u00f8ve immunregulerende virkninger. Derfor udf\u00f8rte denne unders\u00f8gelse dyrefors\u00f8g for at verificere den h\u00e6mmende effekt, den antiinflammatoriske effekt og den immunregulerende effekt af EACN p\u00e5 H1N1-spredning. Fors\u00f8gsresultaterne viste, at EACN kan forbedre v\u00e6gttabet og stigningen i lungeindekset for\u00e5rsaget af H1N1-infektion, reducere den virale belastning i musens lungev\u00e6v, lindre patologiske skader i musens lungev\u00e6v, s\u00e6nke niveauerne af TNF - \u03b1, IFN - \u03b3, IL-1 \u03b2 i perifert blodserum og \u00f8ge niveauet af serumantistof IgG. Denne unders\u00f8gelse brugte f\u00f8rst in vitro-eksperimenter til at screene de aktive ekstraktionssteder i Naked Purple Pearl mod H1N1 og forudsagde de aktive ingredienser i EACN mod H1N1 ved hj\u00e6lp af UPLC-Q-Hexactive-Orbitrap-MS og netv\u00e6rksfarmakologi. De forudsagte resultater blev verificeret ved dyrefors\u00f8g, og potentielle aktive ingredienser i EACN mod H1N1 blev screenet, herunder quercetin, myricetin, luteolin, kaempferol, quercetin, apigenin og acacetin. Det blev forel\u00f8bigt p\u00e5vist, at Naked Purple Pearl kan ud\u00f8ve anti-H1N1-effekter gennem flere veje, s\u00e5som direkte virusinhibering, antiinflammatoriske effekter og immunregulering. I efterf\u00f8lgende eksperimenter er det n\u00f8dvendigt at udf\u00f8re in vitro- og in vivo-eksperimenter for at validere de udvalgte monomere forbindelser og yderligere unders\u00f8ge mekanismen for EACN's anti-H1N1-effekt p\u00e5 mRNA- og proteinniveau.<\/p>","protected":false},"excerpt":{"rendered":"<p>Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation The traditional Chinese medicine, Callicarpa nudiflora Hook.&amp;Arn., is a dried leaf of the plant Callicarpa nudiflora Hook.&amp;Arn. in the family Verbenaceae. Naked Purple Beads are mainly distributed in Hainan, Guangxi, Guangdong and other regions, with [&hellip;]<\/p>","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[20],"tags":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v23.0 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation - China Chemical Manufacturer<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/longchangextracts.com\/da\/callicarpa-nudiflora\/\" \/>\n<meta property=\"og:locale\" content=\"da_DK\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation - China Chemical Manufacturer\" \/>\n<meta property=\"og:description\" content=\"Exploring the Anti H1N1 Active Components and Mechanisms of Naked Purple Beads Based on UPLC-Q-Exactive-Orbitrap-MS, Network Pharmacology, and Experimental Validation The traditional Chinese medicine, Callicarpa nudiflora Hook.&amp;Arn., is a dried leaf of the plant Callicarpa nudiflora Hook.&amp;Arn. in the family Verbenaceae. 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